KR20050109965A - 라파마이신 유도체 및 아로마타제 억제제를 포함하는항종양 배합물 - Google Patents

라파마이신 유도체 및 아로마타제 억제제를 포함하는항종양 배합물 Download PDF

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Publication number
KR20050109965A
KR20050109965A KR1020057016528A KR20057016528A KR20050109965A KR 20050109965 A KR20050109965 A KR 20050109965A KR 1020057016528 A KR1020057016528 A KR 1020057016528A KR 20057016528 A KR20057016528 A KR 20057016528A KR 20050109965 A KR20050109965 A KR 20050109965A
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KR
South Korea
Prior art keywords
tumor
aromatase inhibitor
cancer
cci
letrozole
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
KR1020057016528A
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English (en)
Korean (ko)
Inventor
매튜 엘 셔먼
제임스 제이 쥬니어 깁본스
마크 버거
로버트 티 맥과이어
로버트 프리드먼
Original Assignee
와이어쓰
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32962706&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR20050109965(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 와이어쓰 filed Critical 와이어쓰
Publication of KR20050109965A publication Critical patent/KR20050109965A/ko
Ceased legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4188—1,3-Diazoles condensed with other heterocyclic ring systems, e.g. biotin, sorbinil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • A61K31/5685—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone having an oxo group in position 17, e.g. androsterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
KR1020057016528A 2003-03-05 2004-03-01 라파마이신 유도체 및 아로마타제 억제제를 포함하는항종양 배합물 Ceased KR20050109965A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US45228903P 2003-03-05 2003-03-05
US60/452,289 2003-03-05

Publications (1)

Publication Number Publication Date
KR20050109965A true KR20050109965A (ko) 2005-11-22

Family

ID=32962706

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020057016528A Ceased KR20050109965A (ko) 2003-03-05 2004-03-01 라파마이신 유도체 및 아로마타제 억제제를 포함하는항종양 배합물

Country Status (20)

Country Link
US (1) US20040176339A1 (cg-RX-API-DMAC7.html)
EP (1) EP1603561A2 (cg-RX-API-DMAC7.html)
JP (1) JP2006519862A (cg-RX-API-DMAC7.html)
KR (1) KR20050109965A (cg-RX-API-DMAC7.html)
CN (1) CN1756549A (cg-RX-API-DMAC7.html)
AR (1) AR043403A1 (cg-RX-API-DMAC7.html)
AU (1) AU2004218439A1 (cg-RX-API-DMAC7.html)
BR (1) BRPI0408024A (cg-RX-API-DMAC7.html)
CA (1) CA2516353A1 (cg-RX-API-DMAC7.html)
CR (1) CR7942A (cg-RX-API-DMAC7.html)
EC (1) ECSP056001A (cg-RX-API-DMAC7.html)
MX (1) MXPA05009246A (cg-RX-API-DMAC7.html)
NI (1) NI200500148A (cg-RX-API-DMAC7.html)
NO (1) NO20054133L (cg-RX-API-DMAC7.html)
NZ (1) NZ542738A (cg-RX-API-DMAC7.html)
RU (1) RU2355399C2 (cg-RX-API-DMAC7.html)
TW (1) TW200529829A (cg-RX-API-DMAC7.html)
UA (1) UA83484C2 (cg-RX-API-DMAC7.html)
WO (1) WO2004078133A2 (cg-RX-API-DMAC7.html)
ZA (1) ZA200508029B (cg-RX-API-DMAC7.html)

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AR047988A1 (es) * 2004-03-11 2006-03-15 Wyeth Corp Combinaciones antineoplásicas de cci-779 y rituximab
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CN103110948A (zh) 2005-11-04 2013-05-22 惠氏公司 mTOR抑制剂、赫赛汀和/或HKI-272的抗肿瘤组合
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WO2010008744A2 (en) 2008-06-17 2010-01-21 Wyeth Antineoplastic combinations containing hki-272 and vinorelbine
RU2498804C2 (ru) 2008-08-04 2013-11-20 ВАЙЕТ ЭлЭлСи Противоопухолевые комбинации из 4-анилино-3-цианохинолинов и капецитабина
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JP5992325B2 (ja) 2009-04-06 2016-09-14 ワイス・エルエルシー 乳癌のための、ネラチニブを活用する治療計画
CN102612564B (zh) 2009-04-10 2015-08-26 齐海燕 新的抗衰老试剂及其鉴别方法
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Also Published As

Publication number Publication date
CR7942A (es) 2006-02-07
AR043403A1 (es) 2005-07-27
RU2355399C2 (ru) 2009-05-20
WO2004078133A2 (en) 2004-09-16
JP2006519862A (ja) 2006-08-31
NO20054133L (no) 2005-10-03
MXPA05009246A (es) 2005-10-19
NI200500148A (es) 2006-03-30
AU2004218439A1 (en) 2004-09-16
CA2516353A1 (en) 2004-09-16
RU2005130767A (ru) 2006-02-10
UA83484C2 (uk) 2008-07-25
NO20054133D0 (no) 2005-09-06
WO2004078133A3 (en) 2004-11-11
NZ542738A (en) 2009-02-28
WO2004078133A8 (en) 2005-09-01
TW200529829A (en) 2005-09-16
BRPI0408024A (pt) 2006-02-14
CN1756549A (zh) 2006-04-05
ZA200508029B (en) 2007-04-25
US20040176339A1 (en) 2004-09-09
ECSP056001A (es) 2006-01-27
EP1603561A2 (en) 2005-12-14

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