JP4191825B2 - ５−アミノイソキサゾール誘導体 - Google Patents

５−アミノイソキサゾール誘導体 Download PDF

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Publication number
JP4191825B2
JP4191825B2 JP27246798A JP27246798A JP4191825B2 JP 4191825 B2 JP4191825 B2 JP 4191825B2 JP 27246798 A JP27246798 A JP 27246798A JP 27246798 A JP27246798 A JP 27246798A JP 4191825 B2 JP4191825 B2 JP 4191825B2
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JP
Japan
Prior art keywords
group
isoxazole
pyridyl
fluorophenyl
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP27246798A
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English (en)
Japanese (ja)
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JP2000086657A5 (enExample
JP2000086657A (ja
Inventor
信義 南
通隆 佐藤
幸市 蓮見
則夫 山本
勝幸 慶野
照明 松井
有弘 金田
修治 太田
教久 斎藤
秀一郎 佐藤
章 朝烏
知 土井
基博 小林
潤 佐藤
創 浅野
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aska Pharmaceutical Co Ltd
Original Assignee
Aska Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aska Pharmaceutical Co Ltd filed Critical Aska Pharmaceutical Co Ltd
Priority to JP27246798A priority Critical patent/JP4191825B2/ja
Publication of JP2000086657A publication Critical patent/JP2000086657A/ja
Publication of JP2000086657A5 publication Critical patent/JP2000086657A5/ja
Application granted granted Critical
Publication of JP4191825B2 publication Critical patent/JP4191825B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP27246798A 1998-09-10 1998-09-10 ５−アミノイソキサゾール誘導体 Expired - Lifetime JP4191825B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP27246798A JP4191825B2 (ja) 1998-09-10 1998-09-10 ５−アミノイソキサゾール誘導体

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP27246798A JP4191825B2 (ja) 1998-09-10 1998-09-10 ５−アミノイソキサゾール誘導体

Publications (3)

Publication Number Publication Date
JP2000086657A JP2000086657A (ja) 2000-03-28
JP2000086657A5 JP2000086657A5 (enExample) 2005-10-20
JP4191825B2 true JP4191825B2 (ja) 2008-12-03

Family

ID=17514333

Family Applications (1)

Application Number Title Priority Date Filing Date
JP27246798A Expired - Lifetime JP4191825B2 (ja) 1998-09-10 1998-09-10 ５−アミノイソキサゾール誘導体

Country Status (1)

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JP (1) JP4191825B2 (enExample)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2420042A1 (en) * 2000-08-22 2003-02-18 Mikio Ogawa Carboxylic acid derivatives, processes for the preparation thereof and pharmaceutical agents comprising the same as active ingredient
WO2002020462A1 (en) * 2000-09-01 2002-03-14 Ono Pharmaceutical Co., Ltd. Benzoic acid derivatives and drugs containing the same as the active ingredient
NZ525016A (en) 2000-09-15 2004-10-29 Vertex Pharma Isoxazoles and their use as inhibitors of ERK
EP1345603A4 (en) * 2000-12-20 2004-09-08 Merck & Co Inc (HALO-BENZO-CARBONYL) HETEROCYCLO-CONDENSED PHENYL-P38-KINASE INHIBITING AGENTS
SE0102764D0 (sv) 2001-08-17 2001-08-17 Astrazeneca Ab Compounds
AU2003245989A1 (en) 2002-07-09 2004-01-23 Boehringer Ingelheim Pharma Gmbh And Co. Kg Pharmaceutical compositions of anticholinergics and p38 kinase inhibitors in the treatment of respiratory diseases
GB0226931D0 (en) 2002-11-19 2002-12-24 Astrazeneca Ab Chemical compounds
GB0226930D0 (en) 2002-11-19 2002-12-24 Astrazeneca Ab Chemical compounds
TW200600086A (en) 2004-06-05 2006-01-01 Astrazeneca Ab Chemical compound
US20060035893A1 (en) 2004-08-07 2006-02-16 Boehringer Ingelheim International Gmbh Pharmaceutical compositions for treatment of respiratory and gastrointestinal disorders
CA2581619A1 (en) 2004-10-16 2006-04-20 Astrazeneca Ab Process for making phenoxy benzamide compounds
PE20060777A1 (es) 2004-12-24 2006-10-06 Boehringer Ingelheim Int Derivados de indolinona para el tratamiento o la prevencion de enfermedades fibroticas
ES2375633T3 (es) * 2004-12-28 2012-03-02 Aska Pharmaceutical Co., Ltd. Derivado de pirimidinilisoxazol.
EP1919882A2 (en) 2005-02-17 2008-05-14 Synta Pharmaceuticals Corporation Isoxazole combretastatin derivatives for the treatment of proliferative disorders
TW200714597A (en) 2005-05-27 2007-04-16 Astrazeneca Ab Chemical compounds
NZ564608A (en) 2005-07-09 2009-09-25 Astrazeneca Ab Heteroaryl benzamide derivatives for use as GLK activators in the treatment of diabetes
AU2006306991A1 (en) 2005-10-28 2007-05-03 Takeda Pharmaceutical Company Limited Heterocyclic amide compound and use thereof
TW200738621A (en) 2005-11-28 2007-10-16 Astrazeneca Ab Chemical process
RU2416600C2 (ru) * 2005-12-27 2011-04-20 Универсидад Дель Паис Васко-Еускал Еррико Унибертситатеа (Упв-Ееу) Новые производные пиррола с ингибирующей гистондеацетилазу активностью
ES2396251T3 (es) 2006-06-28 2013-02-20 Aska Pharmaceutical Co., Ltd. Derivado de piridilisoxazol
JPWO2008001929A1 (ja) * 2006-06-28 2009-12-03 あすか製薬株式会社 炎症性腸疾患の処置剤
TW200825063A (en) 2006-10-23 2008-06-16 Astrazeneca Ab Chemical compounds
SA07280576B1 (ar) 2006-10-26 2011-06-22 استرازينيكا ايه بي مركبات بنزويل أمينو سيكليل غير متجانسة بأعتبارها عوامل منشطة للجلوكوكيناز
JP2010513445A (ja) 2006-12-21 2010-04-30 アストラゼネカ アクチボラグ Ｇｌｋアクチベーターとして有用な新規結晶性化合物
AU2008215659B2 (en) 2007-02-16 2012-11-01 Aska Pharmaceutical Co., Ltd. Pharmaceutical composition comprising microparticle oily suspension
EP1992344A1 (en) 2007-05-18 2008-11-19 Institut Curie P38 alpha as a therapeutic target in pathologies linked to FGFR3 mutation
MX2009012847A (es) * 2007-06-13 2009-12-08 Bristol Myers Squibb Co Analogos dipeptidicos como inhibidores de factores de coagulacion.
JP2011529955A (ja) 2008-08-04 2011-12-15 アストラゼネカ アクチボラグ 治療薬４１４
GB0902406D0 (en) 2009-02-13 2009-04-01 Astrazeneca Ab Crystalline polymorphic form
GB0902434D0 (en) 2009-02-13 2009-04-01 Astrazeneca Ab Chemical process
WO2010116176A1 (en) 2009-04-09 2010-10-14 Astrazeneca Ab Pyrazolo [4, 5-e] pyrimidine derivative and its use to treat diabetes and obesity
WO2010116177A1 (en) 2009-04-09 2010-10-14 Astrazeneca Ab A pyrazolo [4,5-e] pyrimidine derivative and its use to treat diabetes and obesity
CA3070938A1 (en) 2017-07-26 2019-01-31 The Doshisha Drug for treating or preventing disorder caused by tgf-.beta. signalling, and application thereof

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Publication number Publication date
JP2000086657A (ja) 2000-03-28

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