JP5474548B2 - 治療用の置換チアゾリジノン類、オキサゾリジノン類および関連化合物 - Google Patents
治療用の置換チアゾリジノン類、オキサゾリジノン類および関連化合物 Download PDFInfo
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- JP5474548B2 JP5474548B2 JP2009525735A JP2009525735A JP5474548B2 JP 5474548 B2 JP5474548 B2 JP 5474548B2 JP 2009525735 A JP2009525735 A JP 2009525735A JP 2009525735 A JP2009525735 A JP 2009525735A JP 5474548 B2 JP5474548 B2 JP 5474548B2
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Ophthalmology & Optometry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US82329706P | 2006-08-23 | 2006-08-23 | |
| US60/823,297 | 2006-08-23 | ||
| PCT/US2007/076410 WO2008024765A2 (en) | 2006-08-23 | 2007-08-21 | Therapeutic substituted thiazolidinones, oxazolidinones, and related compounds |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| JP2014020352A Division JP2014098020A (ja) | 2006-08-23 | 2014-02-05 | 治療用の置換チアゾリジノン類、オキサゾリジノン類および関連化合物 |
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| Publication Number | Publication Date |
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| JP2010501588A JP2010501588A (ja) | 2010-01-21 |
| JP2010501588A5 JP2010501588A5 (https=) | 2010-10-07 |
| JP5474548B2 true JP5474548B2 (ja) | 2014-04-16 |
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| JP2009525735A Expired - Fee Related JP5474548B2 (ja) | 2006-08-23 | 2007-08-21 | 治療用の置換チアゾリジノン類、オキサゾリジノン類および関連化合物 |
| JP2014020352A Abandoned JP2014098020A (ja) | 2006-08-23 | 2014-02-05 | 治療用の置換チアゾリジノン類、オキサゾリジノン類および関連化合物 |
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| JP2014020352A Abandoned JP2014098020A (ja) | 2006-08-23 | 2014-02-05 | 治療用の置換チアゾリジノン類、オキサゾリジノン類および関連化合物 |
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| EP (1) | EP2054409A2 (https=) |
| JP (2) | JP5474548B2 (https=) |
| AU (1) | AU2007286756B2 (https=) |
| BR (1) | BRPI0715974A2 (https=) |
| CA (1) | CA2661827A1 (https=) |
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| RU2010149494A (ru) | 2008-05-09 | 2012-06-20 | Аллерган, Инк. (Us) | Терапевтические замещенные тиазолидиноны, оксазолидиноны и родственные соединения |
| US7985765B2 (en) * | 2008-08-20 | 2011-07-26 | Allergan, Inc. | Therapeutic substituted pyrroles |
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| US4599353A (en) * | 1982-05-03 | 1986-07-08 | The Trustees Of Columbia University In The City Of New York | Use of eicosanoids and their derivatives for treatment of ocular hypertension and glaucoma |
| US5902726A (en) * | 1994-12-23 | 1999-05-11 | Glaxo Wellcome Inc. | Activators of the nuclear orphan receptor peroxisome proliferator-activated receptor gamma |
| JP2004002206A (ja) * | 2000-07-26 | 2004-01-08 | Chugai Pharmaceut Co Ltd | 光学活性なチアゾリジノン誘導体の製造方法 |
| EP1307193A1 (en) * | 2000-07-27 | 2003-05-07 | Affymax Research Institute | Agonists of follicle stimulating hormone activity |
| AU2003258433A1 (en) | 2002-08-28 | 2004-03-19 | Merck Frosst Canada Ltd | Oxazolidin-2-one and thiazolidin-2-one derivatives for use as ep4 receptor agonists in the treatment of glaucoma |
| CA2599425C (en) | 2005-03-10 | 2013-04-30 | Allergan, Inc. | Substituted gamma lactams as therapeutic agents |
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2007
- 2007-08-21 EP EP07841154A patent/EP2054409A2/en not_active Withdrawn
- 2007-08-21 JP JP2009525735A patent/JP5474548B2/ja not_active Expired - Fee Related
- 2007-08-21 WO PCT/US2007/076410 patent/WO2008024765A2/en not_active Ceased
- 2007-08-21 BR BRPI0715974-9A patent/BRPI0715974A2/pt not_active IP Right Cessation
- 2007-08-21 US US11/842,638 patent/US7659295B2/en active Active
- 2007-08-21 CA CA002661827A patent/CA2661827A1/en not_active Abandoned
- 2007-08-21 AU AU2007286756A patent/AU2007286756B2/en not_active Ceased
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2009
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2014
- 2014-02-05 JP JP2014020352A patent/JP2014098020A/ja not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2008024765A2 (en) | 2008-02-28 |
| WO2008024765A3 (en) | 2008-04-24 |
| US20080058387A1 (en) | 2008-03-06 |
| US20100093809A1 (en) | 2010-04-15 |
| EP2054409A2 (en) | 2009-05-06 |
| AU2007286756B2 (en) | 2013-10-17 |
| JP2010501588A (ja) | 2010-01-21 |
| AU2007286756A1 (en) | 2008-02-28 |
| CA2661827A1 (en) | 2008-02-28 |
| US8003678B2 (en) | 2011-08-23 |
| JP2014098020A (ja) | 2014-05-29 |
| US7659295B2 (en) | 2010-02-09 |
| BRPI0715974A2 (pt) | 2014-09-16 |
| WO2008024765B1 (en) | 2008-06-05 |
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