JP4939398B2 - 金属メソポルフィリンハライド化合物の調製 - Google Patents

金属メソポルフィリンハライド化合物の調製 Download PDF

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JP4939398B2
JP4939398B2 JP2007506137A JP2007506137A JP4939398B2 JP 4939398 B2 JP4939398 B2 JP 4939398B2 JP 2007506137 A JP2007506137 A JP 2007506137A JP 2007506137 A JP2007506137 A JP 2007506137A JP 4939398 B2 JP4939398 B2 JP 4939398B2
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Japan
Prior art keywords
mesoporphyrin
metal
halide
formate
tin
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JP2007506137A
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Japanese (ja)
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JP2007530676A (ja
JP2007530676A5 (https=
Inventor
ヴコヴィッチ，ロバート
レヴィンソン，ベンジャミン
ドラモンド，ジョージ・エス
カロセッリ，ロバート・アール，ピーエイチ．
アンチャック，カジミエシュ・ジー
バウチャー，クリストファー
モーティマー，リチャード
レヴィン，ダニー
クック，キース・エイ
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インファケア・ファーマシューティカル・コーポレイション
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/22—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains four or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
    • C07F15/02—Iron compounds
    • C07F15/025—Iron compounds without a metal-carbon linkage
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/003—Compounds containing elements of Groups 4 or 14 of the Periodic Table without C-Metal linkages

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2007506137A 2004-03-29 2004-11-24 金属メソポルフィリンハライド化合物の調製 Expired - Fee Related JP4939398B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US10/812,156 2004-03-29
US10/812,156 US7375216B2 (en) 2002-06-04 2004-03-29 Preparation of metal mesoporphyrin compounds
PCT/US2004/039240 WO2005103056A2 (en) 2004-03-29 2004-11-24 Preparation of metal mesoporphyrin halide compounds

Publications (3)

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JP2007530676A JP2007530676A (ja) 2007-11-01
JP2007530676A5 JP2007530676A5 (https=) 2008-01-10
JP4939398B2 true JP4939398B2 (ja) 2012-05-23

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JP2007506137A Expired - Fee Related JP4939398B2 (ja) 2004-03-29 2004-11-24 金属メソポルフィリンハライド化合物の調製

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Country Link
US (3) US7375216B2 (https=)
EP (1) EP1730150A4 (https=)
JP (1) JP4939398B2 (https=)
CA (1) CA2561487C (https=)
WO (1) WO2005103056A2 (https=)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8530458B2 (en) 2006-10-04 2013-09-10 Infacare Pharmaceutical Corporation High-purity large-scale preparation of stannsoporfin
US8735574B2 (en) 2011-03-30 2014-05-27 Infacare Pharmaceutical Corporation Methods for synthesizing metal mesoporphyrins

Families Citing this family (11)

* Cited by examiner, † Cited by third party
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US7375216B2 (en) * 2002-06-04 2008-05-20 Infacare Pharmaceutical Corporation Preparation of metal mesoporphyrin compounds
GB2397067B (en) 2002-12-23 2005-05-11 Destiny Pharma Ltd Porphin & azaporphin derivatives with at least one cationic-nitrogen-containing meso-substituent for use in photodynamic therapy & in vitro sterilisation
GB2415372A (en) 2004-06-23 2005-12-28 Destiny Pharma Ltd Non photodynamical or sonodynamical antimicrobial use of porphyrins and azaporphyrins containing at least one cationic-nitrogen-containing substituent
US20060222668A1 (en) * 2005-04-01 2006-10-05 Wellspring Pharmaceutical Corporation Stannsoporfin compositions, drug products and methods of manufacture
EP1865777A4 (en) * 2005-04-01 2008-07-16 Infacare Pharmaceutical Corp STANNSOPORFIN COMPOSITIONS AND ADMINISTRATION
US20070077480A1 (en) * 2005-10-05 2007-04-05 Curello Andrew J Scavenger materials in fuel cartridge
US20080113955A1 (en) * 2006-10-04 2008-05-15 Benjamin Levinson Treatment of infant hyperbilirubinemia using low dosages of stannsoporfin
IT1403087B1 (it) * 2010-11-05 2013-10-04 Lombardi Catalizzatori ad alta efficienza, loro preparazione e uso
AU2012345646A1 (en) 2011-12-01 2014-06-26 Infacare Pharmaceutical Corporation Methods for treating hyperbilirubinemia with stannsoporfin
CN103193783A (zh) * 2013-03-29 2013-07-10 甘肃农业大学 一种以牦牛血粉为原料制备氯化血红素的方法
SI3200582T1 (sl) 2014-09-29 2024-04-30 Fred Hutchinson Cancer Center Sestave, kompleti in metode za indukcijo pridobljene citorezistence z uporabo induktorjev stresnih proteinov

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WO2003101999A2 (en) * 2002-06-04 2003-12-11 Wellspring Pharmaceutical Corporation Preparation of metal mesoporphyrin halide compounds

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US4861876A (en) * 1986-11-26 1989-08-29 Wayne State University Hematoporphyrin derivative and method of preparation and purification
US4782049A (en) * 1986-12-08 1988-11-01 The Rockefeller University Tin protoporphyrin and tin mesoporphyrin in the treatment of psoriasis
US4900871A (en) * 1987-01-02 1990-02-13 Sun Refining And Marketing Company Hydrocarbon oxidations catalyzed by iron coordination complexes containing a halogenated ligand
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US5081115A (en) * 1987-10-15 1992-01-14 The Board Of Trustees Of The Leland Stanford Junior University Method to prevent neonatal jaundice with metalloporphyrin compositions
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DE3827940A1 (de) * 1988-08-13 1990-03-01 Schering Ag 13,17-propionsaeure- und propionsaeurederivat- substituierte porphyrin-komplexverbindungen, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische mittel
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US20060222668A1 (en) * 2005-04-01 2006-10-05 Wellspring Pharmaceutical Corporation Stannsoporfin compositions, drug products and methods of manufacture
US20080113955A1 (en) * 2006-10-04 2008-05-15 Benjamin Levinson Treatment of infant hyperbilirubinemia using low dosages of stannsoporfin
US7960371B2 (en) * 2006-10-04 2011-06-14 Infacare Pharmaceutical Corporation High-purity large-scale preparation of stannsoporfin

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003101999A2 (en) * 2002-06-04 2003-12-11 Wellspring Pharmaceutical Corporation Preparation of metal mesoporphyrin halide compounds

Cited By (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8530458B2 (en) 2006-10-04 2013-09-10 Infacare Pharmaceutical Corporation High-purity large-scale preparation of stannsoporfin
US8835416B2 (en) 2006-10-04 2014-09-16 Infacare Pharmaceutical Corporation High-purity large-scale preparation of stannsoporfin
US9107927B2 (en) 2006-10-04 2015-08-18 Infacare Pharmaceutical Corporation High-purity large-scale preparation of stannsoporfin
US9517239B2 (en) 2006-10-04 2016-12-13 Infacare Pharmaceutical Corporation High-purity large-scale preparation of stannsoporfin
US9902745B2 (en) 2006-10-04 2018-02-27 Infacare Pharmaceutical Corporation High-purity large-scale preparation of stannsoporfin
US10273255B2 (en) 2006-10-04 2019-04-30 Infacare Pharmaceutical Corporation High-purity large-scale preparation of stannsoporfin
US10662209B2 (en) 2006-10-04 2020-05-26 Mallinckrodt Hospital Products IP Limited High-purity large-scale preparation of stannsoporfin
US11078220B2 (en) 2006-10-04 2021-08-03 Mallinckrodt Hospital Products IP Limited High-purity large-scale preparation of stannsoporfin
US8735574B2 (en) 2011-03-30 2014-05-27 Infacare Pharmaceutical Corporation Methods for synthesizing metal mesoporphyrins
US9181285B2 (en) 2011-03-30 2015-11-10 Infacare Pharmaceutical Corporation Methods for synthesizing metal mesoporphyrins
US9688705B2 (en) 2011-03-30 2017-06-27 Infacare Pharmaceutical Corporation Methods for synthesizing metal mesoporphyrins
US10533024B2 (en) 2011-03-30 2020-01-14 Mallinckrodt Hosptial Products Ip Limited Methods for synthesizing metal mesoporphyrins

Also Published As

Publication number Publication date
US7777028B2 (en) 2010-08-17
US8178664B2 (en) 2012-05-15
EP1730150A2 (en) 2006-12-13
EP1730150A4 (en) 2011-05-04
JP2007530676A (ja) 2007-11-01
WO2005103056A3 (en) 2007-05-10
WO2005103056A2 (en) 2005-11-03
CA2561487C (en) 2012-05-01
US20040210048A1 (en) 2004-10-21
US20080154033A1 (en) 2008-06-26
CA2561487A1 (en) 2005-11-03
US20100280237A1 (en) 2010-11-04
US7375216B2 (en) 2008-05-20

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