KR20040111348A - 결장 수송체에 의한 치료 화합물의 조작 흡수 - Google Patents
결장 수송체에 의한 치료 화합물의 조작 흡수 Download PDFInfo
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- KR20040111348A KR20040111348A KR10-2004-7011457A KR20047011457A KR20040111348A KR 20040111348 A KR20040111348 A KR 20040111348A KR 20047011457 A KR20047011457 A KR 20047011457A KR 20040111348 A KR20040111348 A KR 20040111348A
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- conjugate
- transporter
- agent
- plasma membrane
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Classifications
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/62—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being a protein, peptide or polyamino acid
- A61K47/64—Drug-peptide, drug-protein or drug-polyamino acid conjugates, i.e. the modifying agent being a peptide, protein or polyamino acid which is covalently bonded or complexed to a therapeutically active agent
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
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- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| US35180802P | 2002-01-24 | 2002-01-24 | |
| US60/351,808 | 2002-01-24 | ||
| US10/351,291 US20030158254A1 (en) | 2002-01-24 | 2003-01-23 | Engineering absorption of therapeutic compounds via colonic transporters |
| US10/351,291 | 2003-01-23 | ||
| PCT/US2003/002206 WO2003065982A2 (en) | 2002-01-24 | 2003-01-24 | Engineering absorption of therapeutic compounds via colonic transporters |
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| KR20040111348A true KR20040111348A (ko) | 2004-12-31 |
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| US (1) | US20030158254A1 (https=) |
| EP (1) | EP1575494A2 (https=) |
| JP (1) | JP2005529847A (https=) |
| KR (1) | KR20040111348A (https=) |
| AU (1) | AU2003244398A1 (https=) |
| CA (1) | CA2473802A1 (https=) |
| WO (1) | WO2003065982A2 (https=) |
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| US7186855B2 (en) * | 2001-06-11 | 2007-03-06 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
| US8048917B2 (en) | 2005-04-06 | 2011-11-01 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
| ATE540678T1 (de) * | 2001-06-11 | 2012-01-15 | Xenoport Inc | Prodrugs aus gaba-analoga, zusammensetzungen und ihre verwendungen |
| UA78529C2 (en) | 2001-10-10 | 2007-04-10 | Wyeth Corp | Derivatives of [[2-(amino-3,4-dioxo-1-cyclobutene-1-yl)amino]alkyl] acid for treating pain |
| JP4395070B2 (ja) * | 2002-06-25 | 2010-01-06 | インデックス・ダイアグノスティックス・アクチエボラーグ | 潰瘍性大腸炎を診断するための方法およびキット |
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-
2003
- 2003-01-23 US US10/351,291 patent/US20030158254A1/en not_active Abandoned
- 2003-01-24 AU AU2003244398A patent/AU2003244398A1/en not_active Abandoned
- 2003-01-24 WO PCT/US2003/002206 patent/WO2003065982A2/en not_active Ceased
- 2003-01-24 JP JP2003565408A patent/JP2005529847A/ja not_active Withdrawn
- 2003-01-24 KR KR10-2004-7011457A patent/KR20040111348A/ko not_active Withdrawn
- 2003-01-24 EP EP03737554A patent/EP1575494A2/en not_active Withdrawn
- 2003-01-24 CA CA002473802A patent/CA2473802A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CA2473802A1 (en) | 2003-08-14 |
| JP2005529847A (ja) | 2005-10-06 |
| WO2003065982A2 (en) | 2003-08-14 |
| AU2003244398A1 (en) | 2003-09-02 |
| US20030158254A1 (en) | 2003-08-21 |
| WO2003065982A3 (en) | 2005-12-08 |
| EP1575494A2 (en) | 2005-09-21 |
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