KR20070048221A - 위장 장애 치료를 위한 프로스타글란딘 유도체 - Google Patents

위장 장애 치료를 위한 프로스타글란딘 유도체 Download PDF

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Publication number
KR20070048221A
KR20070048221A KR1020077004900A KR20077004900A KR20070048221A KR 20070048221 A KR20070048221 A KR 20070048221A KR 1020077004900 A KR1020077004900 A KR 1020077004900A KR 20077004900 A KR20077004900 A KR 20077004900A KR 20070048221 A KR20070048221 A KR 20070048221A
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KR
South Korea
Prior art keywords
halogen
alkyl
composition
aryl
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
KR1020077004900A
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English (en)
Korean (ko)
Inventor
류지 우에노
Original Assignee
수캄포 아게
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35229739&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR20070048221(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 수캄포 아게 filed Critical 수캄포 아게
Publication of KR20070048221A publication Critical patent/KR20070048221A/ko
Ceased legal-status Critical Current

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/94Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems condensed with rings other than six-membered or with ring systems containing such rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/557Eicosanoids, e.g. leukotrienes or prostaglandins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/557Eicosanoids, e.g. leukotrienes or prostaglandins
    • A61K31/558Eicosanoids, e.g. leukotrienes or prostaglandins having heterocyclic rings containing oxygen as the only ring hetero atom, e.g. thromboxanes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/10Laxatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nutrition Science (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
KR1020077004900A 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체 Ceased KR20070048221A (ko)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US60652104P 2004-09-02 2004-09-02
US60/606,521 2004-09-02
US66631705P 2005-03-30 2005-03-30
US60/666,317 2005-03-30
US66659305P 2005-03-31 2005-03-31
US60/666,593 2005-03-31

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1020137034994A Division KR20140019006A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체

Publications (1)

Publication Number Publication Date
KR20070048221A true KR20070048221A (ko) 2007-05-08

Family

ID=35229739

Family Applications (4)

Application Number Title Priority Date Filing Date
KR1020077004900A Ceased KR20070048221A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체
KR1020137034994A Ceased KR20140019006A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체
KR1020167036382A Ceased KR20170003712A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체
KR1020187008381A Ceased KR20180033310A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체

Family Applications After (3)

Application Number Title Priority Date Filing Date
KR1020137034994A Ceased KR20140019006A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체
KR1020167036382A Ceased KR20170003712A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체
KR1020187008381A Ceased KR20180033310A (ko) 2004-09-02 2005-09-01 위장 장애 치료를 위한 프로스타글란딘 유도체

Country Status (16)

Country Link
US (2) US8748481B2 (https=)
EP (1) EP1791545B1 (https=)
JP (4) JP2008511541A (https=)
KR (4) KR20070048221A (https=)
CN (1) CN102885821A (https=)
AR (1) AR050626A1 (https=)
AU (1) AU2005278323B2 (https=)
BR (1) BRPI0514891A (https=)
CA (1) CA2577284A1 (https=)
ES (1) ES2603381T3 (https=)
IL (1) IL181332A (https=)
MX (1) MX2007002602A (https=)
NO (1) NO340989B1 (https=)
NZ (1) NZ553434A (https=)
TW (1) TWI387454B (https=)
WO (1) WO2006025599A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ539582A (en) * 2002-10-23 2007-07-27 Sucampo Ag Prostaglandin compounds for the treatment of obesity
DE602004030245D1 (de) * 2003-07-03 2011-01-05 Sucampo Ag Pharmazeutische magensaftresistent überzogene zusammensetzung enthaltend prostaglandin-analoga als chloridkanalöffner
JP5265369B2 (ja) * 2006-01-24 2013-08-14 株式会社アールテック・ウエノ 二環式化合物を含む医薬組成物およびその二環式化合物の安定化方法
US20090030072A1 (en) * 2007-07-03 2009-01-29 Sucampo Ag Pharmaceutical combination of opioid and prostaglandin compound
CN108685929A (zh) * 2012-04-23 2018-10-23 苏坎波公司 用于治疗具有腹泻的肠易激综合征的方法
EP2952206B1 (en) * 2013-02-04 2018-10-24 Taisho Pharmaceutical Co., Ltd. Prophylactic or therapeutic drug for constipation
WO2014159679A1 (en) 2013-03-12 2014-10-02 The United States Of America, As Represented By The Secretary, Department Of Health & Human Services Methods for using lubiprostone to absorb fluid from the subretinal space

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5225439A (en) 1987-01-28 1993-07-06 K.K. Ueno Seiyaku Oyo Kenkyujo Prostaglandins E and anti ulcers containing same
US5166174A (en) 1987-01-28 1992-11-24 K.K. Ueno Seiyaku Oyo Kenkyujo Prostaglandins E and anti-ulcers containing same
US5428062A (en) 1987-01-28 1995-06-27 K.K. Ueno Seiyaku Oyo Kenkyujo Prostaglandins E and anti ulcers containing same
US5317032A (en) * 1987-10-02 1994-05-31 Kabushiki Kaisha Ueno Seiyaku Oyo Kenkyujo Prostaglandin cathartic
BRPI0014869B8 (pt) 1999-10-15 2021-05-25 Sucampo Ag prostaglandinas bicíclicas, composições estabilizadas das mesmas, bem como processo para sua estabilização
US6414016B1 (en) * 2000-09-05 2002-07-02 Sucampo, A.G. Anti-constipation composition
TWI302100B (en) 2001-05-02 2008-10-21 Sucampo Ag Composition for treating drug-induced constipation
ATE387204T1 (de) 2001-05-18 2008-03-15 Sucampo Ag Zusammensetzung mit induzierendem kathartischen effekt
EP1420794B1 (en) 2001-08-31 2017-12-27 Sucampo AG Prostaglandin analogs as chloride channel openers
AR037524A1 (es) * 2001-11-14 2004-11-17 Sucampo Ag Unidad de dosificacion que comprende un analogo de prostaglandina para el tratamiento de la constipacion
TWI263505B (en) 2001-11-19 2006-10-11 Sucampo Ag Pharmaceutical composition comprising a C1C-2 channel opener
EP1575596B1 (en) * 2002-12-27 2016-06-22 Sucampo AG Derivatives of prostaglandins for treating irritable bowel syndrome and/or functional dyspepsia
DE602004030245D1 (de) 2003-07-03 2011-01-05 Sucampo Ag Pharmazeutische magensaftresistent überzogene zusammensetzung enthaltend prostaglandin-analoga als chloridkanalöffner

Also Published As

Publication number Publication date
AR050626A1 (es) 2006-11-08
US20060063830A1 (en) 2006-03-23
IL181332A0 (en) 2007-07-04
CA2577284A1 (en) 2006-03-09
MX2007002602A (es) 2007-04-25
ES2603381T3 (es) 2017-02-27
JP2013049688A (ja) 2013-03-14
KR20180033310A (ko) 2018-04-02
NO20071704L (no) 2007-05-31
JP2015166377A (ja) 2015-09-24
KR20140019006A (ko) 2014-02-13
EP1791545A1 (en) 2007-06-06
AU2005278323A1 (en) 2006-03-09
WO2006025599A1 (en) 2006-03-09
US20140315994A1 (en) 2014-10-23
NZ553434A (en) 2010-01-29
NO340989B1 (no) 2017-07-31
TW200612901A (en) 2006-05-01
CN102885821A (zh) 2013-01-23
JP2018150354A (ja) 2018-09-27
JP2008511541A (ja) 2008-04-17
KR20170003712A (ko) 2017-01-09
US8748481B2 (en) 2014-06-10
BRPI0514891A (pt) 2008-06-24
IL181332A (en) 2015-09-24
AU2005278323B2 (en) 2011-03-17
JP6408426B2 (ja) 2018-10-17
TWI387454B (zh) 2013-03-01
EP1791545B1 (en) 2016-08-31

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