JPWO2021041276A5 - - Google Patents
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- Publication number
- JPWO2021041276A5 JPWO2021041276A5 JP2022511322A JP2022511322A JPWO2021041276A5 JP WO2021041276 A5 JPWO2021041276 A5 JP WO2021041276A5 JP 2022511322 A JP2022511322 A JP 2022511322A JP 2022511322 A JP2022511322 A JP 2022511322A JP WO2021041276 A5 JPWO2021041276 A5 JP WO2021041276A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- dihydrothieno
- cyclopenta
- indazol
- pyrazole
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962891097P | 2019-08-23 | 2019-08-23 | |
| US62/891,097 | 2019-08-23 | ||
| PCT/US2020/047552 WO2021041276A1 (en) | 2019-08-23 | 2020-08-22 | Heterocyclic pyrazole derivatives as type iii receptor tyrosine kinase inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2022545019A JP2022545019A (ja) | 2022-10-24 |
| JPWO2021041276A5 true JPWO2021041276A5 (ru) | 2023-08-18 |
Family
ID=74685735
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022511322A Pending JP2022545019A (ja) | 2019-08-23 | 2020-08-22 | Ｉｉｉ型受容体チロシンキナーゼ阻害剤としてのヘテロ環式ピラゾール誘導体 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US20220289759A1 (ru) |
| EP (1) | EP4017853A4 (ru) |
| JP (1) | JP2022545019A (ru) |
| KR (1) | KR20220051365A (ru) |
| CN (1) | CN114502553B (ru) |
| AU (1) | AU2020337883A1 (ru) |
| BR (1) | BR112022003383A2 (ru) |
| CA (1) | CA3151821A1 (ru) |
| MX (1) | MX2022002062A (ru) |
| TW (1) | TWI759829B (ru) |
| WO (1) | WO2021041276A1 (ru) |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101146532B (zh) * | 2005-01-21 | 2012-05-09 | 阿斯泰克斯治疗有限公司 | 药物化合物 |
| BRPI0618011A2 (pt) * | 2005-10-28 | 2011-08-16 | Astrazeneca Ab | composto ou um sal farmaceuticamente aceitável do mesmo, processo para a preparação do mesmo, composição farmacêutica, uso de um composto ou um sal farmaceuticamente aceitável do mesmo, e, métodos para produzir um efeito anti-proliferativo e um efeito pró-apoptósico em um animal de sangue quente, para tratar doença e para produzir um efeito inibidor de jak em um animal de sangue quente |
| WO2008045627A2 (en) * | 2006-10-06 | 2008-04-17 | Irm Llc | Protein kinase inhibitors and methods for using thereof |
| EA017269B1 (ru) * | 2007-05-04 | 2012-11-30 | Айрм Ллк | ПРОИЗВОДНЫЕ ПИРИМИДИНА И СОДЕРЖАЩИЕ ИХ КОМПОЗИЦИИ КАК ИНГИБИТОРЫ КИНАЗЫ c-kit И PDGFR |
| CN102811619B (zh) * | 2009-11-13 | 2015-04-22 | 金纳斯克公司 | 激酶抑制剂 |
| GB201007286D0 (en) * | 2010-04-30 | 2010-06-16 | Astex Therapeutics Ltd | New compounds |
| PL2828259T3 (pl) * | 2012-03-22 | 2019-02-28 | Oscotec, Inc. | Podstawione związki pirydopirymidynowe oraz ich zastosowanie jako inhibitory flt3 |
| US8853207B2 (en) * | 2012-04-12 | 2014-10-07 | Development Center For Biotechnology | Heterocyclic pyrazole compounds, method for preparing the same and use thereof |
| CA3007462C (en) * | 2015-12-07 | 2023-10-24 | Plexxikon Inc. | Compounds and methods for kinase modulation, and indications therefor |
-
2020
- 2020-08-21 TW TW109128678A patent/TWI759829B/zh active
- 2020-08-22 AU AU2020337883A patent/AU2020337883A1/en active Pending
- 2020-08-22 US US17/636,116 patent/US20220289759A1/en active Pending
- 2020-08-22 KR KR1020227009059A patent/KR20220051365A/ko unknown
- 2020-08-22 WO PCT/US2020/047552 patent/WO2021041276A1/en unknown
- 2020-08-22 BR BR112022003383A patent/BR112022003383A2/pt unknown
- 2020-08-22 EP EP20856905.3A patent/EP4017853A4/en active Pending
- 2020-08-22 CN CN202080059010.6A patent/CN114502553B/zh active Active
- 2020-08-22 CA CA3151821A patent/CA3151821A1/en active Pending
- 2020-08-22 JP JP2022511322A patent/JP2022545019A/ja active Pending
- 2020-08-22 MX MX2022002062A patent/MX2022002062A/es unknown
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