KR20220044269A - Glp-1 작용제, sglt2 억제제, 및 n-(8-(2-하이드록시벤조일)아미노)카프릴산의 염을 포함하는 고형분 조성물 - Google Patents

Glp-1 작용제, sglt2 억제제, 및 n-(8-(2-하이드록시벤조일)아미노)카프릴산의 염을 포함하는 고형분 조성물 Download PDF

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KR20220044269A
KR20220044269A KR1020227001918A KR20227001918A KR20220044269A KR 20220044269 A KR20220044269 A KR 20220044269A KR 1020227001918 A KR1020227001918 A KR 1020227001918A KR 20227001918 A KR20227001918 A KR 20227001918A KR 20220044269 A KR20220044269 A KR 20220044269A
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glp
ethoxy
agonist
composition
salt
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Korean (ko)
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베티 롬스테인 페더센
비르지트 니센
패트릭 윌리엄 가리바이
카이사 나엘라파
안드레아스 베제
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노보 노르디스크 에이/에스
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    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/7056—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing five-membered rings with nitrogen as a ring hetero atom
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    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

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  • Child & Adolescent Psychology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicinal Preparation (AREA)
KR1020227001918A 2019-08-07 2020-08-06 Glp-1 작용제, sglt2 억제제, 및 n-(8-(2-하이드록시벤조일)아미노)카프릴산의 염을 포함하는 고형분 조성물 Withdrawn KR20220044269A (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP19190623.9 2019-08-07
EP19190623 2019-08-07
EP20172415 2020-04-30
EP20172415.0 2020-04-30
PCT/EP2020/072106 WO2021023811A1 (en) 2019-08-07 2020-08-06 Solid compositions comprising a glp-1 agonist, an sglt2 inhibitor and a salt of n-(8-(2-hydroxybenzoyl)amino)caprylic acid

Publications (1)

Publication Number Publication Date
KR20220044269A true KR20220044269A (ko) 2022-04-07

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KR1020227001918A Withdrawn KR20220044269A (ko) 2019-08-07 2020-08-06 Glp-1 작용제, sglt2 억제제, 및 n-(8-(2-하이드록시벤조일)아미노)카프릴산의 염을 포함하는 고형분 조성물

Country Status (16)

Country Link
US (1) US20220265777A1 (https=)
EP (1) EP4009941A1 (https=)
JP (1) JP2022545156A (https=)
KR (1) KR20220044269A (https=)
CN (1) CN114173766A (https=)
AU (1) AU2020325708A1 (https=)
BR (1) BR112022000490A2 (https=)
CA (1) CA3144611A1 (https=)
CL (1) CL2022000137A1 (https=)
CO (1) CO2022000578A2 (https=)
IL (1) IL289504A (https=)
MX (1) MX2022000827A (https=)
PE (1) PE20220751A1 (https=)
PH (1) PH12022550007A1 (https=)
TW (1) TW202114730A (https=)
WO (1) WO2021023811A1 (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2025143830A1 (ko) * 2023-12-28 2025-07-03 주식회사 대웅제약 이나보글리플로진와 저용량 리라글루타이드의 항비만 병용 요법

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI797133B (zh) * 2017-06-09 2023-04-01 丹麥商諾佛 儂迪克股份有限公司 用於經口投予的固體組成物
JP6898518B2 (ja) * 2018-02-02 2021-07-07 ノヴォ ノルディスク アー／エス Ｇｌｐ−１アゴニスト、ｎ−（８−（２−ヒドロキシベンゾイル）アミノ）カプリル酸の塩及び滑沢剤を含む固形組成物
WO2022268214A1 (zh) * 2021-06-25 2022-12-29 甘李药业股份有限公司 Pcsk9抑制剂和glp-1受体激动剂的药物组合
WO2023065231A1 (en) * 2021-10-21 2023-04-27 Guangzhou Dazhou Biomedicine Ltd. Oral delivery of therapeutic agents
CN114085203A (zh) * 2021-12-17 2022-02-25 宁波高新区美诺华医药创新研究院有限公司 达格列净组合物
CN118742326A (zh) * 2021-12-29 2024-10-01 广州大洲生物医药科技有限公司 口服递送
CN116370609B (zh) * 2023-06-01 2023-08-15 北京普诺旺康医药科技有限公司 包含血管活性肠肽和吸收增强剂的固体组合物

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20130035281A1 (en) * 2011-02-09 2013-02-07 Boehringer Ingelheim International Gmbh Pharmaceutical composition, methods for treating and uses thereof
CN105503802A (zh) * 2016-01-15 2016-04-20 中山大学 一种达格列净-柠檬酸共晶的制备方法
WO2018124497A1 (ko) * 2016-12-30 2018-07-05 한미약품 주식회사 다파글리플로진 l-프롤린과 항당뇨병제를 포함하는 약제학적 복합 제제
TWI797133B (zh) * 2017-06-09 2023-04-01 丹麥商諾佛 儂迪克股份有限公司 用於經口投予的固體組成物

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2025143830A1 (ko) * 2023-12-28 2025-07-03 주식회사 대웅제약 이나보글리플로진와 저용량 리라글루타이드의 항비만 병용 요법

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PE20220751A1 (es) 2022-05-10
TW202114730A (zh) 2021-04-16
JP2022545156A (ja) 2022-10-26
WO2021023811A1 (en) 2021-02-11
CA3144611A1 (en) 2021-02-11
US20220265777A1 (en) 2022-08-25
CN114173766A (zh) 2022-03-11
IL289504A (en) 2022-02-01
EP4009941A1 (en) 2022-06-15
CO2022000578A2 (es) 2022-04-29
BR112022000490A2 (pt) 2022-03-08
MX2022000827A (es) 2022-02-16
PH12022550007A1 (en) 2022-11-21
CL2022000137A1 (es) 2022-10-07
AU2020325708A1 (en) 2022-02-03

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