JPWO2020259584A5 - - Google Patents
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- JPWO2020259584A5 JPWO2020259584A5 JP2021577587A JP2021577587A JPWO2020259584A5 JP WO2020259584 A5 JPWO2020259584 A5 JP WO2020259584A5 JP 2021577587 A JP2021577587 A JP 2021577587A JP 2021577587 A JP2021577587 A JP 2021577587A JP WO2020259584 A5 JPWO2020259584 A5 JP WO2020259584A5
- Authority
- JP
- Japan
- Prior art keywords
- compound according
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Claims (1)
- Lが-C(O)-である、請求項1又は2に記載の化合物。
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CN201910572091.9A CN112142743A (zh) | 2019-06-28 | 2019-06-28 | 杂环类化合物、其制备方法及其在医药学上的应用 |
CN201910572091.9 | 2019-06-28 | ||
PCT/CN2020/098105 WO2020259584A1 (en) | 2019-06-28 | 2020-06-24 | Heterocyclic compounds for mediating tyrosine kinase 2 activity |
Publications (2)
Publication Number | Publication Date |
---|---|
JP2022540353A JP2022540353A (ja) | 2022-09-15 |
JPWO2020259584A5 true JPWO2020259584A5 (ja) | 2023-06-02 |
Family
ID=73869063
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2021577587A Pending JP2022540353A (ja) | 2019-06-28 | 2020-06-24 | チロシンキナーゼ2活性を仲介する複素環式化合物 |
Country Status (11)
Country | Link |
---|---|
US (1) | US20220112200A1 (ja) |
EP (1) | EP3990449A4 (ja) |
JP (1) | JP2022540353A (ja) |
KR (1) | KR20220042344A (ja) |
CN (2) | CN112142743A (ja) |
AU (1) | AU2020301437A1 (ja) |
BR (1) | BR112021026531A2 (ja) |
CA (1) | CA3144799A1 (ja) |
MX (1) | MX2021015969A (ja) |
TW (1) | TW202115034A (ja) |
WO (1) | WO2020259584A1 (ja) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN112142743A (zh) * | 2019-06-28 | 2020-12-29 | 广州诺诚健华医药科技有限公司 | 杂环类化合物、其制备方法及其在医药学上的应用 |
TWI782599B (zh) * | 2020-07-02 | 2022-11-01 | 美商輝瑞股份有限公司 | 胺基嘧啶基衍生物 |
CN113234081A (zh) * | 2021-05-27 | 2021-08-10 | 东南大学 | 一种吡咯并吡唑衍生物与dmpeda做脲的制备方法 |
WO2023076161A1 (en) | 2021-10-25 | 2023-05-04 | Kymera Therapeutics, Inc. | Tyk2 degraders and uses thereof |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN103298794A (zh) * | 2010-11-09 | 2013-09-11 | 塞尔卓姆有限公司 | 作为tyk2抑制剂的吡啶化合物及其氮杂类似物 |
US9586962B2 (en) * | 2011-04-20 | 2017-03-07 | Janssen Pharmaceutica Nv | Disubstituted octahydropyrrolo [3,4-C] pyrroles as orexin receptor modulators |
WO2013146963A1 (ja) * | 2012-03-28 | 2013-10-03 | 武田薬品工業株式会社 | 複素環化合物 |
CN105622638B (zh) * | 2014-10-29 | 2018-10-02 | 广州必贝特医药技术有限公司 | 嘧啶或吡啶并吡啶酮类化合物及其制备方法和应用 |
JP6853234B2 (ja) * | 2015-07-09 | 2021-03-31 | メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung | Btk阻害剤としてのピリミジン誘導体及びその使用 |
TW201920170A (zh) * | 2017-09-20 | 2019-06-01 | 美商庫拉腫瘤技術股份有限公司 | 經取代之menin-mll 抑制劑及使用方法 |
CN112142743A (zh) * | 2019-06-28 | 2020-12-29 | 广州诺诚健华医药科技有限公司 | 杂环类化合物、其制备方法及其在医药学上的应用 |
-
2019
- 2019-06-28 CN CN201910572091.9A patent/CN112142743A/zh active Pending
-
2020
- 2020-06-24 CA CA3144799A patent/CA3144799A1/en active Pending
- 2020-06-24 BR BR112021026531A patent/BR112021026531A2/pt unknown
- 2020-06-24 JP JP2021577587A patent/JP2022540353A/ja active Pending
- 2020-06-24 MX MX2021015969A patent/MX2021015969A/es unknown
- 2020-06-24 EP EP20832538.1A patent/EP3990449A4/en active Pending
- 2020-06-24 TW TW109121616A patent/TW202115034A/zh unknown
- 2020-06-24 AU AU2020301437A patent/AU2020301437A1/en active Pending
- 2020-06-24 CN CN202080047732.XA patent/CN114096532B/zh active Active
- 2020-06-24 WO PCT/CN2020/098105 patent/WO2020259584A1/en active Application Filing
- 2020-06-24 KR KR1020227000934A patent/KR20220042344A/ko unknown
-
2021
- 2021-12-22 US US17/559,330 patent/US20220112200A1/en active Pending
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