JP2025506667A5 - - Google Patents

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Publication number
JP2025506667A5
JP2025506667A5 JP2024547925A JP2024547925A JP2025506667A5 JP 2025506667 A5 JP2025506667 A5 JP 2025506667A5 JP 2024547925 A JP2024547925 A JP 2024547925A JP 2024547925 A JP2024547925 A JP 2024547925A JP 2025506667 A5 JP2025506667 A5 JP 2025506667A5
Authority
JP
Japan
Prior art keywords
alkyl
optionally substituted
represented
pharmaceutically acceptable
acceptable salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024547925A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025506667A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2023/012879 external-priority patent/WO2023154499A1/en
Publication of JP2025506667A publication Critical patent/JP2025506667A/ja
Publication of JP2025506667A5 publication Critical patent/JP2025506667A5/ja
Pending legal-status Critical Current

Links

JP2024547925A 2022-02-14 2023-02-13 エモパミル結合タンパク質阻害剤及びその使用 Pending JP2025506667A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263309923P 2022-02-14 2022-02-14
US63/309,923 2022-02-14
PCT/US2023/012879 WO2023154499A1 (en) 2022-02-14 2023-02-13 Emopamil-binding protein inhibitors and uses thereof

Publications (2)

Publication Number Publication Date
JP2025506667A JP2025506667A (ja) 2025-03-13
JP2025506667A5 true JP2025506667A5 (cg-RX-API-DMAC10.html) 2026-02-24

Family

ID=85505736

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024547925A Pending JP2025506667A (ja) 2022-02-14 2023-02-13 エモパミル結合タンパク質阻害剤及びその使用

Country Status (5)

Country Link
US (1) US20250152574A1 (cg-RX-API-DMAC10.html)
EP (1) EP4479384A1 (cg-RX-API-DMAC10.html)
JP (1) JP2025506667A (cg-RX-API-DMAC10.html)
CN (1) CN119731156A (cg-RX-API-DMAC10.html)
WO (1) WO2023154499A1 (cg-RX-API-DMAC10.html)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UY40865A (es) * 2023-08-23 2025-02-14 Biogen Ma Inc Inhibidores de la proteína de unión al emopamilo y usos de estos
EP4766448A1 (en) * 2023-08-25 2026-07-01 Biogen MA Inc. EMOPAMIL-BINDING PROTEIN INHIBITORS AND THEIR USES
WO2025049419A1 (en) * 2023-08-28 2025-03-06 Genzyme Corporation Pyrazolyl compounds as emopamil binding protein inhibitors
WO2026112292A1 (en) * 2024-11-20 2026-05-28 Convelo Therapeutics, Inc. Spirocyclic compounds for use in promoting remyelination

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10082496B2 (en) * 2014-09-10 2018-09-25 Board Of Regents Of The University Of Texas System Targeting emopamil binding protein (EBP) with small molecules that induce an abnormal feedback response by lowering endogenous cholesterol biosynthesis
MA44037B1 (fr) * 2016-06-06 2020-03-31 Arena Pharm Inc Modulateurs du récepteur adrénergique bêta 3 utile dans le traitement ou la prévention de troubles associés à ceux-ci

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