KR850000978B1 - Omt에스테르 유도체의 제조방법 - Google Patents

Omt에스테르 유도체의 제조방법 Download PDF

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Publication number
KR850000978B1
KR850000978B1 KR8205595A KR820005595A KR850000978B1 KR 850000978 B1 KR850000978 B1 KR 850000978B1 KR 8205595 A KR8205595 A KR 8205595A KR 820005595 A KR820005595 A KR 820005595A KR 850000978 B1 KR850000978 B1 KR 850000978B1
Authority
KR
South Korea
Prior art keywords
omt
acid
optionally substituted
hydrogen
solution
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
KR8205595A
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English (en)
Korean (ko)
Other versions
KR840002855A (ko
Inventor
안드류 커스트 허버트
Original Assignee
아더 알. 웨일
일라이 릴리 앤드 캄파니
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 아더 알. 웨일, 일라이 릴리 앤드 캄파니 filed Critical 아더 알. 웨일
Publication of KR840002855A publication Critical patent/KR840002855A/ko
Application granted granted Critical
Publication of KR850000978B1 publication Critical patent/KR850000978B1/ko
Expired legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
KR8205595A 1981-12-14 1982-12-14 Omt에스테르 유도체의 제조방법 Expired KR850000978B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/330,341 US4401660A (en) 1981-12-14 1981-12-14 Ester derivatives of 5-O-mycaminosyl tylonolide and method of using same
US330341 2006-01-12

Publications (2)

Publication Number Publication Date
KR840002855A KR840002855A (ko) 1984-07-21
KR850000978B1 true KR850000978B1 (ko) 1985-07-05

Family

ID=23289335

Family Applications (1)

Application Number Title Priority Date Filing Date
KR8205595A Expired KR850000978B1 (ko) 1981-12-14 1982-12-14 Omt에스테르 유도체의 제조방법

Country Status (12)

Country Link
US (1) US4401660A (enExample)
EP (1) EP0082003B1 (enExample)
JP (1) JPS58110598A (enExample)
KR (1) KR850000978B1 (enExample)
CA (1) CA1189503A (enExample)
DE (1) DE3268461D1 (enExample)
DK (2) DK153794C (enExample)
GB (1) GB2111497B (enExample)
GR (1) GR77094B (enExample)
HU (1) HU194268B (enExample)
IE (1) IE54283B1 (enExample)
IL (1) IL67452A (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU551142B2 (en) * 1981-07-09 1986-04-17 Zaidan Hojin Biseibutsu Kagaku Kenkyukai Tylosin derivatives
CA1196915A (en) * 1982-01-22 1985-11-19 Hideo Sakakibara 23-0-acyl-23-demycinosyldesmycosin
US4443436A (en) 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin
US4629786A (en) * 1983-02-28 1986-12-16 Eli Lilly And Company C-20- and C-23 modified macrolide derivatives
GB8333624D0 (en) * 1983-12-16 1984-01-25 Lepetit Spa Antibiotics l 17054 and l 17392
US4576931A (en) * 1985-04-03 1986-03-18 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai (Microbial Chemistry Research Foundation) 23-C-Substituted mycaminosyl tylonolide, pharmaceutical compositions and method of use

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE667952A (enExample) * 1964-08-05
US4092473A (en) * 1975-08-01 1978-05-30 Sanraku Ocean Co., Ltd. Tylosin derivatives and their manufacturing process
US4321362A (en) * 1980-06-12 1982-03-23 Eli Lilly And Company De(mycinosyloxy)tylosin and process for its production
US4438109A (en) * 1980-07-25 1984-03-20 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai Tylosin derivatives
US4299953A (en) * 1980-07-29 1981-11-10 Eli Lilly And Company Mycarosyltylactone

Also Published As

Publication number Publication date
DK553982A (da) 1983-06-15
US4401660A (en) 1983-08-30
KR840002855A (ko) 1984-07-21
DK623786A (da) 1986-12-22
GR77094B (enExample) 1984-09-06
EP0082003B1 (en) 1986-01-08
GB2111497A (en) 1983-07-06
DK623786D0 (da) 1986-12-22
IE54283B1 (en) 1989-08-16
HU194268B (en) 1988-01-28
JPS58110598A (ja) 1983-07-01
EP0082003A1 (en) 1983-06-22
IL67452A0 (en) 1983-05-15
DK153794C (da) 1989-02-20
IL67452A (en) 1985-12-31
IE822952L (en) 1983-06-14
GB2111497B (en) 1985-10-30
DK153794B (da) 1988-09-05
CA1189503A (en) 1985-06-25
DE3268461D1 (de) 1986-02-20

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