KR830005120A - Method for preparing 1- (acylamino-aryloxy) -2-hydroxy-3-alkynyl-aminopropane - Google Patents

Method for preparing 1- (acylamino-aryloxy) -2-hydroxy-3-alkynyl-aminopropane Download PDF

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Publication number
KR830005120A
KR830005120A KR1019810000749A KR810000749A KR830005120A KR 830005120 A KR830005120 A KR 830005120A KR 1019810000749 A KR1019810000749 A KR 1019810000749A KR 810000749 A KR810000749 A KR 810000749A KR 830005120 A KR830005120 A KR 830005120A
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South Korea
Prior art keywords
general formula
following general
preparing
carbon atoms
group
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KR1019810000749A
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Korean (ko)
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KR850000698B1 (en
Inventor
쾨페 헤르베르트
쿰머 베르너
쉬텔 헬무트
무아세픽 고코
트라우네커 베르너
Original Assignee
기젤라 벨만 · 오토 핀케
쎄. 하 베링거 존
오토 핀케
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Priority to KR1019810000749A priority Critical patent/KR850000698B1/en
Publication of KR830005120A publication Critical patent/KR830005120A/en
Priority to KR1019850000421A priority patent/KR850000697B1/en
Priority to KR1019850000420A priority patent/KR850000696B1/en
Application granted granted Critical
Publication of KR850000698B1 publication Critical patent/KR850000698B1/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

내용 없음No content

Description

1-(아실아미노-아릴옥시)-2-하이드록시-3-알키닐-아미노프로판의 제조방법Method for preparing 1- (acylamino-aryloxy) -2-hydroxy-3-alkynyl-aminopropane

본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음As this is a public information case, the full text was not included.

Claims (1)

다음 일반식(Ⅱ)화합물은 다음 일반식(Ⅲ)의 아민과 반응시키거나 다음 일반식(Ⅳ)의 옥사졸리딘 유도체를 가수분해하거나 다음 일반식(Ⅴ)화합물(또는 이의 염)을 다음 일반식(Ⅵ)의 아세티디놀 유도체와 반응시킴을 특징으로 하여 다음 일반식(Ⅰ)화합물 및 이의 생리학적으로 무독한 산부가염의 제조방법.The following general formula (II) compound is reacted with an amine of the following general formula (III) or hydrolyzes an oxazolidine derivative of the following general formula (IV) or the following general formula (V) compound (or salt thereof) A method for preparing the following general formula (I) compounds and their physiologically toxic acid addition salts, characterized in that it reacts with an acetidinol derivative of formula (VI). 상기 일반식에서In the above general formula R1은 에틸 또는 이소프로필 그룹이고R 1 is an ethyl or isopropyl group R2는 수소 또는 할로겐원자, 탄소수 1 내지 4의 알킬 또는 알콕시 그룹이거나 C-위치에서의 유리 원자가 결합을 가진 2가 그룹 -CH=CH-CH=OH 또는 (CH2)n(n=3 내지 5의 정수)이고R 2 is hydrogen or a halogen atom, an alkyl or alkoxy group having 1 to 4 carbon atoms or a divalent group having a free valence bond at the C-position —CH═CH—CH═OH or (CH 2 ) n (n = 3 to Is an integer of 5) R3는 수소 또는 탄소수 1 내지 3의 알킬 그룹이고R 3 is hydrogen or an alkyl group having 1 to 3 carbon atoms R4는 탄소수 1 내지 3의 알킬그룹 또는 R3와 함께 (CH2)p(p는 4 내지 6의 정수)이고R 4 is (CH 2 ) p (p is an integer of 4 to 6) together with an alkyl group having 1 to 3 carbon atoms or R 3 또는 -CHOH-CH2-할(할=할로겐)이고 Or -CHOH-CH 2 -hal (hal = halogen) X는 -CO-, -CH2- 또는 -CH-저급알킬 그룹이다.X is a -CO-, -CH 2 -or -CH-lower alkyl group. ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.※ Note: The disclosure is based on the initial application.
KR1019810000749A 1981-03-07 1981-03-07 Process for preparing 1-(acylamino-aryloxy)-2-hydroxy-3-alkinyl-aminopropanes KR850000698B1 (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
KR1019810000749A KR850000698B1 (en) 1981-03-07 1981-03-07 Process for preparing 1-(acylamino-aryloxy)-2-hydroxy-3-alkinyl-aminopropanes
KR1019850000421A KR850000697B1 (en) 1981-03-07 1985-01-24 Process for preparing 1-(acylamino-aryloxy)-2-hydroxy-3-alkinyl-aminopropanes
KR1019850000420A KR850000696B1 (en) 1981-03-07 1985-01-24 Process for preparing 1-(acylamino-aryloxy)-2-hydroxy-3-alkinyl-aminopropanes

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
KR1019810000749A KR850000698B1 (en) 1981-03-07 1981-03-07 Process for preparing 1-(acylamino-aryloxy)-2-hydroxy-3-alkinyl-aminopropanes

Related Child Applications (2)

Application Number Title Priority Date Filing Date
KR1019850000421A Division KR850000697B1 (en) 1981-03-07 1985-01-24 Process for preparing 1-(acylamino-aryloxy)-2-hydroxy-3-alkinyl-aminopropanes
KR1019850000420A Division KR850000696B1 (en) 1981-03-07 1985-01-24 Process for preparing 1-(acylamino-aryloxy)-2-hydroxy-3-alkinyl-aminopropanes

Publications (2)

Publication Number Publication Date
KR830005120A true KR830005120A (en) 1983-07-23
KR850000698B1 KR850000698B1 (en) 1985-05-15

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Application Number Title Priority Date Filing Date
KR1019810000749A KR850000698B1 (en) 1981-03-07 1981-03-07 Process for preparing 1-(acylamino-aryloxy)-2-hydroxy-3-alkinyl-aminopropanes

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KR850000698B1 (en) 1985-05-15

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