MA50899B1 - Composés utiles pour l'inhibition de cdk7 - Google Patents
Composés utiles pour l'inhibition de cdk7Info
- Publication number
- MA50899B1 MA50899B1 MA50899A MA50899A MA50899B1 MA 50899 B1 MA50899 B1 MA 50899B1 MA 50899 A MA50899 A MA 50899A MA 50899 A MA50899 A MA 50899A MA 50899 B1 MA50899 B1 MA 50899B1
- Authority
- MA
- Morocco
- Prior art keywords
- compounds useful
- cdk7 inhibition
- cdk7
- inhibition
- novel
- Prior art date
Links
- 101150059448 cdk7 gene Proteins 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 title 1
- 230000005764 inhibitory process Effects 0.000 title 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La présente invention concerne de nouveaux inhibiteurs de cdk7 et des compositions pharmaceutiques associées : (i), ou un sel pharmaceutiquement acceptable de ceux-ci.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP17382778 | 2017-11-16 | ||
| PCT/US2018/060025 WO2019099298A1 (fr) | 2017-11-16 | 2018-11-09 | Composés utiles pour l'inhibition de cdk7 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MA50899A MA50899A (fr) | 2020-09-23 |
| MA50899B1 true MA50899B1 (fr) | 2022-10-31 |
Family
ID=60484312
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA50899A MA50899B1 (fr) | 2017-11-16 | 2018-11-09 | Composés utiles pour l'inhibition de cdk7 |
Country Status (2)
| Country | Link |
|---|---|
| AR (1) | AR113817A1 (fr) |
| MA (1) | MA50899B1 (fr) |
-
2018
- 2018-10-31 AR ARP180103173A patent/AR113817A1/es unknown
- 2018-11-09 MA MA50899A patent/MA50899B1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MA50899A (fr) | 2020-09-23 |
| AR113817A1 (es) | 2020-06-17 |
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