LTIP916A - Method for preparing aromatase inhibiting 4(5)-imidazole derivatives - Google Patents

Method for preparing aromatase inhibiting 4(5)-imidazole derivatives

Info

Publication number
LTIP916A
LTIP916A LTIP916A LTIP916A LTIP916A LT IP916 A LTIP916 A LT IP916A LT IP916 A LTIP916 A LT IP916A LT IP916 A LTIP916 A LT IP916A LT IP916 A LTIP916 A LT IP916A
Authority
LT
Lithuania
Prior art keywords
imidazole derivatives
aromatase inhibiting
preparing
preparing aromatase
inhibiting
Prior art date
Application number
LTIP916A
Inventor
Arto Johannes Karjalainen
Lauri Veikko Matti Kangas
Kauko Oiva Antero Kurkela
Original Assignee
Orion Yhtymae Oy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Orion Yhtymae Oy filed Critical Orion Yhtymae Oy
Publication of LTIP916A publication Critical patent/LTIP916A/en
Publication of LT3658B publication Critical patent/LT3658B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
LTIP916A 1987-10-09 1993-08-31 Method for preparing aromatase inhibiting 4(5)-imidazole derivatives LT3658B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8723715A GB2210875B (en) 1987-10-09 1987-10-09 Aromatase inhibiting 4(5)-imidazoles

Publications (2)

Publication Number Publication Date
LTIP916A true LTIP916A (en) 1995-03-27
LT3658B LT3658B (en) 1996-01-25

Family

ID=10625036

Family Applications (1)

Application Number Title Priority Date Filing Date
LTIP916A LT3658B (en) 1987-10-09 1993-08-31 Method for preparing aromatase inhibiting 4(5)-imidazole derivatives

Country Status (24)

Country Link
US (1) US5098923A (en)
EP (1) EP0311447B1 (en)
JP (1) JPH01132568A (en)
KR (1) KR890006593A (en)
CN (1) CN1036993C (en)
AU (1) AU615482B2 (en)
CA (1) CA1329616C (en)
DD (1) DD282912A5 (en)
DE (1) DE3874073T2 (en)
DK (1) DK550988A (en)
ES (1) ES2043839T3 (en)
FI (1) FI93105C (en)
GB (1) GB2210875B (en)
GR (1) GR3006343T3 (en)
HU (1) HU201024B (en)
IE (1) IE61180B1 (en)
IL (1) IL87969A (en)
LT (1) LT3658B (en)
NO (1) NO172048C (en)
NZ (1) NZ226483A (en)
PT (1) PT88717B (en)
RU (2) RU1819263C (en)
UA (1) UA13218A (en)
ZA (1) ZA887545B (en)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2210875B (en) 1987-10-09 1991-05-29 Farmos Oy Aromatase inhibiting 4(5)-imidazoles
GB8818561D0 (en) * 1988-08-04 1988-09-07 Ici Plc Diphenylethane derivatives
AU627559B2 (en) * 1989-03-30 1992-08-27 Farmos-Yhtyma Oy Novel aromatase inhibiting 4(5)-imidazoles
US5439928A (en) * 1989-03-30 1995-08-08 Orion-Yhtyma Oy Aromatase inhibiting 4(5)-imidazoles
GB2229719B (en) * 1989-03-30 1992-04-29 Farmos Oy Novel aromatase inhibiting 4(5)-imidazoles
GB2248058B (en) 1990-09-21 1994-09-14 Orion Yhtymae Oy Aromatase inhibiting 4(5)-imidazoles
GB9125924D0 (en) * 1991-06-18 1992-02-05 Orion Yhtymae Oy Stereoisomers of an imidazole derivative
US6479526B1 (en) 1995-04-12 2002-11-12 The Procter & Gamble Company Pharmaceutical composition for inhibiting the growth of viruses and cancers
ZA962879B (en) * 1995-04-12 1997-03-17 Procter & Gamble A pharmaceutical composition for inhibiting the growth of viruses and cancers
US6262093B1 (en) 1995-04-12 2001-07-17 The Proctor & Gamble Company Methods of treating cancer with benzimidazoles
US6265427B1 (en) 1995-06-07 2001-07-24 The Proctor & Gamble Company Pharmaceutical composition for the method of treating leukemia
WO1997026246A1 (en) * 1996-01-16 1997-07-24 Warner-Lambert Company Substituted histidine inhibitors of protein farnesyltransferase
US5900429A (en) * 1997-01-28 1999-05-04 The Procter & Gamble Company Method for inhibiting the growth of cancers
US6506783B1 (en) * 1997-05-16 2003-01-14 The Procter & Gamble Company Cancer treatments and pharmaceutical compositions therefor
US6245789B1 (en) 1998-05-19 2001-06-12 The Procter & Gamble Company HIV and viral treatment
US6423734B1 (en) 1999-08-13 2002-07-23 The Procter & Gamble Company Method of preventing cancer
US6608096B1 (en) 2000-09-26 2003-08-19 University Of Arizona Foundation Compounds and methods for use thereof in the treatment of cancer or viral infections
US6407105B1 (en) 2000-09-26 2002-06-18 The Procter & Gamble Company Compounds and methods for use thereof in the treatment of cancer or viral infections
US6380232B1 (en) 2000-09-26 2002-04-30 The Procter & Gamble Company Benzimidazole urea derivatives, and pharmaceutical compositions and unit dosages thereof
US6462062B1 (en) 2000-09-26 2002-10-08 The Procter & Gamble Company Compounds and methods for use thereof in the treatment of cancer or viral infections
US6515074B2 (en) * 2001-01-22 2003-02-04 Delphi Technologies, Inc. Thermoplastic polymer alloy compositions and process for manufacture thereof
CN1633296A (en) 2002-03-26 2005-06-29 贝林格尔·英格海姆药物公司 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
JP2005521717A (en) * 2002-03-26 2005-07-21 ベーリンガー インゲルハイム ファーマシューティカルズ インコーポレイテッド Glucocorticoid mimetics, process for producing the same, pharmaceutical composition thereof, and use thereof
US7074806B2 (en) 2002-06-06 2006-07-11 Boehringer Ingelheim Pharmaceuticals, Inc. Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
MXPA05006872A (en) 2003-01-03 2005-08-16 Boehringer Ingelheim Pharma 1-propanol and 1-propylamine derivatives and their use as glucocorticoid ligands.
UY28526A1 (en) 2003-09-24 2005-04-29 Boehringer Ingelheim Pharma GLUCOCORTICOID MIMETICS, METHODS OF PREPARATION PHARMACEUTICAL COMPOSITIONS AND USES OF THE SAME
US7795272B2 (en) 2004-03-13 2010-09-14 Boehringer Ingelheim Pharmaceutical, Inc. Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof
ATE433958T1 (en) 2004-12-27 2009-07-15 Boehringer Ingelheim Pharma GLUCOCORTICOID MIMETICS, METHOD FOR THE PRODUCTION THEREOF, PHARMACEUTICAL COMPOSITIONS AND USE THEREOF
AU2007329548A1 (en) 2006-12-06 2008-06-12 Boehringer Ingelheim International Gmbh Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
EP2095819A1 (en) * 2008-02-28 2009-09-02 Maastricht University N-benzyl imidazole derivatives and their use as aldosterone synthase inhibitors
PT2300472E (en) 2008-06-06 2012-02-20 Boehringer Ingelheim Int Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2069481B (en) * 1980-02-13 1983-07-27 Farmos Oy Substituted imidazole derivatives
GB2092569B (en) * 1981-02-05 1984-09-19 Farmos Oy Substituted imidazole derivatives and their preparation and use
GB2096987B (en) * 1981-04-22 1984-04-04 Farmos Oy Substituted imidazole and imidazole derivatives and their preparation and use
GB2101114B (en) * 1981-07-10 1985-05-22 Farmos Group Ltd Substituted imidazole derivatives and their preparation and use
US4605661A (en) * 1984-06-18 1986-08-12 Eli Lilly And Company Aromastase inhibiting α,α-diarylimidazole-4(5)-propionitriles, α,α-diarylimidazole-4(5)-propionamides, and 4(5)-(2,2-diarylethyl)imidazoles
LU85747A1 (en) * 1985-01-28 1986-08-04 Continental Pharma IMIDAZOLE DERIVATIVES, PREPARATION AND USE THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING DERIVATIVES
GB2210875B (en) 1987-10-09 1991-05-29 Farmos Oy Aromatase inhibiting 4(5)-imidazoles
AU627559B2 (en) 1989-03-30 1992-08-27 Farmos-Yhtyma Oy Novel aromatase inhibiting 4(5)-imidazoles

Also Published As

Publication number Publication date
NZ226483A (en) 1991-02-26
IE61180B1 (en) 1994-10-05
FI884497A0 (en) 1988-09-30
KR890006593A (en) 1989-06-14
ES2043839T3 (en) 1994-01-01
ZA887545B (en) 1989-06-28
DD282912A5 (en) 1990-09-26
HUT49582A (en) 1989-10-30
CN1036993C (en) 1998-01-14
RU1819263C (en) 1993-05-30
JPH01132568A (en) 1989-05-25
GB2210875B (en) 1991-05-29
IL87969A (en) 1993-04-04
GB2210875A (en) 1989-06-21
EP0311447A1 (en) 1989-04-12
GR3006343T3 (en) 1993-06-21
US5098923A (en) 1992-03-24
FI93105C (en) 1995-02-27
PT88717B (en) 1992-12-31
NO172048C (en) 1993-06-02
FI884497A (en) 1989-04-10
CA1329616C (en) 1994-05-17
LT3658B (en) 1996-01-25
DE3874073D1 (en) 1992-10-01
DK550988A (en) 1989-04-10
IE883055L (en) 1989-04-09
DK550988D0 (en) 1988-10-03
NO884473L (en) 1989-04-10
UA13218A (en) 1997-02-28
IL87969A0 (en) 1989-03-31
DE3874073T2 (en) 1993-01-21
NO172048B (en) 1993-02-22
EP0311447B1 (en) 1992-08-26
CN1033995A (en) 1989-07-19
NO884473D0 (en) 1988-10-07
RU2045519C1 (en) 1995-10-10
AU2349088A (en) 1989-04-13
FI93105B (en) 1994-11-15
GB8723715D0 (en) 1987-11-11
HU201024B (en) 1990-09-28
AU615482B2 (en) 1991-10-03

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Legal Events

Date Code Title Description
MM9A Lapsed patents

Effective date: 19970831