JP6321020B2 - 二環式複素環化合物およびそれらの治療での使用 - Google Patents

二環式複素環化合物およびそれらの治療での使用 Download PDF

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Publication number
JP6321020B2
JP6321020B2 JP2015537356A JP2015537356A JP6321020B2 JP 6321020 B2 JP6321020 B2 JP 6321020B2 JP 2015537356 A JP2015537356 A JP 2015537356A JP 2015537356 A JP2015537356 A JP 2015537356A JP 6321020 B2 JP6321020 B2 JP 6321020B2
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methyl
dimethyl
pyrrolo
methylpiperazin
alkyl
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Japanese (ja)
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JP2015534976A5 (enExample
JP2015534976A (ja
Inventor
ジャンニ、チェサーリ
クリストファー、ノルベルト、ジョンソン
リー、ウィリアム、ページ
イルディコ、マリア、バック
ジェームズ、エドワード、ハーベイ、デイ
スティーブン、ハワード
ゴードン、サクスティ
クリストファー、ウィリアム、マレー
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Astex Therapeutics Ltd
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Astex Therapeutics Ltd
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Priority claimed from GBGB1218850.4A external-priority patent/GB201218850D0/en
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Publication of JP2015534976A5 publication Critical patent/JP2015534976A5/ja
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
JP2015537356A 2012-10-19 2013-10-18 二環式複素環化合物およびそれらの治療での使用 Active JP6321020B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201261716084P 2012-10-19 2012-10-19
US61/716,084 2012-10-19
GBGB1218850.4A GB201218850D0 (en) 2012-10-19 2012-10-19 Bicyclic heterocycle compounds and their uses in therapy
GB1218850.4 2012-10-19
GB2013005272 2013-10-18

Publications (3)

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JP2015534976A JP2015534976A (ja) 2015-12-07
JP2015534976A5 JP2015534976A5 (enExample) 2016-12-08
JP6321020B2 true JP6321020B2 (ja) 2018-05-09

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Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3455221B1 (en) * 2016-05-09 2020-03-11 H. Hoffnabb-La Roche Ag Dimeric compounds
CN120247907A (zh) * 2020-05-04 2025-07-04 大塚制药株式会社 Iap拮抗剂化合物和中间体及其合成方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8044209B2 (en) * 2006-10-12 2011-10-25 Novartis Ag Pyrrolydine derivatives as IAP inhibitors

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JP2015534976A (ja) 2015-12-07

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