MD4009B1 - Utilizarea 1-metil-4-(N-metilaminobutil-4)-Beta-carbolinei in calitate de remediu antituberculos - Google Patents
Utilizarea 1-metil-4-(N-metilaminobutil-4)-Beta-carbolinei in calitate de remediu antituberculos Download PDFInfo
- Publication number
- MD4009B1 MD4009B1 MDA20080198A MD20080198A MD4009B1 MD 4009 B1 MD4009 B1 MD 4009B1 MD A20080198 A MDA20080198 A MD A20080198A MD 20080198 A MD20080198 A MD 20080198A MD 4009 B1 MD4009 B1 MD 4009B1
- Authority
- MD
- Moldova
- Prior art keywords
- antituberculous
- remedy
- methylaminobutyl
- carboline
- beta
- Prior art date
Links
- 230000002365 anti-tubercular Effects 0.000 title abstract 3
- AIFRHYZBTHREPW-UHFFFAOYSA-N cis-beta-Carboline Acid Natural products N1=CC=C2C3=CC=CC=C3NC2=C1 AIFRHYZBTHREPW-UHFFFAOYSA-N 0.000 title 1
- OMGIBPZQATWNBX-UHFFFAOYSA-N Brevicarine Chemical compound N1C2=CC=CC=C2C2=C1C(C)=NC=C2CCCCNC OMGIBPZQATWNBX-UHFFFAOYSA-N 0.000 abstract 2
- -1 brevicarine alkaloid compound Chemical class 0.000 abstract 1
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Inventia se refera la chimie, si anume la utilizarea compusului alcaloidului brevicarin in calitate de remediu antituberculos. Esenta inventiei consta in utilizarea 1-metil-4-(N-metilaminobutil-4)-Beta-carbolinei (brevicarina) cu formula generala:in calitate de remediu antituberculos.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MDA20080198A MD4009C2 (ro) | 2008-07-15 | 2008-07-15 | Utilizarea 1-metil-4-(N-metilaminobutil-4)-β-carbolinei în calitate de remediu antituberculos |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MDA20080198A MD4009C2 (ro) | 2008-07-15 | 2008-07-15 | Utilizarea 1-metil-4-(N-metilaminobutil-4)-β-carbolinei în calitate de remediu antituberculos |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MD4009B1 true MD4009B1 (ro) | 2010-01-29 |
| MD4009C2 MD4009C2 (ro) | 2010-08-31 |
Family
ID=43568882
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MDA20080198A MD4009C2 (ro) | 2008-07-15 | 2008-07-15 | Utilizarea 1-metil-4-(N-metilaminobutil-4)-β-carbolinei în calitate de remediu antituberculos |
Country Status (1)
| Country | Link |
|---|---|
| MD (1) | MD4009C2 (ro) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MD4404C1 (ro) * | 2015-03-18 | 2016-09-30 | Институт Химии Академии Наук Молдовы | Compusul 2-(propiltio)-5H-[1,3,4]tiadiazolo[2,3-b]chinazolin-5-onă, care manifestă activitate antituberculoasă şi procedeu de sinteză a acestuia |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MD4125C1 (ro) * | 2010-09-17 | 2012-03-31 | Inst De Chimie Al Academiei De Stiinte A Moldovei | Compuşi 1,3,4-oxadiazolici cu proprietăţi antituberculoase conţinând tiouree monosubstituită |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SU859889A1 (ru) * | 1980-01-17 | 1981-08-30 | Читинский Медицинский Институт | Способ количественного определени 1-метил-4-(N-метилпирролидил-1)- -карболин гидрохлорида |
| US5817321A (en) * | 1992-10-08 | 1998-10-06 | Supratek Pharma, Inc. | Biological agent compositions |
| ES2215631T3 (es) * | 1999-03-23 | 2004-10-16 | Hollis-Eden Pharmaceuticals Inc. | Hemihidrato de 16alfa-bromoepiandrosterona. |
| IT1311924B1 (it) * | 1999-04-13 | 2002-03-20 | Nicox Sa | Composti farmaceutici. |
| IT1311923B1 (it) * | 1999-04-13 | 2002-03-20 | Nicox Sa | Composti farmaceutici. |
| UA71629C2 (en) * | 1999-08-03 | 2004-12-15 | Lilli Icos Llc | Composition containing free drug particulate form of ?-carboline (variants), method for its manufacture (variants), and method for treating sexual dysfunction |
| IT1314184B1 (it) * | 1999-08-12 | 2002-12-06 | Nicox Sa | Composizioni farmaceutiche per la terapia di condizioni di stressossidativo |
| DE19951360A1 (de) * | 1999-10-26 | 2001-05-03 | Aventis Pharma Gmbh | Substituierte Indole |
| IT1317735B1 (it) * | 2000-01-26 | 2003-07-15 | Nicox Sa | Sali di agenti antimicrobici. |
| UA74826C2 (en) * | 2000-05-17 | 2006-02-15 | Ortho Mcneil Pharm Inc | ?-carboline derivatives as phosphodiesterase inhibitors |
| TW200403072A (en) * | 2002-01-23 | 2004-03-01 | Upjohn Co | Combination therapy for the treatment of bacterial infections |
| UA78839C2 (en) * | 2002-07-31 | 2007-04-25 | Lilly Icos Llc | Modified pictet-spengler reaction and products prepared therefrom |
| WO2004098519A2 (en) * | 2003-05-02 | 2004-11-18 | Georgetown University | Ginkgo biloba extract as a treatment for therapeutic induced neurotoxicity |
| US20050148553A1 (en) * | 2003-09-05 | 2005-07-07 | Testa Raymond T. | Use of tigecycline, alone, or in combination with rifampin to treat osteomyelitis and/or septic arthritis |
| ES2306146T3 (es) * | 2004-05-28 | 2008-11-01 | Janssen Pharmaceutica Nv | Uso de derivados de quinolina sustituidos para el tratamiento de enfermedades micobacterianas resistentes a farmacos. |
| TW200628161A (en) * | 2004-11-12 | 2006-08-16 | Panacos Pharmaceuticals Inc | Novel betulin derivatives, preparation thereof and use thereof |
-
2008
- 2008-07-15 MD MDA20080198A patent/MD4009C2/ro not_active IP Right Cessation
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MD4404C1 (ro) * | 2015-03-18 | 2016-09-30 | Институт Химии Академии Наук Молдовы | Compusul 2-(propiltio)-5H-[1,3,4]tiadiazolo[2,3-b]chinazolin-5-onă, care manifestă activitate antituberculoasă şi procedeu de sinteză a acestuia |
Also Published As
| Publication number | Publication date |
|---|---|
| MD4009C2 (ro) | 2010-08-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG4A | Patent for invention issued | ||
| KA4A | Patent for invention lapsed due to non-payment of fees (with right of restoration) | ||
| MM4A | Patent for invention definitely lapsed due to non-payment of fees |