KR870003073A - N-phenylsulfonylisonicotinamide derivative - Google Patents

N-phenylsulfonylisonicotinamide derivative Download PDF

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KR870003073A
KR870003073A KR1019860008017A KR860008017A KR870003073A KR 870003073 A KR870003073 A KR 870003073A KR 1019860008017 A KR1019860008017 A KR 1019860008017A KR 860008017 A KR860008017 A KR 860008017A KR 870003073 A KR870003073 A KR 870003073A
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hydrogen
compound
formula
halogen
methylthio
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KR1019860008017A
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Korean (ko)
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히로시 요시다
겐지 고니시
겡고 고이께
다이조 나까가와
시즈오 시마노
세이지 모찌즈끼
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쓰네까즈 사까노
니뽕 가야꾸 가부시끼 가이샤
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Publication of KR870003073A publication Critical patent/KR870003073A/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/44—Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
    • C07D213/53—Nitrogen atoms

Abstract

내용 없음No content

Description

N-페닐술포닐이소니코틴아미드 유도체N-phenylsulfonylisonicotinamide derivative

본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음Since this is an open matter, no full text was included.

Claims (22)

일반식(1)의 화합물:Compound of formula (1): 상기 식에서, X는 할로겐, 저급 알콕시, 저급 알킬티오, 니트로 또는 메틸이고, Y는 수소 또는 염소이고; R은 수소, 저급 알킬 또는 알릴이고; Z는 수소, 저급알킬, 할로겐, 니트로, 메톡시, 메틸티오, 메틸술포닐, -CF3, 페닐, 페녹시 또는 저급 알콕시카보닐이며; 또 n은 1 내지 3의 정수이다.Wherein X is halogen, lower alkoxy, lower alkylthio, nitro or methyl, and Y is hydrogen or chlorine; R is hydrogen, lower alkyl or allyl; Z is hydrogen, lower alkyl, halogen, nitro, methoxy, methylthio, methylsulfonyl, -CF 3 , phenyl, phenoxy or lower alkoxycarbonyl; And n is an integer of 1 to 3. 제1항에 있어서, X가 할로겐, 저급 알콕시 또는 메틸티오이고; Y가 수소 또는 염소이며; R이 수소, 저급 알킬 또는 알릴이고; Z가 수소, 저급 알킬, 할로겐, 니트로, 메톡시, 메틸티오, 메틸술포닐, -CF3, 페닐, 페녹시 또는 저급 알콕시카보닐이며; 또 n이 1 내지 3의 정수인 화합물.The compound of claim 1, wherein X is halogen, lower alkoxy or methylthio; Y is hydrogen or chlorine; R is hydrogen, lower alkyl or allyl; Z is hydrogen, lower alkyl, halogen, nitro, methoxy, methylthio, methylsulfonyl, -CF 3 , phenyl, phenoxy or lower alkoxycarbonyl; And n is an integer of 1 to 3. 제2항에 있어서, X가 할로겐, 저급 알콕시이고; Y가 수소 또는 염소이며; R이 수소 또는 Z가 수소, 저급 알킬, 할로겐, 니트로, 메톡시, 메틸티오, 메틸술포닐, -CF3또는 페녹시이며; 또 n이 1인 화합물.The compound of claim 2, wherein X is halogen, lower alkoxy; Y is hydrogen or chlorine; R is hydrogen or Z is hydrogen, lower alkyl, halogen, nitro, methoxy, methylthio, methylsulfonyl, -CF 3 or phenoxy; And n is 1; 제3항에 있어서, X가 염소 또는 불소이고; Y가 수소이며; R이 수소이고; Z가 수소, 4-F, 4-Cl 또는 4-CH3이며, 또 n이 1인 화합물.The compound of claim 3, wherein X is chlorine or fluorine; Y is hydrogen; R is hydrogen; Z is hydrogen, 4-F, 4-Cl or 4-CH 3 , and n is 1; 제4항에 있어서, 하기 화학식을 갖는 화합물.The compound of claim 4 having the formula 제4항에 있어서, 하기의 화학식을 갖는 화합물.The compound of claim 4 having the formula 하기 일반식(1)의 화합물을 함유하는 살진균제 또는 살균제 조성물:Fungicide or fungicide compositions containing the compound of formula (1): 상기식에서, X는 할로겐, 저급 알콕시, 저급 알킬티오, 니트로 또는 메틸이고; Y는 수소 또는 염소이며; R은 수소, 저급 알킬 또는 알릴이고; Z는 수소, 할로겐, 니트로, 메톡시, 메틸티오, 메틸술포닐, -CF3, 페닐, 페녹시 또는 저급 알콕시카보닐이며; 또 n은 1 내지 3의 정수이다.Wherein X is halogen, lower alkoxy, lower alkylthio, nitro or methyl; Y is hydrogen or chlorine; R is hydrogen, lower alkyl or allyl; Z is hydrogen, halogen, nitro, methoxy, methylthio, methylsulfonyl, -CF 3 , phenyl, phenoxy or lower alkoxycarbonyl; And n is an integer of 1 to 3. 제7항에 있어서, X가 할로겐, 저급 알콕시 또는 메틸티오이고; Y가 수소 또는 염소이며; R이 수소, 저급 알킬 또는 알릴이고; Z가 수소, 저급 알킬, 할로겐, 니트로, 메톡시, 메틸티오, 메틸술포닐, -CF3, 페닐, 페녹시, 또는 저급 알콕시카보닐이며; 또 n이 1 내지 3의 정수인 살진균제 또는 살균제 조성물.8. A compound according to claim 7, wherein X is halogen, lower alkoxy or methylthio; Y is hydrogen or chlorine; R is hydrogen, lower alkyl or allyl; Z is hydrogen, lower alkyl, halogen, nitro, methoxy, methylthio, methylsulfonyl, -CF 3 , phenyl, phenoxy, or lower alkoxycarbonyl; And a fungicide or fungicide composition wherein n is an integer of 1 to 3. 제8항에 있어서, X가 할로겐 또는 저급 알콕시이고; Y가 수소 또는 염소이며; R이 수소이고; Z가 수소, 저급 알킬, 할로겐, 니트로, 메톡시, 메틸티오, 메틸술포닐, -CF3또는 페녹시이며; 또 n이 1인 살진균제 또는 살균제 조성물.The compound of claim 8, wherein X is halogen or lower alkoxy; Y is hydrogen or chlorine; R is hydrogen; Z is hydrogen, lower alkyl, halogen, nitro, methoxy, methylthio, methylsulfonyl, -CF 3 or phenoxy; And n is 1 or a fungicide or bactericide composition. 제9항에 있어서, X가 염소 또는 플루오로이고; Y가 수소이며; R이 수소이고; Z가 수소, 4-F, 4-Cl 또는 4-CH3이며; n이 1인 살진균제 또는 살균제 조성물.The compound of claim 9, wherein X is chlorine or fluoro; Y is hydrogen; R is hydrogen; Z is hydrogen, 4-F, 4-Cl or 4-CH 3 ; Fungicide or fungicide composition wherein n is 1. 제10항에 있어서, 활성성분이 하기 화학식으로 표시되는 살진균제 또는 살균제 조성물.The fungicide or fungicide composition according to claim 10, wherein the active ingredient is represented by the following formula. 제10항에 있어서, 활성성분의 하기 화학식으로 표시되는 살진균제 또는 살균제 조성물.The fungicide or fungicide composition according to claim 10, represented by the following formula of the active ingredient. 일반식(1)의 화합물을 살진균 또는 살균유효용량으로 토양 또는 작물에 투여함으로써 진균 또는 세균에 의해 야기되는 농작물 또는 원예작물의 질병을 예방하는 방법.A method for preventing diseases of crops or horticultural crops caused by fungi or bacteria by administering a compound of formula (1) to soil or crops at an effective or fungicidal dose. 상기 식에서, X는 할로겐, 저급 알콕시, 저급 알킬티오, 니트로 또는 메틸이고; Y는 수소 또는 염소이며; R은 수소, 저급 알킬 또는 알릴이고; Z는 수소, 저급 알킬, 할로겐, 니트로, 메톡시, 메틸티오, 메틸술포닐, -CF3, 페닐, 페녹시 또는 저급 알콕시카보닐이며; 또 n은 1 내지 3의 정수이다.Wherein X is halogen, lower alkoxy, lower alkylthio, nitro or methyl; Y is hydrogen or chlorine; R is hydrogen, lower alkyl or allyl; Z is hydrogen, lower alkyl, halogen, nitro, methoxy, methylthio, methylsulfonyl, -CF 3 , phenyl, phenoxy or lower alkoxycarbonyl; And n is an integer of 1 to 3. 제13항에 있어서, X가 할로겐, 저급 알콕시 또는 메틸티오이고; Y가 수소 또는 염소이며; R이 수소, 저급 알킬 또는 알킬이고; Z가 수소, 저급 알킬, 할로겐, 니트로, 메톡시, 메틸티오, 메틸술포닐, -CF3, 페닐, 페녹시 또는 저급 알콕시카보닐이며; 또 n이 1 내지 3의 정수인 방법.The compound of claim 13, wherein X is halogen, lower alkoxy or methylthio; Y is hydrogen or chlorine; R is hydrogen, lower alkyl or alkyl; Z is hydrogen, lower alkyl, halogen, nitro, methoxy, methylthio, methylsulfonyl, -CF 3 , phenyl, phenoxy or lower alkoxycarbonyl; And n is an integer of 1 to 3. 제14항에 있어서, X가 할로겐 또는 저급 알콕시이고; Y가 수소 또는 염소이며; R이 수소이고; Z가 수소, 저급 알킬, 할로겐, 니트로, 메틸시, 메틸티오, 메틸술포닐, -CF3또는 페녹시이며 또 n이 1인 방법.15. The compound of claim 14, wherein X is halogen or lower alkoxy; Y is hydrogen or chlorine; R is hydrogen; Z is hydrogen, lower alkyl, halogen, nitro, methylcy, methylthio, methylsulfonyl, -CF 3 or phenoxy and n is 1; 제15항에 있어서, X가 염소 또는 플루오로이고; Y가 수소이며; R이 수소이며; Z가 수소, 4-F, 4-Cl 또는 4-CH3이고; 또 n이 1인 방법.The compound of claim 15, wherein X is chlorine or fluoro; Y is hydrogen; R is hydrogen; Z is hydrogen, 4-F, 4-Cl or 4-CH 3 ; And n is one. 제16항에 있어서, 활성 성분이 하기 화학식으로 표시되는 방법.The method of claim 16 wherein the active ingredient is represented by the formula: 제16항에 있어서, 활성 성분이 하기 화학식으로 표시되는 방법.The method of claim 16 wherein the active ingredient is represented by the formula: 불활성 용매 내에서, 경우에 따라 산 결합제의 존재하에, 일반식(2)의 화합물을(3)의 화합물과 반응시켜 이루어지는 일반식(1)화합물의 제조방법.A method for producing a compound of formula (1), wherein the compound of formula (2) is reacted with the compound of (3), optionally in the presence of an acid binder, in an inert solvent. 상기 식에서, X, Y, R, Z 및 n은 상기 정의한 바와 같다.Wherein X, Y, R, Z and n are as defined above. 불활성 용매 내에서 또는 과량의 일반식(5) 화합물 내에서, 일반식(4)의 화합물을 일반식(5)의 화합물과 반응시켜 이루어지는 일반식(1)화합물의 제조방법.A method for producing a compound of formula (1), wherein the compound of formula (4) is reacted with a compound of formula (5) in an inert solvent or in an excess of compound of formula (5). 상기 식에서, X, Y, Z 및 n은 상기 정의한 바와 같고, R은 수소이다.Wherein X, Y, Z and n are as defined above and R is hydrogen. 불활성 용매 내에서 또는 용매없이, 염기 존재하에 일반식(6)의 화합물을 일반식(7)의 화합물과 반응시켜 이루어지는 일반식(1) 화합물의 제조방법.A process for preparing a compound of formula (1), wherein the compound of formula (6) is reacted with a compound of formula (7) in the presence of a base in an inert solvent or without a solvent. 상기 식에서, X, Y, Z, n 및 R은 상기 정의한 바와 같고, R″은 알킬 또는 아릴이다.Wherein X, Y, Z, n and R are as defined above and R " is alkyl or aryl. 불활성 용매 중의 염기 존재하에, 일반식(8)의 화합물을 일반식(9)의 화합물과 반응시켜 이루어지는 일반식(1) 화합물의 제조방법.A method for producing a compound of formula (1), wherein the compound of formula (8) is reacted with a compound of formula (9) in the presence of a base in an inert solvent. 상기 식에서, X, Y, Z 및 n은 상기 정의한 바와 같고; R은 저급 알킬 또는 알릴이며; Q는 할로겐이다.Wherein X, Y, Z and n are as defined above; R is lower alkyl or allyl; Q is halogen. ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.※ Note: The disclosure is based on the initial application.
KR1019860008017A 1985-09-25 1986-09-25 N-phenylsulfonylisonicotinamide derivative KR870003073A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP210097 1985-09-25
JP21009785 1985-09-25
JP68734 1986-03-28
JP61068734A JPS62161761A (en) 1985-09-25 1986-03-28 N-phenylsulfonylisonicotinamide derivative and agricultural and horticultural fungicide composition containing said derivative as active component

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KR870003073A true KR870003073A (en) 1987-04-14

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AR031130A1 (en) * 2000-09-20 2003-09-10 Abbott Lab PROMOTING N-ACILSULFONAMIDS OF APOPTOSIS

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