MX2010008718A - Piperidinas sustituidas como inhibidores de renina. - Google Patents
Piperidinas sustituidas como inhibidores de renina.Info
- Publication number
- MX2010008718A MX2010008718A MX2010008718A MX2010008718A MX2010008718A MX 2010008718 A MX2010008718 A MX 2010008718A MX 2010008718 A MX2010008718 A MX 2010008718A MX 2010008718 A MX2010008718 A MX 2010008718A MX 2010008718 A MX2010008718 A MX 2010008718A
- Authority
- MX
- Mexico
- Prior art keywords
- renin inhibitors
- substituted piperidines
- compounds
- salts
- piperidines
- Prior art date
Links
- 239000002461 renin inhibitor Substances 0.000 title abstract 2
- 229940086526 renin-inhibitors Drugs 0.000 title abstract 2
- 150000003053 piperidines Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 229940079593 drug Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Ophthalmology & Optometry (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
La presente invención se refiere a compuestos de la fórmula general (I) y sales de los mismos, preferentemente las sales farmacéuticamente aceptables de los mismos, en donde R tiene el significado explicado en la descripción, a un proceso para su preparación y al uso de estos compuestos como medicinas especialmente como inhibidores de renina.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP08101428 | 2008-02-08 | ||
| PCT/EP2009/051350 WO2009098276A1 (en) | 2008-02-08 | 2009-02-06 | Substituted piperidines as renin inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2010008718A true MX2010008718A (es) | 2010-09-24 |
Family
ID=40020274
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2010008718A MX2010008718A (es) | 2008-02-08 | 2009-02-06 | Piperidinas sustituidas como inhibidores de renina. |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US8022069B2 (es) |
| EP (1) | EP2250166A1 (es) |
| JP (1) | JP2011511039A (es) |
| KR (1) | KR20100131427A (es) |
| CN (1) | CN101939318A (es) |
| AU (1) | AU2009211378A1 (es) |
| BR (1) | BRPI0907933A2 (es) |
| CA (1) | CA2714350A1 (es) |
| EA (1) | EA201001239A1 (es) |
| MX (1) | MX2010008718A (es) |
| WO (1) | WO2009098276A1 (es) |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW200613274A (en) | 2004-07-09 | 2006-05-01 | Speedel Experimenta Ag | Organic compounds |
| JP2008535825A (ja) | 2005-03-31 | 2008-09-04 | シュペーデル・エクスペリメンタ・アーゲー | レニン阻害剤としての３，４，５−置換ピペリジン |
| TW200833687A (en) | 2005-03-31 | 2008-08-16 | Speedel Experimenta Ag | Substituted piperidines |
-
2009
- 2009-02-06 EP EP09709329A patent/EP2250166A1/en not_active Withdrawn
- 2009-02-06 WO PCT/EP2009/051350 patent/WO2009098276A1/en active Application Filing
- 2009-02-06 CA CA2714350A patent/CA2714350A1/en not_active Abandoned
- 2009-02-06 JP JP2010545472A patent/JP2011511039A/ja active Pending
- 2009-02-06 AU AU2009211378A patent/AU2009211378A1/en not_active Abandoned
- 2009-02-06 KR KR1020107017524A patent/KR20100131427A/ko not_active Application Discontinuation
- 2009-02-06 MX MX2010008718A patent/MX2010008718A/es not_active Application Discontinuation
- 2009-02-06 CN CN2009801044108A patent/CN101939318A/zh active Pending
- 2009-02-06 BR BRPI0907933-5A patent/BRPI0907933A2/pt not_active IP Right Cessation
- 2009-02-06 US US12/865,932 patent/US8022069B2/en not_active Expired - Fee Related
- 2009-02-06 EA EA201001239A patent/EA201001239A1/ru unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AU2009211378A1 (en) | 2009-08-13 |
| CA2714350A1 (en) | 2009-08-13 |
| EP2250166A1 (en) | 2010-11-17 |
| JP2011511039A (ja) | 2011-04-07 |
| US20100331322A1 (en) | 2010-12-30 |
| BRPI0907933A2 (pt) | 2015-07-28 |
| KR20100131427A (ko) | 2010-12-15 |
| EA201001239A1 (ru) | 2011-04-29 |
| US8022069B2 (en) | 2011-09-20 |
| WO2009098276A1 (en) | 2009-08-13 |
| CN101939318A (zh) | 2011-01-05 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |