MA53914A - Polymorphes cristallins d'inhibiteurs de la tyrosine kinase de bruton - Google Patents

Polymorphes cristallins d'inhibiteurs de la tyrosine kinase de bruton

Info

Publication number
MA53914A
MA53914A MA053914A MA53914A MA53914A MA 53914 A MA53914 A MA 53914A MA 053914 A MA053914 A MA 053914A MA 53914 A MA53914 A MA 53914A MA 53914 A MA53914 A MA 53914A
Authority
MA
Morocco
Prior art keywords
bruton
tyrosine kinase
kinase inhibitors
crystalline polymorphs
polymorphs
Prior art date
Application number
MA053914A
Other languages
English (en)
Inventor
Chaomin Li
Yiqing Lin
Daniel B Patience
Anton Peterson
Kalyan Vasudevan
Fengmei Zheng
Original Assignee
Biogen Ma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biogen Ma Inc filed Critical Biogen Ma Inc
Publication of MA53914A publication Critical patent/MA53914A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
MA053914A 2018-10-15 2019-10-15 Polymorphes cristallins d'inhibiteurs de la tyrosine kinase de bruton MA53914A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201862745741P 2018-10-15 2018-10-15

Publications (1)

Publication Number Publication Date
MA53914A true MA53914A (fr) 2021-08-25

Family

ID=68426868

Family Applications (1)

Application Number Title Priority Date Filing Date
MA053914A MA53914A (fr) 2018-10-15 2019-10-15 Polymorphes cristallins d'inhibiteurs de la tyrosine kinase de bruton

Country Status (5)

Country Link
US (1) US11820760B2 (fr)
EP (1) EP3866926A1 (fr)
JP (1) JP7476214B2 (fr)
MA (1) MA53914A (fr)
WO (1) WO2020081514A1 (fr)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4938949A (en) 1988-09-12 1990-07-03 University Of New York Treatment of damaged bone marrow and dosage units therefor
RU2619465C2 (ru) 2012-10-26 2017-05-16 Ф. Хоффманн-Ля Рош Аг Ингибиторы тирозинкиназы брутона
EP3060550B1 (fr) * 2013-10-21 2019-05-15 Merck Patent GmbH Composés hétéroaryle servant d'inhibiteurs de la btk et leurs utilisations
CN108947913A (zh) 2013-12-11 2018-12-07 比奥根Ma公司 可用于治疗人类肿瘤学、神经病学和免疫学疾病的联芳基化合物
US20180282310A1 (en) 2015-06-10 2018-10-04 Biogen Ma Inc. Forms and compositions of biaryl inhibitors of bruton's tyrosine kinase
JOP20190233A1 (ar) 2017-04-14 2019-10-02 Biogen Ma Inc نظائر بنزوازيبين بوصفها عوامل مثبطة لتيروزين كيناز بروتون
ES2968222T3 (es) 2018-05-14 2024-05-08 Biogen Ma Inc Agentes inhibidores para la tirosina cinasa de Bruton

Also Published As

Publication number Publication date
EP3866926A1 (fr) 2021-08-25
JP7476214B2 (ja) 2024-04-30
US11820760B2 (en) 2023-11-21
WO2020081514A1 (fr) 2020-04-23
US20210387972A1 (en) 2021-12-16
JP2022502516A (ja) 2022-01-11
WO2020081514A9 (fr) 2020-05-22

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