KR880002864A - 3-페닐-3-(1h-1,2,4-트리아 3-페닐-3-(1h-1,2,4-트리아졸-1-일메틸)-5-치환된-2-메틸이속사졸리딘 - Google Patents

3-페닐-3-(1h-1,2,4-트리아 3-페닐-3-(1h-1,2,4-트리아졸-1-일메틸)-5-치환된-2-메틸이속사졸리딘 Download PDF

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Publication number
KR880002864A
KR880002864A KR870009310A KR870009310A KR880002864A KR 880002864 A KR880002864 A KR 880002864A KR 870009310 A KR870009310 A KR 870009310A KR 870009310 A KR870009310 A KR 870009310A KR 880002864 A KR880002864 A KR 880002864A
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KR
South Korea
Prior art keywords
compound
methyl
ylmethyl
triazol
isoxazolidine
Prior art date
Application number
KR870009310A
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English (en)
Inventor
스테파노 죠지 바실
바이론 물렌 죠지
Original Assignee
마델린 알·락스니시
펜왈트 코포레이션
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Priority claimed from US06/900,857 external-priority patent/US4727157A/en
Priority claimed from US07/036,831 external-priority patent/US4767866A/en
Priority claimed from US07/036,838 external-priority patent/US4769471A/en
Application filed by 마델린 알·락스니시, 펜왈트 코포레이션 filed Critical 마델린 알·락스니시
Publication of KR880002864A publication Critical patent/KR880002864A/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

내용 없음

Description

3-페닐-3-(1H-1,2,4-트리이졸-1-일메틸)-5-치환된-2-메틸이속사졸리딘
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (11)

  1. 에난티오머, 언급된 에난티오머의 디아스 테레오머 쌍을 포함하는 그들의 에난티오머 혼합물 형태의 하기 일반식의 화합물 및 약제학적으로 허용되는 그의 산부가염.
    상기식에서, a는 1 또는 2이고, R1은 수소, 저급 알킬, 저급 알콕시, 할로겐 및 그의 조합 중에서 선택되며, 단, 오르토 위치는 수소이고,
    (여기서, b=1 또는 2 이고, R2는 수소, 저급알킬, 저급알콕시, 할로겐, 알콕시카보닐, 알카노일아미노, 니트로, 및 그의 조합 중에서 선택된다) (b) 적쇄 또는 측쇄의 -(CH2)nCH3(여기서, n은 내지 18이다) 및 (c)(여기서, b=1 또는 2이고, R2는 수소, 저급알킬, 저급알콕시, 할로겐, 트리플루오로메틸, 니트로, 및 그의 조합중에서 선택된다)중에서 선택된다.
  2. 제 1 항에 있어서, R이 -CH2O이고, 여기서, b는 1 또는 2이며, R2는 수소, 저급알킬, 저급알콕시, 할로겐, 알콕시카보닐, 알카노일아미노, 니트로, 및 그의 조합 중에서 선택되는 화합물.
  3. 제 1 항에 있어서, R이 측쇄 또는 비측쇄의 -(CH2)nCH3(여기서, n은 1 내지 18이다)인 화합물.
  4. 제 1 항에 있어서, R이이고, 여기서 b는 1 또는 2이며, R2는 수소, 저급알킬, 저급알콕시, 할로겐, 트리플루오르메틸, 니트로, 및 그의 조합중에서 선택되는 화합물,
  5. 제 2 항에 있어서, 3-(4-클로로페닐)-3-(1H-1,2,4-트리아졸-1-일메틸)- 2-메틸-5-[(4-클로로펜옥시)메틸] 이속사졸리딘의 화합물.
  6. 제 2 항에 있어서, 3-(4-클로로페닐)-3-(1H-1,2,4-트리아졸-1-일메틸)- 2-메틸-5-[(4-메톡시펜옥시)메틸]-이속사졸리딘의 화합물.
  7. 제 2 항에 있어서, 3-(4-클로로페닐)-3-(1H-1,2,4-트리아졸-1-일메틸)- 2-메틸-5-[(4-클로로-3-메틸페닐)메틸]-이속사졸리딘의 화합물.
  8. 제 2 항에 있어서, 3-(4-메톡시페닐)-3-(1H-1,2,4-트리아졸-1-일메틸)- 2-메틸-5-[(4-클로로펜옥시)메틸]-이속사졸리딘의 화합물.
  9. 제 4 항에 있어서, 3,5-비스(4-클로로페닐)-2-메틸-3-(1H-1,2,4-트리아졸-1-일메틸)이속사졸리딘의 화합물.
  10. 제 4 항에 있어서, 3-(4-클로로페닐)-5-(4플루오로페닐)-2-메틸-3-(1H-1,2,4-트리아졸-1-일메틸)-이속사졸리딘의 화합물.
  11. 제 4 항에 있어서, 3-5-비스(4-플루오로페닐)-2-메틸-3-(1H-1,2,4-트리아졸-1-일메틸)이속사졸리딘의 화합물.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR870009310A 1986-08-27 1987-08-26 3-페닐-3-(1h-1,2,4-트리아 3-페닐-3-(1h-1,2,4-트리아졸-1-일메틸)-5-치환된-2-메틸이속사졸리딘 KR880002864A (ko)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US06/900,857 US4727157A (en) 1986-08-27 1986-08-27 3-(Substituted phenyl)-3-(1H-1,2,4-triazol-1-yl)methyl-2-methyl-5-[(substituted phenoxy)methyl]isoxazolidine derivatives
US900857 1986-08-27
US36831 1987-04-10
US07/036,831 US4767866A (en) 1987-04-10 1987-04-10 3-Phenyl-3-(1H-1,2,4-triazol-1-ylmethyl)-2-methyl-5-alkylisoxazolidines
US36838 1987-04-10
US07/036,838 US4769471A (en) 1987-04-10 1987-04-10 Substituted 3,5-diphenyl-3-(1H-1,2,4-triazol-1-yl-methyl)-2-methylisoxazolidines

Publications (1)

Publication Number Publication Date
KR880002864A true KR880002864A (ko) 1988-05-12

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Family Applications (1)

Application Number Title Priority Date Filing Date
KR870009310A KR880002864A (ko) 1986-08-27 1987-08-26 3-페닐-3-(1h-1,2,4-트리아 3-페닐-3-(1h-1,2,4-트리아졸-1-일메틸)-5-치환된-2-메틸이속사졸리딘

Country Status (8)

Country Link
EP (1) EP0257351A3 (ko)
KR (1) KR880002864A (ko)
AU (1) AU596681B2 (ko)
DK (1) DK444787A (ko)
FI (1) FI873708A (ko)
IL (1) IL83273A0 (ko)
NO (1) NO169071C (ko)
NZ (1) NZ221116A (ko)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL87797A0 (en) * 1987-10-02 1989-03-31 Pennwalt Corp 5-mono or disubstituted-3-(phenyl or 2-naphthalenyl)-3-((1h-imidazol-1-ylmethyl)-and(1h-1,2,4-triazol-1-ylmethyl))-2-(methyl or benzyl)isoxazolidines
DE4013723A1 (de) * 1990-04-28 1991-10-31 Basf Ag 5-(1,2,4-triazol-1-ylmethyl)-isoxazoline

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4870094A (en) * 1984-05-02 1989-09-26 Uniroyal Chemical Company, Inc. Substituted imidazoles and triazoles
ATE67493T1 (de) * 1985-02-04 1991-10-15 Bayer Agrochem Kk Heterocyclische verbindungen.
IL87797A0 (en) * 1987-10-02 1989-03-31 Pennwalt Corp 5-mono or disubstituted-3-(phenyl or 2-naphthalenyl)-3-((1h-imidazol-1-ylmethyl)-and(1h-1,2,4-triazol-1-ylmethyl))-2-(methyl or benzyl)isoxazolidines

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NZ221116A (en) 1990-01-29
FI873708A0 (fi) 1987-08-26
NO873607L (no) 1988-02-29
FI873708A (fi) 1988-02-28
DK444787A (da) 1988-02-28
EP0257351A3 (en) 1989-01-18
AU596681B2 (en) 1990-05-10
EP0257351A2 (en) 1988-03-02
IL83273A0 (en) 1987-12-31
NO169071B (no) 1992-01-27
NO873607D0 (no) 1987-08-26
AU7652287A (en) 1988-03-03
DK444787D0 (da) 1987-08-26
NO169071C (no) 1992-05-06

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