KR850005423A - 아졸일-3- 치환된 부탄 유도체의 제조방법 - Google Patents

아졸일-3- 치환된 부탄 유도체의 제조방법 Download PDF

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KR850005423A
KR850005423A KR1019850000146A KR850000146A KR850005423A KR 850005423 A KR850005423 A KR 850005423A KR 1019850000146 A KR1019850000146 A KR 1019850000146A KR 850000146 A KR850000146 A KR 850000146A KR 850005423 A KR850005423 A KR 850005423A
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methyl
group
triazol
formula
compound
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KR1019850000146A
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English (en)
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요시오 구라하시 (외 4)
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다떼노 고자부로
니혼 도꾸슈 노야꾸 세이조 가부시끼 가이샤
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Application filed by 다떼노 고자부로, 니혼 도꾸슈 노야꾸 세이조 가부시끼 가이샤 filed Critical 다떼노 고자부로
Publication of KR850005423A publication Critical patent/KR850005423A/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C07C45/70—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form
    • C07C45/71—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form being hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/20—Unsaturated compounds containing keto groups bound to acyclic carbon atoms
    • C07C49/255—Unsaturated compounds containing keto groups bound to acyclic carbon atoms containing ether groups, groups, groups, or groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

내용 없음

Description

아졸일-3-치환된 부탄 유도체의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (12)

  1. 일반식(Ⅱ)의 화합물과 일반식(Ⅲ)의 화합물을 반응시키고, 필요하다면 수득된 일반식(Ia)의 화합물을 환원체를 사용하여 환원시킴을 특징으로하여, 일반식(Ⅰ)의 아졸일 -3-치환된 부탄 유도체를 제조하는 방법.
    상기식에서, Ar은 할로겐에 의해 치환될 수 있는 페닐기이며, R¹은 알킬 또는 페닐기이며, X는 -CH(OH)-또는-CO-기이며, Az는 1-이미다졸일 또는 1,2,4-트리아졸-1-일기이며, R²는 알킬기, 시클로알킬기 또는 할로겐 원자, 저급알킬기 및 임의로 할로겐 치환된 페닐기에 의해 치환될 수 있는 페닐기이며, Hal은 할로겐원자이다.
  2. 제1항에 있어서,Ar이 불소, 염소 또는 브롬에 의해 치환될 수 있는 페닐기이며, R¹이 메틸 또는 페닐기이며, X가 -CH(CH)-또는-CO-기이며, Az가, 1-이미다졸일 또는 1,2,4-트리아졸일기이며, R²가 1내지 4의 탄소 원자를 갖는 알킬기,5내지 6의 탄소원자를 갖는 시클로알킬기 또는 불소, 염소 또는 브롬, 메틸, 에틸, 프로필 또는 부틸기, 또는 염소에 의해 치환될 수 있는 페닐기에 의해 치환될 수 있는 페닐기인 일반식(Ⅰ)의 화합물의 제조방법.
  3. 제1항에 있어서, 하기 구조식의 1-(4-클로로페녹시)-1-(1,2,4-트리아졸-1-일)-3-메틸-3-페닐-부탄-2-온의 제조방법
  4. 제1항에 있어서, 하기 구조식의 1-페녹시-1-(1,2,4-트리아졸-1-일)-3-메틸-3-(2-클로로페닐)-부탄-2-온의 제조방법.
  5. 제1항에 있어서, 하기 구조식의 1-(4-클로로페녹시)-1-(1,2,4-트리아졸-1-일)-3-메틸-3-(3-클로로페닐)-부탄-2-온의 제조방법.
  6. 제1항에 있어서, 하기 구조식의 1-(4-클로로페녹시)-1-(1-이미다졸일)-3-메틸-3-페닐-부탄-2-온의 제조방법.
  7. 제1항에 있어서, 하기 구조식의 1-(4-클로로페녹시)-1-(1,2,4-트리아졸-1-일)-3-메틸-3-페닐-부탄-2-올의 제조방법.
  8. 제1항에 있어서, 하기 구조식의 1-(4-클로로페녹시)-1-(1,2,4-트리아졸-1-일)-3-메틸-3-(3-클로로페닐)-부탄-2-올의 제조방법.
  9. 제1항에 있어서, 하기 구조식의 1-(4-클로로페녹시)-1-(1-이미다졸일)-3-메틸-3-(4-클로로페닐)-부탄-2-올의 제조방법.
  10. 제1항에 있어서, 하기 구조식의 1-페녹시-1-(1,2,4-트리아졸-1-일)-3,3-디페닐-부탄-2-온의 제조방법.
  11. 제1항에 있어서, 하기 구조식의 1-페녹시-1-(1,2,3-트리아졸-1-일)-3,3-디페닐-부탄-2-올의 제조방법.
  12. 제1항에 있어서, 하기 구조식의 1-(4-페닐페녹시)-1-(1,2,4-트리아졸-1-일)-3-메틸-3-(4-클로로페닐)-부탄-2-온의 제조방법.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019850000146A 1984-01-12 1985-01-11 아졸일-3- 치환된 부탄 유도체의 제조방법 KR850005423A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP59002683A JPS60146875A (ja) 1984-01-12 1984-01-12 アゾリル−３位−置換ブタン誘導体，その製法及び農園芸用殺菌剤
JP???59-2683? 1984-01-12

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KR850005423A true KR850005423A (ko) 1985-08-26

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EP (1) EP0150499A2 (ko)
JP (1) JPS60146875A (ko)
KR (1) KR850005423A (ko)
BR (1) BR8500126A (ko)
DK (1) DK14785A (ko)
HU (1) HUT36673A (ko)
IL (1) IL74025A0 (ko)
ZA (1) ZA85261B (ko)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0206523B1 (en) * 1985-06-18 1991-12-04 Imperial Chemical Industries Plc Heterocyclic compounds as fungicides
DE3751686T2 (de) * 1986-12-16 1996-06-13 Zeneca Ltd Pyrrol-Derivate und ihre Verwendung in der Landwirtschaft

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JPH0518829B2 (ko) 1993-03-15
HUT36673A (en) 1985-10-28
IL74025A0 (en) 1985-04-30
BR8500126A (pt) 1985-08-20
ZA85261B (en) 1985-09-25
JPS60146875A (ja) 1985-08-02
EP0150499A2 (de) 1985-08-07
DK14785A (da) 1985-07-13
DK14785D0 (da) 1985-01-11

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