MA18762A1 - Acides penicillamiques 6-b-substitues inhibiteurs de b-lactamase,leur procede de production et composition pharmaceutique les contenant - Google Patents

Acides penicillamiques 6-b-substitues inhibiteurs de b-lactamase,leur procede de production et composition pharmaceutique les contenant

Info

Publication number
MA18762A1
MA18762A1 MA18960A MA18960A MA18762A1 MA 18762 A1 MA18762 A1 MA 18762A1 MA 18960 A MA18960 A MA 18960A MA 18960 A MA18960 A MA 18960A MA 18762 A1 MA18762 A1 MA 18762A1
Authority
MA
Morocco
Prior art keywords
penicillamic
acids
substituted
production
pharmaceutical composition
Prior art date
Application number
MA18960A
Other languages
English (en)
Inventor
Seicchi Hamanaka Ernest
Stephen Kellogg Michael
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MA18762A1 publication Critical patent/MA18762A1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • A61K31/43Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MA18960A 1979-03-05 1980-03-04 Acides penicillamiques 6-b-substitues inhibiteurs de b-lactamase,leur procede de production et composition pharmaceutique les contenant MA18762A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US1780979A 1979-03-05 1979-03-05

Publications (1)

Publication Number Publication Date
MA18762A1 true MA18762A1 (fr) 1980-10-01

Family

ID=21784657

Family Applications (1)

Application Number Title Priority Date Filing Date
MA18960A MA18762A1 (fr) 1979-03-05 1980-03-04 Acides penicillamiques 6-b-substitues inhibiteurs de b-lactamase,leur procede de production et composition pharmaceutique les contenant

Country Status (6)

Country Link
JP (3) JPS55129289A (fr)
BE (1) BE882027A (fr)
MA (1) MA18762A1 (fr)
PL (1) PL222471A1 (fr)
ZA (1) ZA80880B (fr)
ZM (1) ZM3080A1 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003224874A1 (en) * 2002-04-04 2003-10-27 Alamx, L.L.C. INHIBITORS OF SERINE AND METALLO-ss-LACTAMASES

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4203992A (en) * 1978-12-11 1980-05-20 E. R. Squibb & Sons, Inc. β-Bromopenicillanic acid sulfone
JPS5598186A (en) * 1979-01-10 1980-07-25 Beecham Group Ltd Manufacture of penicillin derivative

Also Published As

Publication number Publication date
PL222471A1 (fr) 1980-12-01
JPS59161383A (ja) 1984-09-12
JPS55129289A (en) 1980-10-06
BE882027A (fr) 1980-09-03
JPS59161384A (ja) 1984-09-12
ZM3080A1 (en) 1980-11-21
ZA80880B (en) 1981-02-25

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