JPS5436287A - Thiadiazolylthiooxacephalosporin - Google Patents

Thiadiazolylthiooxacephalosporin

Info

Publication number
JPS5436287A
JPS5436287A JP10226077A JP10226077A JPS5436287A JP S5436287 A JPS5436287 A JP S5436287A JP 10226077 A JP10226077 A JP 10226077A JP 10226077 A JP10226077 A JP 10226077A JP S5436287 A JPS5436287 A JP S5436287A
Authority
JP
Japan
Prior art keywords
thiadiazolylthiooxacephalosporin
hal
protected
thiadiazolythiooxacephalosporin
cob
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP10226077A
Other languages
Japanese (ja)
Other versions
JPS6031835B2 (en
Inventor
Masayuki Narisada
Yoshio Hamashima
Sadao Hayashi
Wataru Nagata
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Shionogi and Co Ltd
Original Assignee
Shionogi and Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi and Co Ltd filed Critical Shionogi and Co Ltd
Priority to JP52102260A priority Critical patent/JPS6031835B2/en
Priority to CA300,788A priority patent/CA1100962A/en
Priority to PH21016A priority patent/PH16851A/en
Priority to GB16128/78A priority patent/GB1574273A/en
Priority to US05/900,235 priority patent/US4183928A/en
Priority to GR56114A priority patent/GR69966B/el
Priority to SU782608717A priority patent/SU784779A3/en
Priority to NZ187086A priority patent/NZ187086A/en
Priority to DK182878A priority patent/DK182878A/en
Priority to MX787044U priority patent/MX5952E/en
Priority to NO781502A priority patent/NO158506C/en
Priority to ES469206A priority patent/ES469206A1/en
Priority to HU78SI1625A priority patent/HU178105B/en
Priority to AR271935A priority patent/AR227614A1/en
Priority to IL54596A priority patent/IL54596A0/en
Priority to FR7812532A priority patent/FR2388815A1/en
Priority to AU35527/78A priority patent/AU522851B2/en
Priority to SE7804873A priority patent/SE447115B/en
Priority to FI781313A priority patent/FI63410C/en
Priority to PT67957A priority patent/PT67957B/en
Priority to DD78205105A priority patent/DD135908A5/en
Priority to YU1035/78A priority patent/YU42477B/en
Priority to NLAANVRAGE7804628,A priority patent/NL189669C/en
Priority to DE2818985A priority patent/DE2818985C2/en
Priority to IE844/78A priority patent/IE46627B1/en
Priority to PL1978206451A priority patent/PL110680B1/en
Priority to IT67986/78A priority patent/IT1111469B/en
Priority to BG7839585A priority patent/BG34337A3/en
Priority to CS782774A priority patent/CS199726B2/en
Priority to CH470478A priority patent/CH640535A5/en
Priority to AT311378A priority patent/AT357674B/en
Publication of JPS5436287A publication Critical patent/JPS5436287A/en
Publication of JPS6031835B2 publication Critical patent/JPS6031835B2/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40—Unsaturated compounds
    • C07C59/42—Unsaturated compounds containing hydroxy or O-metal groups
    • C07C59/56—Unsaturated compounds containing hydroxy or O-metal groups containing halogen

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

PURPOSE:Thiadiazolythiooxacephalosporin of formula I [Ar is formulas II, III, IV, etc. [Hal, Hal', is halogen; R'O is (protected) hydroxy]; R is H, lower alkyl; COA, COB are (protected) carboxy).
JP52102260A 1977-04-18 1977-08-25 Thiadiazolylthiooxacephalosporin Expired JPS6031835B2 (en)

Priority Applications (31)

Application Number Priority Date Filing Date Title
JP52102260A JPS6031835B2 (en) 1977-08-25 1977-08-25 Thiadiazolylthiooxacephalosporin
CA300,788A CA1100962A (en) 1977-04-28 1978-04-10 Haloarylmalonamidooxacephalosporins
PH21016A PH16851A (en) 1977-04-28 1978-04-17 Haloarylmalonamidooxacephalosporins
GB16128/78A GB1574273A (en) 1977-04-28 1978-04-24 Haloarylmalonamidooxacephalosporins
US05/900,235 US4183928A (en) 1977-04-28 1978-04-26 Haloarylmalonamidooxacephalosporins
GR56114A GR69966B (en) 1977-04-28 1978-04-26
SU782608717A SU784779A3 (en) 1977-04-28 1978-04-26 Method of preparing 7-beta-halogenarylmalonamido-7-alpha-methoxy-heterocyclylthiomethyl-1-dethia-1-oxa-3-cephem-4-carboxylic acid derivatives or their salts with organic or inorganic bases
NZ187086A NZ187086A (en) 1977-04-28 1978-04-26 7-(halophenylmalonamido)-7a-methoxy-3-(optionally alkylated tetrazol-5-yl or 1,3,4-thiadiazol-2-yl)-thiomethyl-1-dethia-1-oxa-3-cephem-4-carboxylic acid derivatives and pharmaceutical compositions
DK182878A DK182878A (en) 1977-04-28 1978-04-26 HALOARYLMALONAMIDOOXACEPHALOSPORINS AND METHODS FOR THE PREPARATION
MX787044U MX5952E (en) 1977-04-28 1978-04-27 PROCEDURE FOR THE PREPARATION OF ACIDS 7BETA HALOARILMALONAMIDO-7ALFA-METOXI-3-TIOMETIL HETEROAROMATICO-1-DETIA-1-OXA-3-CEFEM-4-CARBOXILICOS
NO781502A NO158506C (en) 1977-04-28 1978-04-27 ANALOGY PROCEDURE FOR THE PREPARATION OF PHARMACOLOGICAL ACTIVE 7BETA-HALOARYLMALON-AMIDO-7ALFA-METOXY-3- (1-METHYLTETRAZOL-5-YL) THIOMETHYL-1-DETIA-1-OKSA-3-CEFEMY-4-CEFEMY-5-CEFEMY-5-CEFEMY-5-CEFEMY-5-CEFEMY-5
ES469206A ES469206A1 (en) 1977-04-28 1978-04-27 Haloarylmalonamidooxacephalosporins
HU78SI1625A HU178105B (en) 1977-04-28 1978-04-27 Process for preparing 7beta-/halo-aryl /-malonamido/- 7alpha-methoxy-3-/ alkyl-tetrazol-5-yl- or -1,3,4-thiadiazol-2-yl /-thiomethyl/- 1-dethia-1-oxa-3-cephem-4-carboxylic acid derivatives
AR271935A AR227614A1 (en) 1977-04-28 1978-04-27 PROCEDURE FOR THE OBTAINING OF 7BETA-HALOARILMALONAMIDO-7ALPHA-METOXI-3-THOMETHYL HETEROCICLICO-1-DETIA-1-OXO-3-CEFEM-4-CARBOXILICOS
IL54596A IL54596A0 (en) 1977-04-28 1978-04-27 Haloraylmalonamidooxacephalosporins and processes for the preparation thereof
FR7812532A FR2388815A1 (en) 1977-04-28 1978-04-27 PROCESS FOR THE PREPARATION OF HALOARYLMALONAMIDOOXACEPHALOSPORINS, NEW PRODUCTS THUS OBTAINED AND THEIR USE FOR THE TREATMENT OF DISEASES DUE TO BACTERIA
AU35527/78A AU522851B2 (en) 1977-04-28 1978-04-27 Haloarylhalonamidooxacephalosporins
SE7804873A SE447115B (en) 1977-04-18 1978-04-27 PROCEDURE FOR PREPARING 7BETA-HALOARYLMALONAMIDO-7ALFA-METOXY-3-HETEROCYCLIC THIOMETHYL-1-DETIA-1-OXA-3-CEFEM-4-CARBOXYLIC ACID OR DERIVATIVE THEREOF
FI781313A FI63410C (en) 1977-04-28 1978-04-27 EXAMINATION OF ANTIBACTERIAL 7BETA-HALOARYLMALONAMIDO-7ALFA-METHOXY-3-HETEROCYCLISK THIOMETHYL-1-DETIA-1-OXA-3-CEFEM-4-CARBOXYL SYRICATE
PT67957A PT67957B (en) 1977-04-28 1978-04-27 Process for preparing haloarylmalonamidooxacephalosporins
DD78205105A DD135908A5 (en) 1977-04-28 1978-04-28 PROCESS FOR PREPARING HALOGENARYLMALONAMIDEOOXACEPHALOSPORINES
YU1035/78A YU42477B (en) 1977-04-28 1978-04-28 Process for obtaining haloarylmalone amido-1-dethio-1-oxa-cephalosporins
NLAANVRAGE7804628,A NL189669C (en) 1977-04-28 1978-04-28 METHOD FOR PREPARING A MEDICINAL PRODUCT WITH ANTIBACTERIAL ACTION AND METHOD FOR PREPARING MEDICINAL OXADETHIACEPHALOSPORINE DERIVATIVES
DE2818985A DE2818985C2 (en) 1977-04-28 1978-04-28 Halogenarylmalonamidooxacephalosporins and their use in combating bacterial infections
IE844/78A IE46627B1 (en) 1977-04-28 1978-04-28 Haloarylmalonamidooxacephalosporins
PL1978206451A PL110680B1 (en) 1977-04-28 1978-04-28 Method of producing new derivatives of 7-beta-halogeno-arylomalonamido-7-alpha-metoxy-3-heterocyclothiomethylo-1-dethia-1-oxa-3-cephamocarboxylic-4-acid
IT67986/78A IT1111469B (en) 1977-04-28 1978-04-28 CEPHALOSPORINE WITH ANTIBACTERIAL ACTION PROCEDURE FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
BG7839585A BG34337A3 (en) 1977-04-28 1978-04-28 Method for obtaining haloarylmalonamido- 1- dethia- 1- oxacephalosporines
CS782774A CS199726B2 (en) 1977-04-28 1978-04-28 Method of producing 7 beta-halogenaryl-malonamido-7-alpha-methoxy-3-heterocyclylthiomethyl-1-dethia-1-oxa-3-cephem-4-carboxylic acid and derivatives of the same
CH470478A CH640535A5 (en) 1977-04-28 1978-04-28 HALOGEN OR TRIFLUORMETHYLARYLMALONAMIDO-1-DETHIA-1-OXACEPHALOSPORINE AND METHOD FOR THE PRODUCTION THEREOF.
AT311378A AT357674B (en) 1977-04-28 1978-04-28 METHOD FOR PRODUCING NEW HALOGEN ARYLMALONAMIDOOXACEPHALOSPORINES

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP52102260A JPS6031835B2 (en) 1977-08-25 1977-08-25 Thiadiazolylthiooxacephalosporin

Publications (2)

Publication Number Publication Date
JPS5436287A true JPS5436287A (en) 1979-03-16
JPS6031835B2 JPS6031835B2 (en) 1985-07-24

Family

ID=14322614

Family Applications (1)

Application Number Title Priority Date Filing Date
JP52102260A Expired JPS6031835B2 (en) 1977-04-18 1977-08-25 Thiadiazolylthiooxacephalosporin

Country Status (1)

Country Link
JP (1) JPS6031835B2 (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6195421A (en) * 1984-10-16 1986-05-14 Sanyo Electric Co Ltd Constant current circuit

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS61153530U (en) * 1985-03-15 1986-09-24
JPH0349529Y2 (en) * 1985-07-19 1991-10-23

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6195421A (en) * 1984-10-16 1986-05-14 Sanyo Electric Co Ltd Constant current circuit

Also Published As

Publication number Publication date
JPS6031835B2 (en) 1985-07-24

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