JPWO2020259584A5 - - Google Patents

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Publication number
JPWO2020259584A5
JPWO2020259584A5 JP2021577587A JP2021577587A JPWO2020259584A5 JP WO2020259584 A5 JPWO2020259584 A5 JP WO2020259584A5 JP 2021577587 A JP2021577587 A JP 2021577587A JP 2021577587 A JP2021577587 A JP 2021577587A JP WO2020259584 A5 JPWO2020259584 A5 JP WO2020259584A5
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JP
Japan
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JP2021577587A
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JP2022540353A (ja
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Priority claimed from CN201910572091.9A external-priority patent/CN112142743A/zh
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Publication of JP2022540353A publication Critical patent/JP2022540353A/ja
Publication of JPWO2020259584A5 publication Critical patent/JPWO2020259584A5/ja
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Claims (1)

  1. Lが-C(O)-である、請求項1又は2に記載の化合物。
JP2021577587A 2019-06-28 2020-06-24 チロシンキナーゼ2活性を仲介する複素環式化合物 Pending JP2022540353A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN201910572091.9A CN112142743A (zh) 2019-06-28 2019-06-28 杂环类化合物、其制备方法及其在医药学上的应用
CN201910572091.9 2019-06-28
PCT/CN2020/098105 WO2020259584A1 (en) 2019-06-28 2020-06-24 Heterocyclic compounds for mediating tyrosine kinase 2 activity

Publications (2)

Publication Number Publication Date
JP2022540353A JP2022540353A (ja) 2022-09-15
JPWO2020259584A5 true JPWO2020259584A5 (ja) 2023-06-02

Family

ID=73869063

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021577587A Pending JP2022540353A (ja) 2019-06-28 2020-06-24 チロシンキナーゼ2活性を仲介する複素環式化合物

Country Status (11)

Country Link
US (1) US20220112200A1 (ja)
EP (1) EP3990449A4 (ja)
JP (1) JP2022540353A (ja)
KR (1) KR20220042344A (ja)
CN (2) CN112142743A (ja)
AU (1) AU2020301437A1 (ja)
BR (1) BR112021026531A2 (ja)
CA (1) CA3144799A1 (ja)
MX (1) MX2021015969A (ja)
TW (1) TW202115034A (ja)
WO (1) WO2020259584A1 (ja)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN112142743A (zh) * 2019-06-28 2020-12-29 广州诺诚健华医药科技有限公司 杂环类化合物、其制备方法及其在医药学上的应用
TWI782599B (zh) * 2020-07-02 2022-11-01 美商輝瑞股份有限公司 胺基嘧啶基衍生物
CN113234081A (zh) * 2021-05-27 2021-08-10 东南大学 一种吡咯并吡唑衍生物与dmpeda做脲的制备方法
WO2023076161A1 (en) 2021-10-25 2023-05-04 Kymera Therapeutics, Inc. Tyk2 degraders and uses thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103298794A (zh) * 2010-11-09 2013-09-11 塞尔卓姆有限公司 作为tyk2抑制剂的吡啶化合物及其氮杂类似物
US9586962B2 (en) * 2011-04-20 2017-03-07 Janssen Pharmaceutica Nv Disubstituted octahydropyrrolo [3,4-C] pyrroles as orexin receptor modulators
WO2013146963A1 (ja) * 2012-03-28 2013-10-03 武田薬品工業株式会社 複素環化合物
CN105622638B (zh) * 2014-10-29 2018-10-02 广州必贝特医药技术有限公司 嘧啶或吡啶并吡啶酮类化合物及其制备方法和应用
JP6853234B2 (ja) * 2015-07-09 2021-03-31 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung Btk阻害剤としてのピリミジン誘導体及びその使用
TW201920170A (zh) * 2017-09-20 2019-06-01 美商庫拉腫瘤技術股份有限公司 經取代之menin-mll 抑制劑及使用方法
CN112142743A (zh) * 2019-06-28 2020-12-29 广州诺诚健华医药科技有限公司 杂环类化合物、其制备方法及其在医药学上的应用

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