JP2025509955A - リン酸ヒドロコルチゾンナトリウム及びモノチオグリセロール水性医薬製剤 - Google Patents

リン酸ヒドロコルチゾンナトリウム及びモノチオグリセロール水性医薬製剤 Download PDF

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Publication number
JP2025509955A
JP2025509955A JP2024556125A JP2024556125A JP2025509955A JP 2025509955 A JP2025509955 A JP 2025509955A JP 2024556125 A JP2024556125 A JP 2024556125A JP 2024556125 A JP2024556125 A JP 2024556125A JP 2025509955 A JP2025509955 A JP 2025509955A
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JP
Japan
Prior art keywords
sodium phosphate
hydrocortisone
pharmaceutical formulation
monothioglycerol
clause
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
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JP2024556125A
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English (en)
Japanese (ja)
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JP2025509955A5 (https=
Inventor
チェン,シャオミン
オング,シャオウェイ
Original Assignee
アンタレス・ファーマ・インコーポレーテッド
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Application filed by アンタレス・ファーマ・インコーポレーテッド filed Critical アンタレス・ファーマ・インコーポレーテッド
Priority claimed from PCT/US2023/064771 external-priority patent/WO2023183807A1/en
Publication of JP2025509955A publication Critical patent/JP2025509955A/ja
Publication of JP2025509955A5 publication Critical patent/JP2025509955A5/ja
Pending legal-status Critical Current

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183Amino acids, e.g. glycine, EDTA or aspartame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/20Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing sulfur, e.g. dimethyl sulfoxide [DMSO], docusate, sodium lauryl sulfate or aminosulfonic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
JP2024556125A 2022-03-21 2023-03-21 リン酸ヒドロコルチゾンナトリウム及びモノチオグリセロール水性医薬製剤 Pending JP2025509955A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US202263321997P 2022-03-21 2022-03-21
US63/321,997 2022-03-21
US202263322934P 2022-03-23 2022-03-23
US63/322,934 2022-03-23
US202263387727P 2022-12-16 2022-12-16
US63/387,727 2022-12-16
PCT/US2023/064771 WO2023183807A1 (en) 2022-03-21 2023-03-21 Aqueous pharmaceutical formulation of hydrocortisone sodium phosphate and monothioglycerol

Publications (2)

Publication Number Publication Date
JP2025509955A true JP2025509955A (ja) 2025-04-11
JP2025509955A5 JP2025509955A5 (https=) 2026-03-31

Family

ID=88094934

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024556125A Pending JP2025509955A (ja) 2022-03-21 2023-03-21 リン酸ヒドロコルチゾンナトリウム及びモノチオグリセロール水性医薬製剤

Country Status (4)

Country Link
US (3) US12102643B2 (https=)
EP (1) EP4496575A4 (https=)
JP (1) JP2025509955A (https=)
CA (1) CA3246335A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2025509955A (ja) * 2022-03-21 2025-04-11 アンタレス・ファーマ・インコーポレーテッド リン酸ヒドロコルチゾンナトリウム及びモノチオグリセロール水性医薬製剤

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2970944A (en) 1958-04-04 1961-02-07 Merck & Co Inc Parenteral solutions of steroid phosphates stabilized with creatinines
IL34366A (en) * 1969-05-07 1973-06-29 Lepetit Spa Stable aqueous 21-hydroxy steroid phosphate solutions
US5173488A (en) 1989-08-21 1992-12-22 American Cyanamid Company Stable injectable pharmaceutical formulation for folic acid and leucovorin salts and method
US5733572A (en) 1989-12-22 1998-03-31 Imarx Pharmaceutical Corp. Gas and gaseous precursor filled microspheres as topical and subcutaneous delivery vehicles
US6090800A (en) 1997-05-06 2000-07-18 Imarx Pharmaceutical Corp. Lipid soluble steroid prodrugs
US20020039594A1 (en) 1997-05-13 2002-04-04 Evan C. Unger Solid porous matrices and methods of making and using the same
CN101132820B (zh) 2005-01-24 2010-05-19 安塔雷斯制药公司 预充式针辅助喷射注入器
JP2009514969A (ja) 2005-11-09 2009-04-09 コンビナトアールエックス インコーポレーティッド 医学的状態を治療するための方法、組成物、およびキット
EP2990067B1 (en) 2008-03-10 2019-09-04 Antares Pharma, Inc. Injector safety device
AU2010226442A1 (en) 2009-03-20 2011-10-13 Antares Pharma, Inc. Hazardous agent injection system
US10300207B2 (en) 2013-03-13 2019-05-28 Antares Pharma, Inc. Multiple dosage injector with rotating screw dosage system
ES2673290T3 (es) 2016-01-11 2018-06-21 Lamda Laboratories S.A. Soluciones farmacéuticas orales que contienen fosfato sódico de hidrocortisona
FR3047904B1 (fr) 2016-02-18 2018-03-23 Crossject Dispositif d’injection sans aiguille a membrane coulissante
FR3057775B1 (fr) * 2016-10-26 2018-11-02 Crossject Solution pharmaceutique d’hydrocortisone pour dispositif d’injection
US11814341B2 (en) 2018-05-04 2023-11-14 Ohio State Innovation Foundation Non-peptidic cell-penetrating motifs
US11034710B2 (en) 2018-12-04 2021-06-15 Sumitomo Dainippon Pharma Oncology, Inc. CDK9 inhibitors and polymorphs thereof for use as agents for treatment of cancer
MX2023003197A (es) 2020-09-21 2023-08-04 Antares Pharma Inc Formulacion farmaceutica acuosa de fosfato sodico de hidrocortisona y monotioglicerol.
FR3128874B1 (fr) 2021-11-09 2025-04-18 Crossject Solution pharmaceutique d’hydrocortisone pour dispositif d’injection
JP2025509955A (ja) * 2022-03-21 2025-04-11 アンタレス・ファーマ・インコーポレーテッド リン酸ヒドロコルチゾンナトリウム及びモノチオグリセロール水性医薬製剤

Also Published As

Publication number Publication date
CA3246335A1 (en) 2023-09-28
US20230302016A1 (en) 2023-09-28
US20260091042A1 (en) 2026-04-02
EP4496575A4 (en) 2026-04-01
EP4496575A1 (en) 2025-01-29
US20240238311A1 (en) 2024-07-18
US12521404B2 (en) 2026-01-13
US12102643B2 (en) 2024-10-01

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