KR880001628A - 비사이클릭 방향족 설포닐 클로라이드의 합성 - Google Patents

비사이클릭 방향족 설포닐 클로라이드의 합성 Download PDF

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Publication number
KR880001628A
KR880001628A KR1019870007931A KR870007931A KR880001628A KR 880001628 A KR880001628 A KR 880001628A KR 1019870007931 A KR1019870007931 A KR 1019870007931A KR 870007931 A KR870007931 A KR 870007931A KR 880001628 A KR880001628 A KR 880001628A
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KR
South Korea
Prior art keywords
bicyclic aromatic
sulfonyl chloride
aromatic sulfonyl
synthesis
formula
Prior art date
Application number
KR1019870007931A
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English (en)
Other versions
KR950001041B1 (ko
Inventor
아브라함 아이킨스 제임스
비-핑 타오 에디
Original Assignee
메리 앤 터커
일라이 릴리 앤드 캄파니
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Application filed by 메리 앤 터커, 일라이 릴리 앤드 캄파니 filed Critical 메리 앤 터커
Publication of KR880001628A publication Critical patent/KR880001628A/ko
Application granted granted Critical
Publication of KR950001041B1 publication Critical patent/KR950001041B1/ko

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D317/00Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/62Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D319/00Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/101,4-Dioxanes; Hydrogenated 1,4-dioxanes
    • C07D319/141,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
    • C07D319/161,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D319/18Ethylenedioxybenzenes, not substituted on the hetero ring

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Furan Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

내용 없음

Description

비사이클릭 방향족 설포닐 클로라이드의 합성
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (4)

  1. 일반식(II)의 화합물을 일반식(III)의 빌스마이어(Villsmeier) 시약과 반응시켜 일반식(I)의 비사이클릭 방향족 설포닐 클로라이드를 제조하는 방법.
    상기식에서,
    n은 1 또는 2이고;
    A는 -O- 또는 -CH2-이며;
    B는 -O-, -CH2-, 또는 -NCH3-이고, 단, A 또는 B 중의 적어도 하나는 -O-이다.
  2. 제1항에 있어서, 생성물이 1, 3-벤조 디옥설-5-설포닐 클로라이드인 방법.
  3. 제1항에 있어서, 생성물이 디하이드로벤조푸란-5-설포닐 클로라이드인 방법.
  4. 제1항에 있어서, 생성물이 1, 4-벤조디옥산-6-설포닐 클로라이드인 방법.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019870007931A 1986-07-23 1987-07-22 이환식 방향족 설포닐 클로라이드의 합성방법 KR950001041B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US88914186A 1986-07-23 1986-07-23
US889,141 1986-07-23
US889141 1986-07-23

Publications (2)

Publication Number Publication Date
KR880001628A true KR880001628A (ko) 1988-04-25
KR950001041B1 KR950001041B1 (ko) 1995-02-08

Family

ID=25394575

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019870007931A KR950001041B1 (ko) 1986-07-23 1987-07-22 이환식 방향족 설포닐 클로라이드의 합성방법

Country Status (9)

Country Link
EP (1) EP0254577B1 (ko)
JP (1) JPS6345275A (ko)
KR (1) KR950001041B1 (ko)
AT (1) ATE46691T1 (ko)
DE (1) DE3760618D1 (ko)
ES (1) ES2011293B3 (ko)
GR (1) GR3000192T3 (ko)
HU (1) HU198197B (ko)
IL (1) IL83215A (ko)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW221049B (ko) * 1991-12-20 1994-02-11 Lilly Co Eli
US5258406A (en) * 1991-12-20 1993-11-02 Eli Lilly And Company Sulfonimidamides
US5387681A (en) * 1992-08-19 1995-02-07 Eli Lilly And Company Synthesis of bicyclic aromatic sulfonic acids sulfonyl chlorides and sulfonamides
US6140505A (en) * 1995-03-10 2000-10-31 G. D. Searle & Co. Synthesis of benzo fused heterocyclic sulfonyl chlorides

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES8705871A1 (es) * 1984-12-29 1987-05-16 Kaken Pharma Co Ltd Un procedimiento para preparar un derivado de benzofurano

Also Published As

Publication number Publication date
GR3000192T3 (en) 1990-12-31
ES2011293B3 (es) 1990-01-01
HU198197B (en) 1989-08-28
EP0254577B1 (en) 1989-09-27
KR950001041B1 (ko) 1995-02-08
ATE46691T1 (de) 1989-10-15
HUT46685A (en) 1988-11-28
JPS6345275A (ja) 1988-02-26
EP0254577A1 (en) 1988-01-27
DE3760618D1 (en) 1989-11-02
IL83215A (en) 1991-12-15
IL83215A0 (en) 1987-12-31

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