MC1982A1 - PROCESS FOR THE PREPARATION OF DIDESOXYCITIDIN DERIVATIVES - Google Patents
PROCESS FOR THE PREPARATION OF DIDESOXYCITIDIN DERIVATIVESInfo
- Publication number
- MC1982A1 MC1982A1 MC882009A MC2009A MC1982A1 MC 1982 A1 MC1982 A1 MC 1982A1 MC 882009 A MC882009 A MC 882009A MC 2009 A MC2009 A MC 2009A MC 1982 A1 MC1982 A1 MC 1982A1
- Authority
- MC
- Monaco
- Prior art keywords
- didesoxycitidin
- derivatives
- preparation
- didesoxycitidin derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US10722187A | 1987-10-09 | 1987-10-09 |
Publications (1)
Publication Number | Publication Date |
---|---|
MC1982A1 true MC1982A1 (en) | 1989-11-23 |
Family
ID=22315505
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MC882009A MC1982A1 (en) | 1987-10-09 | 1988-10-07 | PROCESS FOR THE PREPARATION OF DIDESOXYCITIDIN DERIVATIVES |
Country Status (14)
Country | Link |
---|---|
EP (1) | EP0311100A3 (en) |
JP (1) | JPH01132597A (en) |
KR (1) | KR890006624A (en) |
AU (1) | AU2355488A (en) |
DK (1) | DK564088A (en) |
FI (1) | FI884627A (en) |
HU (1) | HU201090B (en) |
IL (1) | IL87949A0 (en) |
MC (1) | MC1982A1 (en) |
NO (1) | NO884497L (en) |
NZ (1) | NZ226481A (en) |
PT (1) | PT88716B (en) |
YU (1) | YU187788A (en) |
ZA (1) | ZA886890B (en) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6448392B1 (en) | 1985-03-06 | 2002-09-10 | Chimerix, Inc. | Lipid derivatives of antiviral nucleosides: liposomal incorporation and method of use |
US5223263A (en) * | 1988-07-07 | 1993-06-29 | Vical, Inc. | Liponucleotide-containing liposomes |
NZ223910A (en) * | 1987-03-20 | 1991-02-26 | Bristol Myers Co | 2',3'-dideoxynucleosides, process for their production and intermediates therefor |
US5631370A (en) * | 1988-01-20 | 1997-05-20 | Regents Of The University Of Minnesota | Optically-active isomers of dideoxycarbocyclic nucleosides |
US6599887B2 (en) | 1988-07-07 | 2003-07-29 | Chimerix, Inc. | Methods of treating viral infections using antiviral liponucleotides |
US6252060B1 (en) | 1988-07-07 | 2001-06-26 | Nexstar Pharmaceuticals, Inc. | Antiviral liponucleosides: treatment of hepatitis B |
US5817638A (en) * | 1988-07-07 | 1998-10-06 | Nexstar Pharmaceuticals, Inc. | Antiviral liponucleosides: treatment of hepatitis B |
GB8823320D0 (en) * | 1988-10-05 | 1988-11-09 | Nycomed As | Chemical compounds |
AU636678B2 (en) * | 1989-11-06 | 1993-05-06 | Nycomed Imaging As | Nucleoside derivatives |
US5192764A (en) * | 1991-05-30 | 1993-03-09 | Research Foundation Of State Of N.Y. | Pyrazinone n-oxide nucleosides and analogs thereof |
CA2079413C (en) * | 1991-09-30 | 2003-09-09 | Masakatsu Kaneko | Pyrimidine nucleoside derivatives having anti-tumor activity, their preparation and use |
US6576636B2 (en) | 1996-05-22 | 2003-06-10 | Protarga, Inc. | Method of treating a liver disorder with fatty acid-antiviral agent conjugates |
AU1412299A (en) * | 1997-11-25 | 1999-06-15 | Protarga, Inc. | Nucleoside analog compositions and uses thereof |
EP1427407A4 (en) | 2001-03-23 | 2005-05-11 | Luitpold Pharm Inc | Fatty amine drug conjugates |
ATE556706T1 (en) | 2001-03-23 | 2012-05-15 | Luitpold Pharm Inc | FAT ALCOHOL-DRUG CONJUGATES |
CN100560073C (en) | 2001-12-14 | 2009-11-18 | 法玛塞特公司 | The N that is used for the treatment of viral infection 4-acyl group cytidine |
US9326983B2 (en) | 2013-08-01 | 2016-05-03 | University Of Kentucky Research Foundation | Compositions and methods for treating retinal degradation |
EP4215527A1 (en) * | 2015-02-26 | 2023-07-26 | University Of Kentucky Research Foundation | Compositions and methods for treating retinal degradation |
US11219623B2 (en) | 2015-02-26 | 2022-01-11 | University Of Kentucky Research Foundation | Inflammasome inhibition for the treatment of Parkinson's disease, Alzheimer's disease and multiple sclerosis |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5943550B2 (en) * | 1975-08-29 | 1984-10-23 | 田辺製薬株式会社 | Process for producing unsaturated nucleosides |
HU196607B (en) * | 1985-05-15 | 1988-12-28 | Wellcome Found | Process for producing dideoxy-nucleosides and pharmaceutics comprising such compounds |
AU613026B2 (en) * | 1987-03-24 | 1991-07-25 | Nycomed As | 2',3' dideoxyribofuranoxide derivatives |
EP0294113A1 (en) * | 1987-05-29 | 1988-12-07 | The Wellcome Foundation Limited | Therapeutic nucleosides |
US4837311A (en) * | 1987-06-22 | 1989-06-06 | Hoffman-La Roche Inc. | Anti-retroviral compounds |
-
1988
- 1988-09-15 ZA ZA886890A patent/ZA886890B/en unknown
- 1988-10-06 IL IL87949A patent/IL87949A0/en unknown
- 1988-10-06 NZ NZ226481A patent/NZ226481A/en unknown
- 1988-10-07 MC MC882009A patent/MC1982A1/en unknown
- 1988-10-07 FI FI884627A patent/FI884627A/en not_active IP Right Cessation
- 1988-10-07 PT PT88716A patent/PT88716B/en not_active IP Right Cessation
- 1988-10-07 HU HU885191A patent/HU201090B/en not_active IP Right Cessation
- 1988-10-07 NO NO88884497A patent/NO884497L/en unknown
- 1988-10-07 KR KR1019880013065A patent/KR890006624A/en not_active Application Discontinuation
- 1988-10-07 EP EP19880116655 patent/EP0311100A3/en not_active Withdrawn
- 1988-10-07 DK DK564088A patent/DK564088A/en not_active Application Discontinuation
- 1988-10-07 AU AU23554/88A patent/AU2355488A/en not_active Abandoned
- 1988-10-07 YU YU01877/88A patent/YU187788A/en unknown
- 1988-10-08 JP JP63254668A patent/JPH01132597A/en active Pending
Also Published As
Publication number | Publication date |
---|---|
IL87949A0 (en) | 1989-03-31 |
KR890006624A (en) | 1989-06-14 |
JPH01132597A (en) | 1989-05-25 |
DK564088A (en) | 1989-04-10 |
HUT47592A (en) | 1989-03-28 |
DK564088D0 (en) | 1988-10-07 |
FI884627A (en) | 1989-04-10 |
ZA886890B (en) | 1989-05-30 |
NO884497L (en) | 1989-04-10 |
FI884627A0 (en) | 1988-10-07 |
NO884497D0 (en) | 1988-10-07 |
PT88716B (en) | 1992-12-31 |
NZ226481A (en) | 1992-01-29 |
HU201090B (en) | 1990-09-28 |
AU2355488A (en) | 1989-04-13 |
EP0311100A2 (en) | 1989-04-12 |
EP0311100A3 (en) | 1990-10-31 |
YU187788A (en) | 1990-04-30 |
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Legal Events
Date | Code | Title | Description |
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YP | Annual fee paid |