JPS6422858A - Fluorine-containing pyrimidine derivative and its preparation - Google Patents
Fluorine-containing pyrimidine derivative and its preparationInfo
- Publication number
- JPS6422858A JPS6422858A JP17604987A JP17604987A JPS6422858A JP S6422858 A JPS6422858 A JP S6422858A JP 17604987 A JP17604987 A JP 17604987A JP 17604987 A JP17604987 A JP 17604987A JP S6422858 A JPS6422858 A JP S6422858A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- fluorine
- derivative
- preparation
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
NEW MATERIAL:A fluorine-containing pyrimidine derivative of formula I (R is H, alkyl, phenyl, NH2; R<1> is alkyl, cycloalkyl, phenyl; R<f> is perfluoroalkyl). EXAMPLE:5-Fluoro-4-trifluoromethyl-6-hexyl-2-methylpyrimidine. USE:Medicines of agrochemicals such as antibacterial, herbicide or physiologically active substance or an intermediate thereof. PREPARATION:The reaction between a fluorine-containing phosphate derivative of formula II (R<2> is lower alkyl) and an amidine derivative of formula III is carried out in an inert solvent to give the compound of formula I easily in high yield. The compound of formula II is readily prepared from a fluorine- containing ketone derivative of formula IV and dialkyl phosphite of formula IV.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP17604987A JPS6422858A (en) | 1987-07-16 | 1987-07-16 | Fluorine-containing pyrimidine derivative and its preparation |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP17604987A JPS6422858A (en) | 1987-07-16 | 1987-07-16 | Fluorine-containing pyrimidine derivative and its preparation |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS6422858A true JPS6422858A (en) | 1989-01-25 |
Family
ID=16006823
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP17604987A Pending JPS6422858A (en) | 1987-07-16 | 1987-07-16 | Fluorine-containing pyrimidine derivative and its preparation |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS6422858A (en) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2001010843A1 (en) * | 1999-08-05 | 2001-02-15 | Mitsubishi Chemical Corporation | 4-(substituted phenyl)-5-halopyrimidine derivatives and herbicides containing the same as the active ingredient |
JP2005529184A (en) * | 2002-06-13 | 2005-09-29 | バイエル・クロツプサイエンス・アクチエンゲゼルシヤフト | Process for the preparation of 4,6-dichloro-5-fluoropyrimidine |
-
1987
- 1987-07-16 JP JP17604987A patent/JPS6422858A/en active Pending
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2001010843A1 (en) * | 1999-08-05 | 2001-02-15 | Mitsubishi Chemical Corporation | 4-(substituted phenyl)-5-halopyrimidine derivatives and herbicides containing the same as the active ingredient |
JP2005529184A (en) * | 2002-06-13 | 2005-09-29 | バイエル・クロツプサイエンス・アクチエンゲゼルシヤフト | Process for the preparation of 4,6-dichloro-5-fluoropyrimidine |
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