JP4532910B2 - エタン−１，２−ジアミニウムビス［（２ｒ）−２−ブロモ−３−フェニルプロパノエート］、その製造方法およびその使用 - Google Patents

エタン−１，２−ジアミニウムビス［（２ｒ）−２−ブロモ−３−フェニルプロパノエート］、その製造方法およびその使用 Download PDF

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JP4532910B2
JP4532910B2 JP2003576439A JP2003576439A JP4532910B2 JP 4532910 B2 JP4532910 B2 JP 4532910B2 JP 2003576439 A JP2003576439 A JP 2003576439A JP 2003576439 A JP2003576439 A JP 2003576439A JP 4532910 B2 JP4532910 B2 JP 4532910B2
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bromo
phenylpropanoate
ethane
phenylpropionic acid
formula
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Japanese (ja)
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JP2005528358A5 (https=
JP2005528358A (ja
Inventor
ハビエル・マーネロ
トビーアス・メッツェンティン
ライナー・ガウラー
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サノフィ−アベンティス・ドイチュラント・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/62—Quaternary ammonium compounds
    • C07C211/63—Quaternary ammonium compounds having quaternised nitrogen atoms bound to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
JP2003576439A 2002-03-19 2003-03-07 エタン−１，２−ジアミニウムビス［（２ｒ）−２−ブロモ−３−フェニルプロパノエート］、その製造方法およびその使用 Expired - Fee Related JP4532910B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10212198A DE10212198A1 (de) 2002-03-19 2002-03-19 Ethan-1-diaminium-bis(2R)-2-brom-3-phenylpropanoat), Verfahren zu dessen Herstellung und dessen Verwendung
PCT/EP2003/002353 WO2003078434A1 (de) 2002-03-19 2003-03-07 Ethan-1,2-diaminium-bis[(2r)-2-brom-3-phenylpropanoat],verfahren zu dessen herstellung und dessen verwendung

Publications (3)

Publication Number Publication Date
JP2005528358A JP2005528358A (ja) 2005-09-22
JP2005528358A5 JP2005528358A5 (https=) 2006-04-20
JP4532910B2 true JP4532910B2 (ja) 2010-08-25

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Family Applications (1)

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JP2003576439A Expired - Fee Related JP4532910B2 (ja) 2002-03-19 2003-03-07 エタン−１，２−ジアミニウムビス［（２ｒ）−２−ブロモ−３−フェニルプロパノエート］、その製造方法およびその使用

Country Status (10)

Country Link
EP (1) EP1487836B1 (https=)
JP (1) JP4532910B2 (https=)
AT (1) ATE338756T1 (https=)
AU (1) AU2003219027A1 (https=)
BR (1) BR0308485A (https=)
CA (1) CA2479620A1 (https=)
DE (2) DE10212198A1 (https=)
IL (1) IL164042A0 (https=)
MX (1) MXPA04008490A (https=)
WO (1) WO2003078434A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5726530B2 (ja) * 2007-12-05 2015-06-03 クゥアルコム・インコーポレイテッドＱｕａｌｃｏｍｍ Ｉｎｃｏｒｐｏｒａｔｅｄ 全地球ナビゲーション受信機

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2678759B2 (ja) * 1988-02-23 1997-11-17 日本合成化学工業株式会社 固体状高分子化合物のアンモニウム塩類の製造法
CA2053340C (en) * 1990-10-18 2002-04-02 Timothy P. Burkholder Mercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace
JPH1014590A (ja) * 1996-06-28 1998-01-20 Kanegafuchi Chem Ind Co Ltd 光学活性２−置換−３−フェニルプロピオン酸及びそのエステルの製造方法
IT1298267B1 (it) * 1998-02-18 1999-12-20 Zambon Spa Procedimento per la preparazione dell'acido (s)-2-acetiltio-3-fenil- propionico e dei suoi sali
NL1014354C2 (nl) * 2000-02-11 2001-08-14 Dsm Nv Werkwijze voor de bereiding van (S) -2-acethylthio-3-fenylpropaanzuur.
NL1014353C2 (nl) * 2000-02-11 2001-08-15 Dsm Nv Werkwijze voor de bereiding van (R) -2-broom-3-fenylpropaanzuur.

Also Published As

Publication number Publication date
WO2003078434A1 (de) 2003-09-25
CA2479620A1 (en) 2003-09-25
EP1487836B1 (de) 2006-09-06
IL164042A0 (en) 2005-12-18
ATE338756T1 (de) 2006-09-15
DE50304950D1 (de) 2006-10-19
AU2003219027A1 (en) 2003-09-29
DE10212198A1 (de) 2003-10-02
MXPA04008490A (es) 2004-12-06
BR0308485A (pt) 2005-01-18
EP1487836A1 (de) 2004-12-22
JP2005528358A (ja) 2005-09-22

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