JPS5289681A - Preparation of aracytidine -5# phosphoric acid ester derivatives - Google Patents

Preparation of aracytidine -5# phosphoric acid ester derivatives

Info

Publication number
JPS5289681A
JPS5289681A JP546176A JP546176A JPS5289681A JP S5289681 A JPS5289681 A JP S5289681A JP 546176 A JP546176 A JP 546176A JP 546176 A JP546176 A JP 546176A JP S5289681 A JPS5289681 A JP S5289681A
Authority
JP
Japan
Prior art keywords
aracytidine
phosphoric acid
preparation
acid ester
ester derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP546176A
Other languages
Japanese (ja)
Other versions
JPS5549588B2 (en
Inventor
Masami Morozumi
Morio Suzuki
Hiroshi Yoshino
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Yamasa Shoyu KK
Original Assignee
Yamasa Shoyu KK
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yamasa Shoyu KK filed Critical Yamasa Shoyu KK
Priority to JP546176A priority Critical patent/JPS5289681A/en
Publication of JPS5289681A publication Critical patent/JPS5289681A/en
Publication of JPS5549588B2 publication Critical patent/JPS5549588B2/ja
Granted legal-status Critical Current

Links

Landscapes

  • Saccharide Compounds (AREA)

Abstract

PURPOSE: To obtain aracytidine - 5' - phosphoric acid with alcohols by the use of an arylsulfonyl chloride which is available and easily handled as a condensing agent.
COPYRIGHT: (C)1977,JPO&Japio
JP546176A 1976-01-22 1976-01-22 Preparation of aracytidine -5# phosphoric acid ester derivatives Granted JPS5289681A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP546176A JPS5289681A (en) 1976-01-22 1976-01-22 Preparation of aracytidine -5# phosphoric acid ester derivatives

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP546176A JPS5289681A (en) 1976-01-22 1976-01-22 Preparation of aracytidine -5# phosphoric acid ester derivatives

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP3163780A Division JPS55129299A (en) 1980-03-14 1980-03-14 1-beta-d-arabinofuranosyl-cytosine-5'-phosphoric alkyl ester

Publications (2)

Publication Number Publication Date
JPS5289681A true JPS5289681A (en) 1977-07-27
JPS5549588B2 JPS5549588B2 (en) 1980-12-12

Family

ID=11611855

Family Applications (1)

Application Number Title Priority Date Filing Date
JP546176A Granted JPS5289681A (en) 1976-01-22 1976-01-22 Preparation of aracytidine -5# phosphoric acid ester derivatives

Country Status (1)

Country Link
JP (1) JPS5289681A (en)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS552601A (en) * 1978-06-20 1980-01-10 Yamasa Shoyu Co Ltd Anti-tumor agent for non-injection use
JPS552602A (en) * 1978-06-20 1980-01-10 Yamasa Shoyu Co Ltd 1-beta-d-arabinofranosylcytosine-5'-phosphoric acid oleyl ester
US5049663A (en) * 1986-03-24 1991-09-17 Nippon Kayaku Kabushiki Kaisha Process for producing 1-β-D-arabinofuranosylcytosine-5'-stearylphosphate monosodium salt and monohydrate thereof
JPH09508135A (en) * 1994-01-28 1997-08-19 ベーリンガー マンハイム ゲゼルシャフト ミット ベシュレンクテル ハフツング Process for producing asymmetric phosphoric acid diester and salt thereof

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS552601A (en) * 1978-06-20 1980-01-10 Yamasa Shoyu Co Ltd Anti-tumor agent for non-injection use
JPS552602A (en) * 1978-06-20 1980-01-10 Yamasa Shoyu Co Ltd 1-beta-d-arabinofranosylcytosine-5'-phosphoric acid oleyl ester
DE2924692A1 (en) 1978-06-20 1980-01-17 Saneyoshi Mineo 1- BETA -D-ARABINOFURANOSYLCYTOSINE- 5'-OLEYL PHOSPHATE AND ITS SALTS
JPS5726680B2 (en) * 1978-06-20 1982-06-05
JPS5748091B2 (en) * 1978-06-20 1982-10-14
US5049663A (en) * 1986-03-24 1991-09-17 Nippon Kayaku Kabushiki Kaisha Process for producing 1-β-D-arabinofuranosylcytosine-5'-stearylphosphate monosodium salt and monohydrate thereof
JPH09508135A (en) * 1994-01-28 1997-08-19 ベーリンガー マンハイム ゲゼルシャフト ミット ベシュレンクテル ハフツング Process for producing asymmetric phosphoric acid diester and salt thereof

Also Published As

Publication number Publication date
JPS5549588B2 (en) 1980-12-12

Similar Documents

Publication Publication Date Title
JPS5377015A (en) Preparation of fluorine-containing phosphoric acid ester
JPS5289681A (en) Preparation of aracytidine -5# phosphoric acid ester derivatives
JPS5340779A (en) Optically active tolpertisone, their preparation and pharmaceuticals containting the same
JPS5318529A (en) Optically active mandelic acid phenylglycinol salt and its preparation
JPS5356390A (en) Preparation of d-ribose-5'-phosphoric acid derivatives
JPS5296721A (en) Stable pharmaceutical dispersion
JPS536414A (en) Carboxylic acid aluminum salts and their preparation
JPS5422326A (en) 3-trimethylsilymethyl-3-butenoic acid and its preparation
JPS52102280A (en) 5,7,8-trimethyltocotrienol-nicotinic acid esters and preparation there of
JPS52100425A (en) Preparation of thioether derivatives
JPS5359674A (en) 1-piperidinoalkane-1,1-diphosphonic acid derivatives and herbicidescontaining the same as active agent
JPS5344572A (en) 5-alkoxy-picolic acid, its preparation and hypotensives containing the same
JPS5334752A (en) Preparation of gamma-ionones and their derivatives
JPS5341478A (en) Preparation of yeast cells
JPS5295674A (en) Preparation of 4#-substituted-2-methyl-2-piperidinopropiophenone and i ts salts
JPS52148037A (en) Preparation of per-#-toluylic acid
JPS5334772A (en) Preparation of 2-benzothiazolines
JPS53124619A (en) Agent for preventing plant phytotoxicity
JPS5371005A (en) Preparation of geranylacetone
JPS5325561A (en) Optical active lactam-2-acetic acid esters and their preparation
JPS53124293A (en) Novel adenosine derivatives
JPS52128369A (en) Alpha-isopropyl-substituted pyrrole-1-acetic acid ester
JPS52113917A (en) Preparation of alpha-chloroacrylic acid esters
JPS5231082A (en) Preparation of 2- piperazinophenylpropionic acid
JPS5424847A (en) Optical active methionine-mandelic acid complex and its preparation