JP5577256B2 - 抗腫瘍化合物 - Google Patents

抗腫瘍化合物 Download PDF

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Publication number
JP5577256B2
JP5577256B2 JP2010537432A JP2010537432A JP5577256B2 JP 5577256 B2 JP5577256 B2 JP 5577256B2 JP 2010537432 A JP2010537432 A JP 2010537432A JP 2010537432 A JP2010537432 A JP 2010537432A JP 5577256 B2 JP5577256 B2 JP 5577256B2
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Japan
Prior art keywords
substituted
unsubstituted
group
carbamate
methyl
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Expired - Fee Related
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JP2010537432A
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English (en)
Japanese (ja)
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JP2011506393A5 (es
JP2011506393A (ja
Inventor
フディット・トゥッラ−プチェ
エレオノーラ・マルクッチ
ヌリア・バヨ−プクサン
フェルナンド・アルベリシオ
マリア・デル・カルメン・クエヴァス・マルチャンテ
Original Assignee
ファルマ・マール・ソシエダード・アノニマ
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Publication of JP2011506393A5 publication Critical patent/JP2011506393A5/ja
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50—Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
JP2010537432A 2007-12-14 2008-12-10 抗腫瘍化合物 Expired - Fee Related JP5577256B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP07380361.1 2007-12-14
EP07380361 2007-12-14
PCT/EP2008/067189 WO2009077401A1 (en) 2007-12-14 2008-12-10 Antitumoral compounds

Publications (3)

Publication Number Publication Date
JP2011506393A JP2011506393A (ja) 2011-03-03
JP2011506393A5 JP2011506393A5 (es) 2013-01-17
JP5577256B2 true JP5577256B2 (ja) 2014-08-20

Family

ID=40290734

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010537432A Expired - Fee Related JP5577256B2 (ja) 2007-12-14 2008-12-10 抗腫瘍化合物

Country Status (9)

Country Link
US (1) US8748388B2 (es)
EP (1) EP2231695B1 (es)
JP (1) JP5577256B2 (es)
CN (1) CN101932592B (es)
AU (1) AU2008337605B2 (es)
CA (1) CA2708080C (es)
ES (1) ES2406107T3 (es)
HK (1) HK1149022A1 (es)
WO (1) WO2009077401A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20110027417A1 (en) 2009-07-31 2011-02-03 Patrick Joseph Corrigan Process for Dusting Animal Food
EP2771478B1 (en) * 2011-10-25 2018-03-14 The Scripps Research Institute Synthesis of libraries of peptide tertiary amides
JOP20190254A1 (ar) 2017-04-27 2019-10-27 Pharma Mar Sa مركبات مضادة للأورام
CN111777668B (zh) * 2020-07-28 2022-02-25 安徽工程大学 一种基于海洋环肽Samoamide A的改造多肽、合成方法及应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5681813A (en) * 1994-04-06 1997-10-28 Pharma Mar, S.A. Thiodepsipeptide isolated from a marine actinomycete
NZ526279A (en) 2000-12-21 2005-01-28 Scripps Research Inst Analogues of thiocoraline and BE-22179

Also Published As

Publication number Publication date
ES2406107T3 (es) 2013-06-05
AU2008337605A1 (en) 2009-06-25
US20100292163A1 (en) 2010-11-18
CN101932592B (zh) 2014-02-26
AU2008337605B2 (en) 2013-08-29
EP2231695B1 (en) 2013-02-13
CA2708080A1 (en) 2009-06-25
WO2009077401A1 (en) 2009-06-25
JP2011506393A (ja) 2011-03-03
EP2231695A1 (en) 2010-09-29
HK1149022A1 (en) 2011-09-23
CN101932592A (zh) 2010-12-29
US8748388B2 (en) 2014-06-10
US20110207674A2 (en) 2011-08-25
CA2708080C (en) 2016-06-14

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