MX2010011643A - Tiofencarboxamidas sustituidas como inhibidores de la proteina cinasa ikk-beta serina, treonina. - Google Patents
Tiofencarboxamidas sustituidas como inhibidores de la proteina cinasa ikk-beta serina, treonina.Info
- Publication number
- MX2010011643A MX2010011643A MX2010011643A MX2010011643A MX2010011643A MX 2010011643 A MX2010011643 A MX 2010011643A MX 2010011643 A MX2010011643 A MX 2010011643A MX 2010011643 A MX2010011643 A MX 2010011643A MX 2010011643 A MX2010011643 A MX 2010011643A
- Authority
- MX
- Mexico
- Prior art keywords
- radical
- compounds
- alkyl
- mmol
- intermediary
- Prior art date
Links
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Classifications
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- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0807642A GB0807642D0 (en) | 2008-04-26 | 2008-04-26 | IKK- serine-threonine protein kinase inhibitors |
| GB0815550A GB0815550D0 (en) | 2008-08-27 | 2008-08-27 | IKK-beta serine-threonine protein kinase inhibitors |
| PCT/GB2009/001051 WO2009130475A1 (en) | 2008-04-26 | 2009-04-23 | Substituted thiophenecarboxamides as ikk-beta serine-, threonine-protein kinase inhibitors |
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| MX2010011643A true MX2010011643A (es) | 2010-11-30 |
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| MX2010011643A MX2010011643A (es) | 2008-04-26 | 2009-04-23 | Tiofencarboxamidas sustituidas como inhibidores de la proteina cinasa ikk-beta serina, treonina. |
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| Country | Link |
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| US (1) | US20110046210A1 (enExample) |
| EP (1) | EP2285797A1 (enExample) |
| JP (1) | JP2011518817A (enExample) |
| KR (1) | KR20110020784A (enExample) |
| CN (1) | CN102036980A (enExample) |
| AU (1) | AU2009239772A1 (enExample) |
| BR (1) | BRPI0911480A2 (enExample) |
| CA (1) | CA2722660A1 (enExample) |
| EA (1) | EA201001708A1 (enExample) |
| IL (1) | IL208654A0 (enExample) |
| MX (1) | MX2010011643A (enExample) |
| WO (1) | WO2009130475A1 (enExample) |
| ZA (1) | ZA201008027B (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012046793A1 (ja) * | 2010-10-07 | 2012-04-12 | 参天製薬株式会社 | ウレイド基とアミノカルボニル基を置換基として有するチオフェン誘導体を有効成分として含有する新規ｊａｋ３阻害剤 |
| GB201211310D0 (en) | 2012-06-26 | 2012-08-08 | Chroma Therapeutics Ltd | CSF-1R kinase inhibitors |
| CA2888928C (en) | 2012-10-17 | 2020-05-26 | Chroma Therapeutics Ltd | Tert-butyl n-[2-{4-[6-amino-5-(2,4-difluorobenzoyl)-2-oxopyridin-1(2h)-yl]-3,5- difluorophenyl}ethyl]-l-alaninate or a salt, hydrate or solvate thereof |
| JP6321042B2 (ja) | 2013-02-06 | 2018-05-09 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | 新規なハロゲン置換された化合物 |
| GB201713975D0 (en) | 2017-08-31 | 2017-10-18 | Macrophage Pharma Ltd | Medical use |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0102616D0 (sv) * | 2001-07-25 | 2001-07-25 | Astrazeneca Ab | Novel compounds |
| SE0300092D0 (sv) * | 2003-01-15 | 2003-01-15 | Astrazeneca Ab | Novel compounds |
| WO2008002246A1 (en) * | 2006-06-28 | 2008-01-03 | Astrazeneca Ab | A pharmaceutical composition comprising an ikk2 inhibitor and a second active ingrdient. |
| AU2007315943A1 (en) * | 2006-11-01 | 2008-05-08 | Chroma Therapeutics Ltd. | IKK-beta serine-threonine protein kinase inhibitors |
| US8106091B2 (en) * | 2006-11-01 | 2012-01-31 | Chroma Therapeutics Ltd. | Inhibitors of IKK-beta serine-threonine protein kinase |
-
2009
- 2009-04-23 CN CN2009801189111A patent/CN102036980A/zh active Pending
- 2009-04-23 EP EP09733957A patent/EP2285797A1/en not_active Withdrawn
- 2009-04-23 JP JP2011505589A patent/JP2011518817A/ja not_active Withdrawn
- 2009-04-23 AU AU2009239772A patent/AU2009239772A1/en not_active Abandoned
- 2009-04-23 KR KR1020107026507A patent/KR20110020784A/ko not_active Withdrawn
- 2009-04-23 CA CA2722660A patent/CA2722660A1/en not_active Abandoned
- 2009-04-23 EA EA201001708A patent/EA201001708A1/ru unknown
- 2009-04-23 BR BRPI0911480A patent/BRPI0911480A2/pt not_active IP Right Cessation
- 2009-04-23 US US12/989,271 patent/US20110046210A1/en not_active Abandoned
- 2009-04-23 MX MX2010011643A patent/MX2010011643A/es not_active Application Discontinuation
- 2009-04-23 WO PCT/GB2009/001051 patent/WO2009130475A1/en not_active Ceased
-
2010
- 2010-10-12 IL IL208654A patent/IL208654A0/en unknown
- 2010-11-09 ZA ZA2010/08027A patent/ZA201008027B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2722660A1 (en) | 2009-10-29 |
| EA201001708A1 (ru) | 2011-06-30 |
| EP2285797A1 (en) | 2011-02-23 |
| BRPI0911480A2 (pt) | 2018-04-03 |
| WO2009130475A1 (en) | 2009-10-29 |
| CN102036980A (zh) | 2011-04-27 |
| KR20110020784A (ko) | 2011-03-03 |
| JP2011518817A (ja) | 2011-06-30 |
| IL208654A0 (en) | 2010-12-30 |
| AU2009239772A1 (en) | 2009-10-29 |
| ZA201008027B (en) | 2011-07-27 |
| US20110046210A1 (en) | 2011-02-24 |
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| Date | Code | Title | Description |
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| FA | Abandonment or withdrawal |