JP7564620B2 - カテコールアミン分泌腫瘍の処置における糖質コルチイド受容体モジレータの使用 - Google Patents
カテコールアミン分泌腫瘍の処置における糖質コルチイド受容体モジレータの使用 Download PDFInfo
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- JP7564620B2 JP7564620B2 JP2019548370A JP2019548370A JP7564620B2 JP 7564620 B2 JP7564620 B2 JP 7564620B2 JP 2019548370 A JP2019548370 A JP 2019548370A JP 2019548370 A JP2019548370 A JP 2019548370A JP 7564620 B2 JP7564620 B2 JP 7564620B2
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- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/575—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
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- A—HUMAN NECESSITIES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
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- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
- A61P5/46—Drugs for disorders of the endocrine system of the suprarenal hormones for decreasing, blocking or antagonising the activity of glucocorticosteroids
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- Chemical & Material Sciences (AREA)
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| JP2022070027A JP2022090003A (ja) | 2017-03-09 | 2022-04-21 | カテコールアミン分泌腫瘍の処置における糖質コルチイド受容体モジレータの使用 |
| JP2024053332A JP2024074854A (ja) | 2017-03-09 | 2024-03-28 | カテコールアミン分泌腫瘍の処置における糖質コルチイド受容体モジレータの使用 |
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| JP2022070027A Withdrawn JP2022090003A (ja) | 2017-03-09 | 2022-04-21 | カテコールアミン分泌腫瘍の処置における糖質コルチイド受容体モジレータの使用 |
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| JP2024053332A Pending JP2024074854A (ja) | 2017-03-09 | 2024-03-28 | カテコールアミン分泌腫瘍の処置における糖質コルチイド受容体モジレータの使用 |
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| SG11202105746TA (en) | 2018-12-20 | 2021-07-29 | Corcept Therapeutics Inc | Methods for imaging and treatment of somatostatin-receptor positive tumors |
| JP2021079146A (ja) * | 2021-02-22 | 2021-05-27 | 株式会社三洋物産 | 遊技機 |
| JP7315071B2 (ja) * | 2021-03-03 | 2023-07-26 | 株式会社三洋物産 | 遊技機 |
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| CA2246791A1 (en) | 1998-09-01 | 2000-03-01 | Alison Buchan | Treatment of endothelium with somatostatin analogues |
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| US6139845A (en) | 1999-12-07 | 2000-10-31 | Allergan Sales, Inc. | Method for treating cancer with a neurotoxin |
| DE60232956D1 (de) | 2001-03-23 | 2009-08-27 | Corcept Therapeutics Inc | Verfahren zur behandlung von stressbedingten erkrankungen unter verwendung von glucocorticoid-rezepto-spezifischen antagonisten |
| US7189856B2 (en) | 2001-12-28 | 2007-03-13 | Gideon Shapiro | Non-peptide somatostatin receptor ligands |
| CA2558899C (en) | 2004-03-09 | 2013-02-05 | Corcept Therapeutics, Inc. | Fused ring azadecalin glucocorticoid receptor modulators |
| GB0428151D0 (en) * | 2004-12-22 | 2005-01-26 | Novartis Ag | Organic compounds |
| US20100178663A1 (en) * | 2007-05-15 | 2010-07-15 | Waters Technologies Corporation | Apparatus And Methods For The Detection Of Plasma Metanephrines |
| US20100261693A1 (en) | 2007-10-17 | 2010-10-14 | Ulmann Andre | Method for treating cushing's syndrome |
| ES2351569B8 (es) | 2009-05-07 | 2012-06-20 | Bcn Peptides S.A. | Ligandos peptídicos de receptores de somatostatina. |
| JP5637568B2 (ja) | 2009-05-12 | 2014-12-10 | コーセプト セラピューティクス， インコーポレイテッド | 固体形態および調製のためのプロセス |
| ES2999020T3 (en) * | 2010-02-05 | 2025-02-24 | Phosphagenics Ltd | Carrier comprising non-neutralised tocopheryl phosphate |
| MY161170A (en) | 2011-03-18 | 2017-04-14 | Corcept Therapeutics Inc | Pyrimidine cyclohexyl glucocorticoid receptor modulators |
| US8859774B2 (en) | 2012-05-25 | 2014-10-14 | Corcept Therapeutics, Inc. | Heteroaryl-ketone fused azadecalin glucocorticoid receptor modulators |
| PL3848027T3 (pl) | 2013-11-25 | 2023-07-24 | Corcept Therapeutics Incorporated | Skondensowane oktahydrozwiązki azadekaliny jako modulatory receptora glukokortykoidowego |
| AU2016226451B2 (en) * | 2015-03-02 | 2019-12-19 | Corcept Therapeutics, Inc. | Use of glucocorticoid receptor antagonist and somatostatin analogues to treat ACTH-secreting tumors |
| US9943526B2 (en) * | 2015-04-21 | 2018-04-17 | Corcept Therapeutics, Inc. | Optimizing mifepristone levels for cushing's patients |
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Patent Citations (1)
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| WO2013039916A1 (en) | 2011-09-12 | 2013-03-21 | The United States Of America, Represented By The Secretary, Dept. Of Health And Human Services | Compositions for and methods of treatment and enhanced detection of non-pituitary tumors |
Non-Patent Citations (1)
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| ＣＬＩＮＩＣＡＬ ＯＢＳＴＥＴＲＩＣＳ ＡＮＤ ＧＹＮＥＣＯＬＯＧＹ，１９９６年，Ｖｏｌ．３９，Ｎｏ．２，ｐｐ．５０６－５１０ |
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| AU2018230429A1 (en) | 2019-09-05 |
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| EP3592358A4 (en) | 2020-12-16 |
| AU2018230429B2 (en) | 2023-06-15 |
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| WO2018165460A1 (en) | 2018-09-13 |
| US20180256604A1 (en) | 2018-09-13 |
| CN110475558A (zh) | 2019-11-19 |
| US11045482B2 (en) | 2021-06-29 |
| CA3053806A1 (en) | 2018-09-13 |
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