JP5938422B2 - Pet前駆体の製造 - Google Patents

Pet前駆体の製造 Download PDF

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Publication number
JP5938422B2
JP5938422B2 JP2013557076A JP2013557076A JP5938422B2 JP 5938422 B2 JP5938422 B2 JP 5938422B2 JP 2013557076 A JP2013557076 A JP 2013557076A JP 2013557076 A JP2013557076 A JP 2013557076A JP 5938422 B2 JP5938422 B2 JP 5938422B2
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JP
Japan
Prior art keywords
compound
palladium
catalyst
formula
group
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Active
Application number
JP2013557076A
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English (en)
Japanese (ja)
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JP2014514268A (ja
Inventor
フェアウェイ,スティーブン・マイケル
ローラン−ディスガード,マリット
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GE Healthcare Ltd
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GE Healthcare Ltd
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Publication of JP2014514268A publication Critical patent/JP2014514268A/ja
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Publication of JP5938422B2 publication Critical patent/JP5938422B2/ja
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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/14Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
    • C07C227/16Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions not involving the amino or carboxyl groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/46Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • C07C229/48Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups and carboxyl groups bound to carbon atoms of the same non-condensed ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/0404Lipids, e.g. triglycerides; Polycationic carriers
    • A61K51/0406Amines, polyamines, e.g. spermine, spermidine, amino acids, (bis)guanidines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/06Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/04Systems containing only non-condensed rings with a four-membered ring
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Physics & Mathematics (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Optics & Photonics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
JP2013557076A 2011-03-08 2012-03-07 Pet前駆体の製造 Active JP5938422B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161450177P 2011-03-08 2011-03-08
US61/450,177 2011-03-08
PCT/EP2012/053867 WO2012120025A1 (en) 2011-03-08 2012-03-07 Preparation of a 1-amino-3-hydroxy-cyclobutane-1-carboxylic acid derivative

Publications (2)

Publication Number Publication Date
JP2014514268A JP2014514268A (ja) 2014-06-19
JP5938422B2 true JP5938422B2 (ja) 2016-06-22

Family

ID=45808953

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013557076A Active JP5938422B2 (ja) 2011-03-08 2012-03-07 Pet前駆体の製造

Country Status (14)

Country Link
US (1) US9242924B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EP (1) EP2683684B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (1) JP5938422B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
KR (1) KR101904565B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CN (1) CN103415503B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (1) AU2012224634B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BR (1) BR112013020627B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA2828975C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (1) DK2683684T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (1) ES2657894T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
MX (1) MX341089B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NO (1) NO2683684T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
RU (1) RU2596829C2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
WO (1) WO2012120025A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU4314700A (en) 1999-04-28 2000-11-17 Banyu Pharmaceutical Co., Ltd. Processes for the preparation of piperidylmethylpyridine derivatives
JP4744163B2 (ja) * 2005-02-28 2011-08-10 広栄化学工業株式会社 ビピリジン類の製造方法
TW200736203A (en) 2005-11-18 2007-10-01 Glaxo Group Ltd New pleuromutilin derivative and its use
PL1978015T3 (pl) * 2005-11-29 2018-07-31 Nihon Medi-Physics Co., Ltd. Związek prekursorowy związku organicznego znakowanego radioaktywnym halogenem
EP2128130B1 (en) * 2006-12-27 2018-10-10 Nihon Medi-Physics Co., Ltd. Process for production of precursor compound for radioactive halogen-labeled organic compound
ES2602577T3 (es) 2008-03-11 2017-02-21 Incyte Holdings Corporation Derivados de azetidina y ciclobutano como inhibidores de JAK
CA2741030A1 (en) 2008-10-20 2010-04-29 Marvin C. Gershengorn Low molecular weight thyroid stimulating hormone receptor (tshr) agonists
US20120189546A1 (en) 2009-07-11 2012-07-26 Bayer Pharma Aktiengesellschaft Radiolabelling Method Using Cycloalkyl Groups

Also Published As

Publication number Publication date
ES2657894T3 (es) 2018-03-07
AU2012224634B2 (en) 2016-09-08
KR101904565B1 (ko) 2018-10-04
CN103415503A (zh) 2013-11-27
EP2683684B1 (en) 2018-01-03
EP2683684A1 (en) 2014-01-15
RU2013139061A (ru) 2015-04-20
JP2014514268A (ja) 2014-06-19
NO2683684T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 2018-06-02
RU2596829C2 (ru) 2016-09-10
WO2012120025A1 (en) 2012-09-13
BR112013020627B1 (pt) 2019-12-03
CA2828975A1 (en) 2012-09-13
US9242924B2 (en) 2016-01-26
MX341089B (es) 2016-08-08
KR20140049975A (ko) 2014-04-28
MX2013010254A (es) 2013-11-18
DK2683684T3 (en) 2018-02-05
US20130345468A1 (en) 2013-12-26
CN103415503B (zh) 2015-09-16
BR112013020627A2 (pt) 2016-10-04
CA2828975C (en) 2019-07-09

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