MX2019002901A - Tratamiento de esclerosis multiple con chs-131. - Google Patents
Tratamiento de esclerosis multiple con chs-131.Info
- Publication number
- MX2019002901A MX2019002901A MX2019002901A MX2019002901A MX2019002901A MX 2019002901 A MX2019002901 A MX 2019002901A MX 2019002901 A MX2019002901 A MX 2019002901A MX 2019002901 A MX2019002901 A MX 2019002901A MX 2019002901 A MX2019002901 A MX 2019002901A
- Authority
- MX
- Mexico
- Prior art keywords
- chs
- treatment
- multiple sclerosis
- prodrug
- women
- Prior art date
Links
- 201000006417 multiple sclerosis Diseases 0.000 title abstract 3
- NMRWDFUZLLQSBN-UHFFFAOYSA-N 2,4-dichloro-n-(3,5-dichloro-4-quinolin-3-yloxyphenyl)benzenesulfonamide Chemical compound ClC1=CC(Cl)=CC=C1S(=O)(=O)NC(C=C1Cl)=CC(Cl)=C1OC1=CN=C(C=CC=C2)C2=C1 NMRWDFUZLLQSBN-UHFFFAOYSA-N 0.000 abstract 2
- 229940002612 prodrug Drugs 0.000 abstract 1
- 239000000651 prodrug Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Epidemiology (AREA)
- Immunology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662394046P | 2016-09-13 | 2016-09-13 | |
| US201662436356P | 2016-12-19 | 2016-12-19 | |
| US201762460868P | 2017-02-19 | 2017-02-19 | |
| US201762491071P | 2017-04-27 | 2017-04-27 | |
| PCT/US2017/051414 WO2018053040A1 (en) | 2016-09-13 | 2017-09-13 | Treatment of multiple sclerosis with chs-131 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2019002901A true MX2019002901A (es) | 2019-09-26 |
Family
ID=61619253
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2019002901A MX2019002901A (es) | 2016-09-13 | 2017-09-13 | Tratamiento de esclerosis multiple con chs-131. |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20190224186A1 (enExample) |
| EP (1) | EP3512512A4 (enExample) |
| JP (1) | JP2019531286A (enExample) |
| KR (1) | KR20190064583A (enExample) |
| CN (1) | CN110461318A (enExample) |
| AU (1) | AU2017326261A1 (enExample) |
| BR (1) | BR112019004791A2 (enExample) |
| CA (1) | CA3036694A1 (enExample) |
| IL (1) | IL265259A (enExample) |
| MX (1) | MX2019002901A (enExample) |
| SG (1) | SG10202102198RA (enExample) |
| WO (1) | WO2018053040A1 (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20130158077A1 (en) | 2011-12-19 | 2013-06-20 | Ares Trading S.A. | Pharmaceutical compositions |
| WO2016144862A1 (en) | 2015-03-09 | 2016-09-15 | Intekrin Therapeutics, Inc. | Methods for the treatment of nonalcoholic fatty liver disease and/or lipodystrophy |
| KR20200036808A (ko) | 2017-04-03 | 2020-04-07 | 코히러스 바이오사이언시스, 인크. | 진행성 핵상 마비 치료를 위한 PPARγ 작용제 |
| EA201992364A1 (ru) * | 2018-04-02 | 2020-03-23 | Кохерус Байосайенсис Инк. | АГОНИСТ PPARγ ДЛЯ ЛЕЧЕНИЯ ПРОГРЕССИРУЮЩЕГО НАДЪЯДЕРНОГО ПАРАЛИЧА |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7223761B2 (en) * | 2003-10-03 | 2007-05-29 | Amgen Inc. | Salts and polymorphs of a potent antidiabetic compound |
| EA201590726A1 (ru) * | 2012-10-12 | 2015-10-30 | Тева Фармасьютикал Индастриз Лтд. | Лахинимод для уменьшения таламического поражения при рассеянном склерозе |
| BR112015018048A2 (pt) * | 2013-01-30 | 2020-01-28 | Intekrin Therapeutics Inc | agonistas de ppary para tratamento de esclerose múltipla |
-
2017
- 2017-09-13 SG SG10202102198RA patent/SG10202102198RA/en unknown
- 2017-09-13 JP JP2019513922A patent/JP2019531286A/ja active Pending
- 2017-09-13 BR BR112019004791A patent/BR112019004791A2/pt not_active Application Discontinuation
- 2017-09-13 MX MX2019002901A patent/MX2019002901A/es unknown
- 2017-09-13 US US16/333,171 patent/US20190224186A1/en not_active Abandoned
- 2017-09-13 CA CA3036694A patent/CA3036694A1/en not_active Abandoned
- 2017-09-13 AU AU2017326261A patent/AU2017326261A1/en not_active Abandoned
- 2017-09-13 KR KR1020197009963A patent/KR20190064583A/ko not_active Ceased
- 2017-09-13 WO PCT/US2017/051414 patent/WO2018053040A1/en not_active Ceased
- 2017-09-13 CN CN201780069826.5A patent/CN110461318A/zh not_active Withdrawn
- 2017-09-13 EP EP17851479.0A patent/EP3512512A4/en not_active Withdrawn
-
2019
- 2019-03-10 IL IL265259A patent/IL265259A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN110461318A (zh) | 2019-11-15 |
| IL265259A (en) | 2019-05-30 |
| EP3512512A1 (en) | 2019-07-24 |
| WO2018053040A1 (en) | 2018-03-22 |
| BR112019004791A2 (pt) | 2019-06-04 |
| CA3036694A1 (en) | 2018-03-22 |
| EP3512512A4 (en) | 2020-06-03 |
| AU2017326261A1 (en) | 2019-04-04 |
| SG10202102198RA (en) | 2021-04-29 |
| JP2019531286A (ja) | 2019-10-31 |
| US20190224186A1 (en) | 2019-07-25 |
| KR20190064583A (ko) | 2019-06-10 |
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