KR20080110837A - 아데노신 수용체 활성화제로서의 퓨린 유도체 - Google Patents
아데노신 수용체 활성화제로서의 퓨린 유도체 Download PDFInfo
- Publication number
- KR20080110837A KR20080110837A KR1020087025546A KR20087025546A KR20080110837A KR 20080110837 A KR20080110837 A KR 20080110837A KR 1020087025546 A KR1020087025546 A KR 1020087025546A KR 20087025546 A KR20087025546 A KR 20087025546A KR 20080110837 A KR20080110837 A KR 20080110837A
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- South Korea
- Prior art keywords
- compound
- purin
- mmol
- formula
- diphenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 108050000203 Adenosine receptors Proteins 0.000 title 1
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- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
- C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Diabetes (AREA)
- Neurology (AREA)
- Physical Education & Sports Medicine (AREA)
- Hematology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Rheumatology (AREA)
- Ophthalmology & Optometry (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Vascular Medicine (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Immunology (AREA)
- Otolaryngology (AREA)
- Gastroenterology & Hepatology (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0607945.3 | 2006-04-21 | ||
| GBGB0607945.3A GB0607945D0 (en) | 2006-04-21 | 2006-04-21 | Organic compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20080110837A true KR20080110837A (ko) | 2008-12-19 |
Family
ID=36581042
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020087025546A Withdrawn KR20080110837A (ko) | 2006-04-21 | 2007-04-19 | 아데노신 수용체 활성화제로서의 퓨린 유도체 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20090281127A1 (enExample) |
| EP (1) | EP2018382A2 (enExample) |
| JP (1) | JP2009534335A (enExample) |
| KR (1) | KR20080110837A (enExample) |
| CN (1) | CN101421271A (enExample) |
| AU (1) | AU2007241340A1 (enExample) |
| BR (1) | BRPI0710484A2 (enExample) |
| CA (1) | CA2648810A1 (enExample) |
| GB (1) | GB0607945D0 (enExample) |
| MX (1) | MX2008013522A (enExample) |
| RU (1) | RU2008145714A (enExample) |
| WO (1) | WO2007121917A2 (enExample) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GT200500281A (es) | 2004-10-22 | 2006-04-24 | Novartis Ag | Compuestos organicos. |
| GB0500785D0 (en) * | 2005-01-14 | 2005-02-23 | Novartis Ag | Organic compounds |
| GB0607950D0 (en) | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| GB0607948D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| GB0607953D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| GB0607944D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| AR060607A1 (es) | 2006-04-21 | 2008-07-02 | Novartis Ag | Derivados de purina,composiciones farmaceuticas que los contienen, metodo de preparacion y usos en enfermedades obstructivas o inflamatorias de las vias respiratorias. |
| GB0607954D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| EP1889846A1 (en) | 2006-07-13 | 2008-02-20 | Novartis AG | Purine derivatives as A2a agonists |
| EP1903044A1 (en) * | 2006-09-14 | 2008-03-26 | Novartis AG | Adenosine Derivatives as A2A Receptor Agonists |
| KR20090087054A (ko) * | 2006-11-10 | 2009-08-14 | 노파르티스 아게 | 시클로펜텐 디올 모노아세테이트 유도체 |
| US20100197914A1 (en) * | 2007-10-17 | 2010-08-05 | Robin Alec Fairhurst | Purine Derivatives as Adenosine Al Receptor Ligands |
| US20090181934A1 (en) * | 2007-10-17 | 2009-07-16 | Novartis Ag | Organic Compounds |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2264826T3 (es) * | 1998-10-16 | 2007-01-16 | Pfizer Inc. | Derivados de adenina. |
| US20040162422A1 (en) * | 2001-03-20 | 2004-08-19 | Adrian Hall | Chemical compounds |
| GT200500281A (es) * | 2004-10-22 | 2006-04-24 | Novartis Ag | Compuestos organicos. |
| GB0500785D0 (en) * | 2005-01-14 | 2005-02-23 | Novartis Ag | Organic compounds |
| DK1848718T3 (da) * | 2005-02-04 | 2012-08-27 | Millennium Pharm Inc | E1 aktiveringsenzymhæmmere |
| PT1989206E (pt) * | 2006-02-02 | 2012-10-15 | Millennium Pharm Inc | Inibidores da enzima de ativação e1 |
| GB0607948D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| GB0607953D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| GB0607944D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| GB0607954D0 (en) * | 2006-04-21 | 2006-05-31 | Novartis Ag | Organic compounds |
| US8008307B2 (en) * | 2006-08-08 | 2011-08-30 | Millennium Pharmaceuticals, Inc. | Heteroaryl compounds useful as inhibitors of E1 activating enzymes |
| US20090181934A1 (en) * | 2007-10-17 | 2009-07-16 | Novartis Ag | Organic Compounds |
-
2006
- 2006-04-21 GB GBGB0607945.3A patent/GB0607945D0/en not_active Ceased
-
2007
- 2007-04-19 US US12/297,007 patent/US20090281127A1/en not_active Abandoned
- 2007-04-19 MX MX2008013522A patent/MX2008013522A/es not_active Application Discontinuation
- 2007-04-19 KR KR1020087025546A patent/KR20080110837A/ko not_active Withdrawn
- 2007-04-19 EP EP07724369A patent/EP2018382A2/en not_active Withdrawn
- 2007-04-19 JP JP2009505776A patent/JP2009534335A/ja active Pending
- 2007-04-19 BR BRPI0710484-7A patent/BRPI0710484A2/pt not_active IP Right Cessation
- 2007-04-19 WO PCT/EP2007/003432 patent/WO2007121917A2/en not_active Ceased
- 2007-04-19 CN CNA2007800136743A patent/CN101421271A/zh active Pending
- 2007-04-19 RU RU2008145714/04A patent/RU2008145714A/ru not_active Application Discontinuation
- 2007-04-19 CA CA002648810A patent/CA2648810A1/en not_active Abandoned
- 2007-04-19 AU AU2007241340A patent/AU2007241340A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| EP2018382A2 (en) | 2009-01-28 |
| CN101421271A (zh) | 2009-04-29 |
| WO2007121917A2 (en) | 2007-11-01 |
| GB0607945D0 (en) | 2006-05-31 |
| RU2008145714A (ru) | 2010-05-27 |
| BRPI0710484A2 (pt) | 2011-08-16 |
| MX2008013522A (es) | 2008-10-29 |
| CA2648810A1 (en) | 2007-11-01 |
| WO2007121917A3 (en) | 2007-12-06 |
| US20090281127A1 (en) | 2009-11-12 |
| AU2007241340A1 (en) | 2007-11-01 |
| JP2009534335A (ja) | 2009-09-24 |
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Legal Events
| Date | Code | Title | Description |
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| PA0105 | International application |
Patent event date: 20081020 Patent event code: PA01051R01D Comment text: International Patent Application |
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| PG1501 | Laying open of application | ||
| PC1203 | Withdrawal of no request for examination | ||
| WITN | Application deemed withdrawn, e.g. because no request for examination was filed or no examination fee was paid |