JPS57501427A - - Google Patents

Info

Publication number
JPS57501427A
JPS57501427A JP56503061A JP50306181A JPS57501427A JP S57501427 A JPS57501427 A JP S57501427A JP 56503061 A JP56503061 A JP 56503061A JP 50306181 A JP50306181 A JP 50306181A JP S57501427 A JPS57501427 A JP S57501427A
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP56503061A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of JPS57501427A publication Critical patent/JPS57501427A/ja
Pending legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP56503061A 1980-09-29 1981-09-21 Pending JPS57501427A (ja)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8020861A FR2491066A1 (fr) 1980-09-29 1980-09-29 Benzoxazolinones substituees en 6 par une chaine aminoalcool ou aminocetone, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
JPS57501427A true JPS57501427A (ja) 1982-08-12

Family

ID=9246379

Family Applications (1)

Application Number Title Priority Date Filing Date
JP56503061A Pending JPS57501427A (ja) 1980-09-29 1981-09-21

Country Status (10)

Country Link
EP (1) EP0049203A1 (ja)
JP (1) JPS57501427A (ja)
CA (1) CA1179343A (ja)
DK (1) DK49682A (ja)
FR (1) FR2491066A1 (ja)
GR (1) GR82309B (ja)
HU (1) HU185975B (ja)
PT (1) PT73740B (ja)
WO (1) WO1982001186A1 (ja)
ZA (1) ZA816555B (ja)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH02289557A (ja) * 1989-03-30 1990-11-29 Adir 新規な5―アシルベンゾキサゾリノン誘導体

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0105053B1 (en) * 1982-10-01 1988-01-20 Merck & Co. Inc. Aralkylaminoethanol heterocyclic compounds
FR2536749A1 (fr) * 1982-11-25 1984-06-01 Cerm Cent Europ Rech Mauvernay (amino-2 ethyl)-6 benzoxazolinones substituees, leur preparation et leurs applications en therapeutique
GB8325370D0 (en) * 1983-09-22 1983-10-26 Fujisawa Pharmaceutical Co Benzoxazoline and benzothiazoline derivatives
FR2637286A1 (fr) * 1988-10-04 1990-04-06 Adir Nouveaux derives benzoxazolinoniques, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent
FR2643634A1 (fr) * 1989-02-28 1990-08-31 Adir Nouveaux derives benzoxazolinoniques, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent
US5182278A (en) * 1989-02-28 1993-01-26 Adir Et Compagnie Analgesic benzoxazolinones having at the 6-position a 1-hydroxy-3-morpholinopropyl side chain
IL93473A0 (en) * 1989-02-28 1990-11-29 Pfizer Antiinflammatory benzoxazolones
FR2646350B1 (fr) * 1989-04-28 1991-06-28 Adir Nouveaux derives benzothiazolinoniques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US5166353A (en) * 1989-04-28 1992-11-24 Adir Et Compagnie Benzothiazolinone compounds
FR2663634B1 (fr) * 1990-06-22 1992-09-04 Adir Nouvelles acyl benzoxazolinones, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
EP0567090B1 (en) * 1992-04-24 2000-07-26 Takeda Chemical Industries, Ltd. Benzoxazepine derivatives as cholinesterase inhibitors
JP2009521415A (ja) * 2005-12-21 2009-06-04 コーティカル・ピーティーワイ・リミテッド Mif阻害剤
DE102007047737A1 (de) 2007-10-05 2009-04-30 Merck Patent Gmbh Piperidin- und Piperazinderivate
CN101759665B (zh) 2008-12-23 2012-03-28 江苏恩华药业股份有限公司 取代苯基哌嗪芳烷醇衍生物及其在制备镇痛药物中的应用
DE102009049211A1 (de) 2009-10-13 2011-04-28 Merck Patent Gmbh Sulfoxide

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2244507A1 (en) * 1973-06-26 1975-04-18 Inst Nat Sante Rech Med Chalcones and analogues - analgesics having low toxicity
CA1041523A (en) * 1974-06-19 1978-10-31 Queen's University Preparation of 1-oxapenicillins and novel intermediates therefor

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH02289557A (ja) * 1989-03-30 1990-11-29 Adir 新規な5―アシルベンゾキサゾリノン誘導体

Also Published As

Publication number Publication date
DK49682A (da) 1982-04-15
ZA816555B (en) 1982-09-29
HU185975B (en) 1985-04-28
CA1179343A (en) 1984-12-11
WO1982001186A1 (en) 1982-04-15
GR82309B (ja) 1984-12-13
FR2491066A1 (fr) 1982-04-02
FR2491066B1 (ja) 1983-06-17
PT73740A (en) 1981-10-01
PT73740B (en) 1982-12-30
EP0049203A1 (fr) 1982-04-07

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