JPS5791987A - Aminoquinazoline derivative and its preparation - Google Patents
Aminoquinazoline derivative and its preparationInfo
- Publication number
- JPS5791987A JPS5791987A JP16632680A JP16632680A JPS5791987A JP S5791987 A JPS5791987 A JP S5791987A JP 16632680 A JP16632680 A JP 16632680A JP 16632680 A JP16632680 A JP 16632680A JP S5791987 A JPS5791987 A JP S5791987A
- Authority
- JP
- Japan
- Prior art keywords
- expressed
- lower alkyl
- formulai
- phenyl
- derivative
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- CZAAKPFIWJXPQT-UHFFFAOYSA-N quinazolin-2-amine Chemical class C1=CC=CC2=NC(N)=NC=C21 CZAAKPFIWJXPQT-UHFFFAOYSA-N 0.000 title abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 101800000734 Angiotensin-1 Proteins 0.000 abstract 1
- 102400000344 Angiotensin-1 Human genes 0.000 abstract 1
- 102000004190 Enzymes Human genes 0.000 abstract 1
- 108090000790 Enzymes Proteins 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 125000004423 acyloxy group Chemical group 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- ORWYRWWVDCYOMK-HBZPZAIKSA-N angiotensin I Chemical compound C([C@@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CC=1NC=NC=1)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CC=1C=CC=CC=1)C(=O)N[C@@H](CC=1NC=NC=1)C(=O)N[C@@H](CC(C)C)C(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H](N)CC(O)=O)C(C)C)C1=CC=C(O)C=C1 ORWYRWWVDCYOMK-HBZPZAIKSA-N 0.000 abstract 1
- 239000002220 antihypertensive agent Substances 0.000 abstract 1
- 150000001732 carboxylic acid derivatives Chemical class 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 230000001077 hypotensive effect Effects 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 239000000463 material Substances 0.000 abstract 1
- 150000003246 quinazolines Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Landscapes
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP16632680A JPS5791987A (en) | 1980-11-26 | 1980-11-26 | Aminoquinazoline derivative and its preparation |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP16632680A JPS5791987A (en) | 1980-11-26 | 1980-11-26 | Aminoquinazoline derivative and its preparation |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS5791987A true JPS5791987A (en) | 1982-06-08 |
| JPS6324513B2 JPS6324513B2 (enrdf_load_stackoverflow) | 1988-05-20 |
Family
ID=15829277
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP16632680A Granted JPS5791987A (en) | 1980-11-26 | 1980-11-26 | Aminoquinazoline derivative and its preparation |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JPS5791987A (enrdf_load_stackoverflow) |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS52102286A (en) * | 1976-02-18 | 1977-08-27 | Bristol Myers Co | 1*3*44oxadiazoleamides |
| JPS53103485A (en) * | 1977-02-22 | 1978-09-08 | Bristol Myers Co | Quinazoline compounds |
| JPS5459292A (enrdf_load_stackoverflow) * | 1977-09-30 | 1979-05-12 | Bristol Myers Co |
-
1980
- 1980-11-26 JP JP16632680A patent/JPS5791987A/ja active Granted
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS52102286A (en) * | 1976-02-18 | 1977-08-27 | Bristol Myers Co | 1*3*44oxadiazoleamides |
| JPS53103485A (en) * | 1977-02-22 | 1978-09-08 | Bristol Myers Co | Quinazoline compounds |
| JPS5459292A (enrdf_load_stackoverflow) * | 1977-09-30 | 1979-05-12 | Bristol Myers Co |
Also Published As
| Publication number | Publication date |
|---|---|
| JPS6324513B2 (enrdf_load_stackoverflow) | 1988-05-20 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CA2195677A1 (en) | Endothelin antagonists | |
| EP0386675A3 (en) | Xanthine derivatives | |
| IE902139L (en) | Imidazolyl alkenoic acids | |
| HU9200278D0 (en) | 2,3,6.-substituted kinazolinon derivatives with angiotenzyn ii receptor blocing effect | |
| MX9705675A (es) | Antagonistas alfa-1-adrenergicos de hexahidrobenz[e]isoindol sustituidos biciclicos. | |
| SK1452000A3 (en) | Pyrrolidine-3-carboxylic acid derivatives and their use as endothelin antagonists | |
| EP1609790A3 (en) | Benzo-1,3-dioxolyl- and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists | |
| CA2205274A1 (en) | Novel 2,3 disubstituted-(5,6)-heteroarylfused-pyrimidine-4-ones | |
| CA2227386A1 (en) | Piperazine derivatives and their use as 5-ht1a antagonists | |
| EP0296581A3 (en) | Amino acid 1,2-diketo derivatives as renin inhibitors | |
| WO2002102978A3 (en) | Human growth hormone antagonists | |
| ES8607218A1 (es) | Un procedimiento para preparar compuestos de amidina | |
| WO1997031016A3 (en) | New inhibitors of sh2-mediated processes | |
| NO932431L (no) | Fremgangsmaate og mellomprodukter for fremstilling av azabicyklo(2,2,2)oktan-3-iminer | |
| IL148548A0 (en) | Bicyclic vasopressin agonists | |
| JPS5793977A (en) | Acylaminoquinazoline derivative and its preparation | |
| EP0168921A3 (en) | Chemical compounds | |
| JPS5791987A (en) | Aminoquinazoline derivative and its preparation | |
| AU3635893A (en) | Triazolopyrimidin derivatives as antiotensin II receptor antagonists | |
| EP0331078A3 (en) | Process for the preparation of optically active 4-oxo-1-benzopyran-2-carboxylic acid derivatives and intermediates thereof | |
| CA2118425A1 (en) | Benzothiazolesulfonamide derivative, Method for Preparing the Same, and Use Thereof | |
| EP0987255A3 (en) | Substituted aminoquinazolinone (thione) derivatives | |
| NO950974L (no) | Nye N,N,N',N'-tetrasubstituert-1,2-etandiaminderivatforbindelser | |
| BG103986A (en) | Derivatives of pyrrolidinecarboxylic acids as endotheline antagonists | |
| EP0701551A1 (en) | 3- (INDOL-3-YL) PROPENIC ACID DERIVATIVES AS NMDA ANTAGONISTS |