KR20180100567A - 질 삽입식 에스트라디올 약제학적 조성물 및 방법 - Google Patents
질 삽입식 에스트라디올 약제학적 조성물 및 방법 Download PDFInfo
- Publication number
- KR20180100567A KR20180100567A KR1020187019331A KR20187019331A KR20180100567A KR 20180100567 A KR20180100567 A KR 20180100567A KR 1020187019331 A KR1020187019331 A KR 1020187019331A KR 20187019331 A KR20187019331 A KR 20187019331A KR 20180100567 A KR20180100567 A KR 20180100567A
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- South Korea
- Prior art keywords
- estradiol
- vaginal
- vva
- suppository
- administering
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
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- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
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- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
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- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
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- Pain & Pain Management (AREA)
- Medicinal Preparation (AREA)
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| US201562264309P | 2015-12-07 | 2015-12-07 | |
| US62/264,309 | 2015-12-07 | ||
| US201662296552P | 2016-02-17 | 2016-02-17 | |
| US62/296,552 | 2016-02-17 | ||
| US201662324838P | 2016-04-19 | 2016-04-19 | |
| US62/324,838 | 2016-04-19 | ||
| US201662329940P | 2016-04-29 | 2016-04-29 | |
| US62/329,940 | 2016-04-29 | ||
| US201662348820P | 2016-06-10 | 2016-06-10 | |
| US62/348,820 | 2016-06-10 | ||
| PCT/US2016/065466 WO2017100378A2 (en) | 2015-12-07 | 2016-12-07 | Vaginal inserted estradiol pharmaceutical compositions and methods |
Publications (1)
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| KR20180100567A true KR20180100567A (ko) | 2018-09-11 |
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| JP (2) | JP2018538290A (enExample) |
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| WO (1) | WO2017100378A2 (enExample) |
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| KR20220105717A (ko) | 2021-01-20 | 2022-07-28 | 주식회사 바이올렛드림 | 질 내 수용성 겔 조성물 |
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| US20220378697A1 (en) * | 2019-10-31 | 2022-12-01 | R.P. Scherer Technologies, Llc | Suppository capsule |
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| FR2739558B1 (fr) * | 1995-10-05 | 1997-11-28 | Innothera Lab Sa | Forme galenique unitaire pour hormonotherapie locale de la secheresse vaginale |
| US6117446A (en) * | 1999-01-26 | 2000-09-12 | Place; Virgil A. | Drug dosage unit for buccal administration of steroidal active agents |
| MX368189B (es) * | 2004-10-20 | 2019-09-23 | Endorecherche Inc | Precursores esteroides sexuales solos o en combinación con un modulador receptor de estrógeno selectivo y/o con estrógenos y/o con un inhibidor de fosfodiesterasa gmpc de tipo 5 para la prevención y tratamiento de sequedad vaginal y disfunción sexual en mujeres post-menopáusicas. |
| US10806697B2 (en) * | 2012-12-21 | 2020-10-20 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
| PL2861073T3 (pl) * | 2012-06-18 | 2021-09-27 | Therapeuticsmd, Inc. | Rozpuszczalna kapsułka estradiolu do wprowadzania do pochwy |
| US9180091B2 (en) * | 2012-12-21 | 2015-11-10 | Therapeuticsmd, Inc. | Soluble estradiol capsule for vaginal insertion |
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2016
- 2016-12-07 JP JP2018529574A patent/JP2018538290A/ja active Pending
- 2016-12-07 AU AU2016366200A patent/AU2016366200B2/en not_active Ceased
- 2016-12-07 EP EP16873806.0A patent/EP3386514A4/en not_active Withdrawn
- 2016-12-07 BR BR112018011483A patent/BR112018011483A2/pt not_active Application Discontinuation
- 2016-12-07 MX MX2018006882A patent/MX384850B/es unknown
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| KR20220105717A (ko) | 2021-01-20 | 2022-07-28 | 주식회사 바이올렛드림 | 질 내 수용성 겔 조성물 |
Also Published As
| Publication number | Publication date |
|---|---|
| BR112018011483A2 (pt) | 2018-12-04 |
| MX384850B (es) | 2025-03-14 |
| EP3386514A4 (en) | 2019-07-24 |
| JP2018538290A (ja) | 2018-12-27 |
| WO2017100378A3 (en) | 2018-02-22 |
| EP3386514A2 (en) | 2018-10-17 |
| WO2017100378A2 (en) | 2017-06-15 |
| AU2016366200A1 (en) | 2018-06-28 |
| IL259884A (en) | 2018-07-31 |
| AU2016366200B2 (en) | 2022-10-20 |
| CA3007636A1 (en) | 2017-06-15 |
| MX2018006882A (es) | 2019-05-16 |
| JP2021119155A (ja) | 2021-08-12 |
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