MX2016001302A - Compuesto y metodos para tratar el sindrome de qt largo. - Google Patents

Compuesto y metodos para tratar el sindrome de qt largo.

Info

Publication number
MX2016001302A
MX2016001302A MX2016001302A MX2016001302A MX2016001302A MX 2016001302 A MX2016001302 A MX 2016001302A MX 2016001302 A MX2016001302 A MX 2016001302A MX 2016001302 A MX2016001302 A MX 2016001302A MX 2016001302 A MX2016001302 A MX 2016001302A
Authority
MX
Mexico
Prior art keywords
syndrome
compound
methods
treating long
treating
Prior art date
Application number
MX2016001302A
Other languages
English (en)
Inventor
Luiz Belardinelli
Dewan Zeng
Sridharan Rajamani
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Publication of MX2016001302A publication Critical patent/MX2016001302A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/553Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Dermatology (AREA)

Abstract

Se describe en la presente un método para tratar el síndrome de QT largo por la administración de una cantidad eficaz de un bloqueador de canales iónicos de sodio tardíos potente y selectivo.
MX2016001302A 2013-08-01 2014-07-31 Compuesto y metodos para tratar el sindrome de qt largo. MX2016001302A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361861344P 2013-08-01 2013-08-01
US201361900235P 2013-11-05 2013-11-05
PCT/US2014/049155 WO2015017661A1 (en) 2013-08-01 2014-07-31 Compound and methods for treating long qt syndrome

Publications (1)

Publication Number Publication Date
MX2016001302A true MX2016001302A (es) 2016-04-07

Family

ID=51352867

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016001302A MX2016001302A (es) 2013-08-01 2014-07-31 Compuesto y metodos para tratar el sindrome de qt largo.

Country Status (12)

Country Link
US (1) US9126989B2 (es)
EP (1) EP3027190A1 (es)
JP (1) JP2016525580A (es)
KR (1) KR20160035061A (es)
CN (1) CN105611931A (es)
AU (1) AU2014296145A1 (es)
CA (1) CA2919757A1 (es)
EA (1) EA201690215A1 (es)
HK (1) HK1219893A1 (es)
MX (1) MX2016001302A (es)
SG (1) SG11201600119PA (es)
WO (1) WO2015017661A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105497876B (zh) 2014-09-24 2021-01-15 上海泽生科技开发股份有限公司 神经调节蛋白用于预防、治疗或延迟心脏室性心律失常的方法和组合物
US10575744B2 (en) 2017-02-24 2020-03-03 Medtronic Cryocath Lp Pericardial balloon mapping

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030220344A1 (en) 2002-04-04 2003-11-27 Luiz Belardinelli Method of treating arrhythmias
TWI478908B (zh) 2011-07-01 2015-04-01 Gilead Sciences Inc 作為離子通道調節劑之稠合雜環化合物
WO2013112932A1 (en) * 2012-01-27 2013-08-01 Gilead Sciences, Inc. Combination therapies using late sodium ion channel blockers and potassium ion channel blockers

Also Published As

Publication number Publication date
EP3027190A1 (en) 2016-06-08
HK1219893A1 (zh) 2017-04-21
US9126989B2 (en) 2015-09-08
CA2919757A1 (en) 2015-02-05
EA201690215A1 (ru) 2016-07-29
JP2016525580A (ja) 2016-08-25
WO2015017661A1 (en) 2015-02-05
AU2014296145A1 (en) 2016-01-28
SG11201600119PA (en) 2016-02-26
KR20160035061A (ko) 2016-03-30
CN105611931A (zh) 2016-05-25
US20150038489A1 (en) 2015-02-05

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