JPS5251379A - Preparation 3,4-dihydro-2(1h)-quinazoline derivates - Google Patents
Preparation 3,4-dihydro-2(1h)-quinazoline derivatesInfo
- Publication number
- JPS5251379A JPS5251379A JP50128578A JP12857875A JPS5251379A JP S5251379 A JPS5251379 A JP S5251379A JP 50128578 A JP50128578 A JP 50128578A JP 12857875 A JP12857875 A JP 12857875A JP S5251379 A JPS5251379 A JP S5251379A
- Authority
- JP
- Japan
- Prior art keywords
- dihydro
- preparation
- derivates
- quinazoline
- quinazoline derivates
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 239000002253 acid Substances 0.000 abstract 1
- 229940035676 analgesics Drugs 0.000 abstract 1
- 239000000730 antalgic agent Substances 0.000 abstract 1
- 239000002260 anti-inflammatory agent Substances 0.000 abstract 1
- 229940121363 anti-inflammatory agent Drugs 0.000 abstract 1
- 230000003110 anti-inflammatory effect Effects 0.000 abstract 1
- 239000003054 catalyst Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000006210 cyclodehydration reaction Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/78—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
- C07D239/80—Oxygen atoms
- C07D239/82—Oxygen atoms with an aryl radical attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/78—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Priority Applications (14)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP50128578A JPS5251379A (en) | 1975-10-24 | 1975-10-24 | Preparation 3,4-dihydro-2(1h)-quinazoline derivates |
AU18545/76A AU490219B2 (en) | 1975-10-24 | 1976-10-11 | A novel process for preparing 3, 4-dihydro-2(1h)-quinazolinone derivatives |
NL7611210.A NL166934B (nl) | 1975-10-24 | 1976-10-11 | Werkwijze voor het bereiden van 3,4-dihydro-2(1h)- -chinazolinon- en -chinazolinethionderivaten. |
US05/731,574 US4202974A (en) | 1975-10-24 | 1976-10-12 | Process for preparing 3,4-dihydro-2(1H)-quinazolinone derivatives |
GB42337/76A GB1510068A (en) | 1975-10-24 | 1976-10-12 | Process for preparing 3,4-dihydro-2(1h)-quinazolinone derivatives |
AT770976A AT353796B (de) | 1975-10-24 | 1976-10-15 | Verfahren zur herstellung von 3,4-dihydro-2- (1h)-chinazolinonen und 3,4-dihydro-2(1h)- chinazolinthionen |
FR7631342A FR2328700A1 (fr) | 1975-10-24 | 1976-10-19 | Procede pour la preparation de derives 3,4-dihydro-2-(1h)-quinazolinoniques |
SE7611693A SE422577B (sv) | 1975-10-24 | 1976-10-21 | Forfarande for framstellning av 3,4-dihydro-2(1h)-kinazolinonderivat |
CH1331876A CH601259A5 (US07122603-20061017-C00187.png) | 1975-10-24 | 1976-10-21 | |
DK480976AA DK137534B (da) | 1975-10-24 | 1976-10-22 | Fremgangsmåde til fremstilling af 3,4-dihydro-2(1H)-quinazolinonderivater. |
HU76SU932A HU173529B (hu) | 1975-10-24 | 1976-10-22 | Sposob poluchenija proizvodnykh 3,4-digidro-2/1h/-khinazolina |
DE19762647853 DE2647853A1 (de) | 1975-10-24 | 1976-10-22 | Verfahren zur herstellung von 3,4- dihydro-2-(1h)-chinazolinonen und 3,4-dihydro- 2(1h)-chinazolinthionen |
MX765006U MX3743E (es) | 1975-10-24 | 1976-10-22 | Procedimiento para la preparacion de derivados 3,4-dihidro-2 (lh)-quinazolinona |
CA263,980A CA1049521A (en) | 1975-10-24 | 1976-10-22 | Process for preparing 3,4-dihydro-2(1h)-quinazolinone derivatives |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP50128578A JPS5251379A (en) | 1975-10-24 | 1975-10-24 | Preparation 3,4-dihydro-2(1h)-quinazoline derivates |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS5251379A true JPS5251379A (en) | 1977-04-25 |
JPS5416513B2 JPS5416513B2 (US07122603-20061017-C00187.png) | 1979-06-22 |
Family
ID=14988206
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP50128578A Granted JPS5251379A (en) | 1975-10-24 | 1975-10-24 | Preparation 3,4-dihydro-2(1h)-quinazoline derivates |
Country Status (13)
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5080208A (en) * | 1988-12-22 | 1992-01-14 | Kabushiki Kaisha Tokai-Rika-Denki-Seisakusho | Shift lever apparatus for automatic transmission of vehicle |
WO1998042688A1 (fr) * | 1997-03-26 | 1998-10-01 | Sumitomo Pharmaceuticals Co., Ltd. | Derives de 4-arylmethylene-1,4-dihydro-2h-azine |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5271483A (en) * | 1975-12-11 | 1977-06-14 | Sumitomo Chem Co Ltd | Synthesis of 2(1h)-quinazolinone derivatives |
US4622398A (en) * | 1985-06-24 | 1986-11-11 | Eli Lilly And Company | Dialkylaminotetrahydroquinazoline |
AU2436792A (en) * | 1991-08-16 | 1993-03-16 | Merck & Co., Inc. | Quinazoline derivatives as inhibitors of hiv reverse transcriptase |
IL102764A0 (en) * | 1991-08-16 | 1993-01-31 | Merck & Co Inc | Quinazoline derivatives,and pharmaceutical compositions containing them |
AR038658A1 (es) * | 2001-06-15 | 2005-01-26 | Novartis Ag | Derivados de 4-aril-2(1h) quinazolinona y 4-aril-quinazolina 2-sustituidas, un proceso para su preparacion, composiciones farmaceuticas y el uso de dichos derivados para la preparacion de un medicamento |
EP1394242A3 (en) * | 2002-08-07 | 2004-04-21 | Rohm And Haas Company | Cyclic thioureas and their use as additives for lubricating oils |
GB0230015D0 (en) * | 2002-12-23 | 2003-01-29 | Novartis Ag | Organic compounds |
CA2513708C (en) * | 2003-01-23 | 2011-01-04 | Shire Holdings Ag | Formulation and methods for the treatment of thrombocythemia |
US20060030574A1 (en) * | 2004-08-04 | 2006-02-09 | Shire Holdings Ag | Quinazoline derivatives useful for the treatment of peripheral arterial disease and as phosphodiesterase inhibitors |
US7700608B2 (en) * | 2004-08-04 | 2010-04-20 | Shire Holdings Ag | Quinazoline derivatives and their use in the treatment of thrombocythemia |
US7910597B2 (en) * | 2006-11-28 | 2011-03-22 | Shire Llc | Substituted quinazolines |
US8304420B2 (en) | 2006-11-28 | 2012-11-06 | Shire Llc | Substituted quinazolines for reducing platelet count |
WO2015120059A1 (en) * | 2014-02-04 | 2015-08-13 | Yates Charles Ryan | Inhibitors of paxillin function and related compositions and methods |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3829420A (en) * | 1970-07-13 | 1974-08-13 | Sumitomo Chemical Co | 3,4-dihydro-2(1h)-quinazolinones and preparation thereof |
US3686178A (en) * | 1970-09-16 | 1972-08-22 | Sandoz Ag | Preparation of 4-aryl-2(1h)-quinazolinones and thiones |
US3764600A (en) * | 1970-10-06 | 1973-10-09 | Sandoz Ag | 1-substituted-quinazoline-2(1h)-thiones |
US3748331A (en) * | 1971-05-06 | 1973-07-24 | Sandoz Ag | 1,4-disubstituted-methylenedioxy -2-(1h)-quinazolinones and quinazolinthiones |
-
1975
- 1975-10-24 JP JP50128578A patent/JPS5251379A/ja active Granted
-
1976
- 1976-10-11 NL NL7611210.A patent/NL166934B/xx not_active IP Right Cessation
- 1976-10-12 GB GB42337/76A patent/GB1510068A/en not_active Expired
- 1976-10-12 US US05/731,574 patent/US4202974A/en not_active Expired - Lifetime
- 1976-10-15 AT AT770976A patent/AT353796B/de not_active IP Right Cessation
- 1976-10-19 FR FR7631342A patent/FR2328700A1/fr active Granted
- 1976-10-21 SE SE7611693A patent/SE422577B/xx unknown
- 1976-10-21 CH CH1331876A patent/CH601259A5/xx not_active IP Right Cessation
- 1976-10-22 CA CA263,980A patent/CA1049521A/en not_active Expired
- 1976-10-22 DE DE19762647853 patent/DE2647853A1/de not_active Withdrawn
- 1976-10-22 HU HU76SU932A patent/HU173529B/hu unknown
- 1976-10-22 DK DK480976AA patent/DK137534B/da not_active IP Right Cessation
- 1976-10-22 MX MX765006U patent/MX3743E/es unknown
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5080208A (en) * | 1988-12-22 | 1992-01-14 | Kabushiki Kaisha Tokai-Rika-Denki-Seisakusho | Shift lever apparatus for automatic transmission of vehicle |
WO1998042688A1 (fr) * | 1997-03-26 | 1998-10-01 | Sumitomo Pharmaceuticals Co., Ltd. | Derives de 4-arylmethylene-1,4-dihydro-2h-azine |
Also Published As
Publication number | Publication date |
---|---|
JPS5416513B2 (US07122603-20061017-C00187.png) | 1979-06-22 |
AT353796B (de) | 1979-12-10 |
SE7611693L (sv) | 1977-04-25 |
DE2647853A1 (de) | 1977-05-05 |
DK480976A (US07122603-20061017-C00187.png) | 1977-04-25 |
GB1510068A (en) | 1978-05-10 |
FR2328700B1 (US07122603-20061017-C00187.png) | 1979-03-02 |
NL7611210A (nl) | 1977-04-26 |
DK137534C (US07122603-20061017-C00187.png) | 1978-08-14 |
US4202974A (en) | 1980-05-13 |
CH601259A5 (US07122603-20061017-C00187.png) | 1978-06-30 |
AU1854576A (en) | 1978-02-16 |
NL166934B (nl) | 1981-05-15 |
CA1049521A (en) | 1979-02-27 |
MX3743E (es) | 1981-06-10 |
SE422577B (sv) | 1982-03-15 |
ATA770976A (de) | 1979-05-15 |
FR2328700A1 (fr) | 1977-05-20 |
DK137534B (da) | 1978-03-20 |
HU173529B (hu) | 1979-06-28 |
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