JP2022551067A - カンナビノイド誘導体 - Google Patents
カンナビノイド誘導体 Download PDFInfo
- Publication number
- JP2022551067A JP2022551067A JP2022520063A JP2022520063A JP2022551067A JP 2022551067 A JP2022551067 A JP 2022551067A JP 2022520063 A JP2022520063 A JP 2022520063A JP 2022520063 A JP2022520063 A JP 2022520063A JP 2022551067 A JP2022551067 A JP 2022551067A
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- hydroxy
- benzo
- pentyl
- chromene
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/78—Ring systems having three or more relevant rings
- C07D311/80—Dibenzopyrans; Hydrogenated dibenzopyrans
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962909370P | 2019-10-02 | 2019-10-02 | |
| US62/909,370 | 2019-10-02 | ||
| PCT/CA2020/051328 WO2021062557A1 (en) | 2019-10-02 | 2020-10-02 | Cannabinoid derivatives |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022551067A true JP2022551067A (ja) | 2022-12-07 |
| JP2022551067A5 JP2022551067A5 (https=) | 2023-10-11 |
| JPWO2021062557A5 JPWO2021062557A5 (https=) | 2023-10-11 |
Family
ID=75336679
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022520063A Pending JP2022551067A (ja) | 2019-10-02 | 2020-10-02 | カンナビノイド誘導体 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US20220340582A1 (https=) |
| EP (1) | EP4038058A4 (https=) |
| JP (1) | JP2022551067A (https=) |
| WO (1) | WO2021062557A1 (https=) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3997098A4 (en) | 2019-07-12 | 2023-10-11 | Canopy Growth Corporation | CANNABINOIDS DERIVATIVES |
| WO2021007663A1 (en) | 2019-07-12 | 2021-01-21 | Canopy Growth Corporation | Cannabinoid derivatives |
| JP2022540586A (ja) | 2019-07-12 | 2022-09-16 | キャノピー グロウス コーポレイション | カンナビノイド誘導体 |
| WO2021062559A1 (en) | 2019-10-02 | 2021-04-08 | Canopy Growth Corporation | Cannabinoid derivatives |
| EP4065554A4 (en) | 2019-11-26 | 2024-01-10 | Canopy Growth Corporation | CANNABIGEROL DERIVATIVES AND THEIR USE AS CANNABINOID RECEPTOR MODULATORS |
| KR20240096817A (ko) | 2020-05-19 | 2024-06-26 | 사이빈 아이알엘 리미티드 | 중수소화된 트립타민 유도체 및 사용 방법 |
| US20240317701A1 (en) | 2020-12-17 | 2024-09-26 | Nalu Bio, Inc. | Synthesis of cannabidiol and analogs thereof, and related compounds, formulations, and methods of use |
| US12091396B1 (en) * | 2021-10-07 | 2024-09-17 | Adam Woodson | System and method for reacting one or more compounds to form tetrahydrocannabinolic acid (THCA) |
| CA3237951A1 (en) * | 2021-11-10 | 2023-05-19 | Mahmoud Mohamed Abdrabo MOUSTAFA | New cannabinoid-gabapentinoid conjugates and uses thereof |
| EP4434975A4 (en) * | 2021-11-16 | 2025-11-05 | K Medichem Co Ltd | NEW CANABICHROMENIC ACID DERIVATIVE, ASSOCIATED PREPARATION PROCESS, AND COMPOSITION COMPRISING THEREOF INTENDED TO IMPROVE COGNITIVE FUNCTION |
| AU2024236787A1 (en) * | 2023-03-15 | 2025-09-18 | Bessor Pharma, Llc | Analogs of cannabichromene and cannabichromenic acid and process of preparing |
Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006012176A1 (en) * | 2004-06-24 | 2006-02-02 | Virginia Commonwealth University | Water-soluble cannabinoids |
| WO2014039042A1 (en) * | 2012-09-06 | 2014-03-13 | Northeastern University | Novel cannabinergic compounds and uses thereof |
| WO2014134127A1 (en) * | 2013-02-26 | 2014-09-04 | Northeastern University | Cannabinergic nitrate esters and related analogs |
| WO2019234728A1 (en) * | 2018-06-04 | 2019-12-12 | Al&Am Pharmachem Ltd. | Cannabinolic acid derivatives and uses thereof |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2021007659A1 (en) * | 2019-07-12 | 2021-01-21 | Canopy Growth Corporation | Cannabinoid derivatives |
-
2020
- 2020-10-02 EP EP20872491.4A patent/EP4038058A4/en active Pending
- 2020-10-02 JP JP2022520063A patent/JP2022551067A/ja active Pending
- 2020-10-02 WO PCT/CA2020/051328 patent/WO2021062557A1/en not_active Ceased
- 2020-10-02 US US17/765,853 patent/US20220340582A1/en active Pending
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006012176A1 (en) * | 2004-06-24 | 2006-02-02 | Virginia Commonwealth University | Water-soluble cannabinoids |
| WO2014039042A1 (en) * | 2012-09-06 | 2014-03-13 | Northeastern University | Novel cannabinergic compounds and uses thereof |
| WO2014134127A1 (en) * | 2013-02-26 | 2014-09-04 | Northeastern University | Cannabinergic nitrate esters and related analogs |
| WO2019234728A1 (en) * | 2018-06-04 | 2019-12-12 | Al&Am Pharmachem Ltd. | Cannabinolic acid derivatives and uses thereof |
Non-Patent Citations (6)
| Title |
|---|
| DATABASE REGISTRY [ONLINE] RETRIEVED FROM STN, JPN7024004035, January 2017 (2017-01-01), ISSN: 0005426712 * |
| JACEK SOSNICKI, TADEUSZ JAGODZINSKI AND MIROSLAWA KROLIKOWSKA: "Thioamide derivatives of cannabinoids. A study of the infl uence of the thethioamide function on reg", JOURNAL OF HETROCYCLIC CHEMISTRY, vol. 36(4), JPN6024038760, August 1999 (1999-08-01), US, pages 1033 - 1041, ISSN: 0005426710 * |
| MALTE ROSENTHAL, FRANZISKA PFEIFFER AND GGNTER MAYER: "A Receptor-Guided Design Strategy for Ligand Identification", ANGEWANDTE CHEMIE INTERNATIONAL EDITION, vol. 58(31), JPN6024038762, 26 June 2019 (2019-06-26), DE, pages 10752 - 10755, ISSN: 0005426713 * |
| OSAMU MORINAGA, WARAPORN PUTALUN, NORIKO FUKUDA, SHAO-JIE SHAN, YUH KANETSUKI, HIROYUKI TANAKA AND Y: "Development of analytical system for pharmacologically active compounds using monoclonal antibodies", CURRENT TOPICS IN ANALYTICAL CHEMISTRY, vol. 2, JPN7024004036, 2001, pages 147 - 158, ISSN: 0005426714 * |
| YECHIEL GAONI AND RAPHAEL MECHOULAM: "Isolation and structure of .DELTA.+- tetrahydrocannabinol and other neutral cannabinoids from hashis", JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, vol. 93(1), JPN6024038761, 13 January 1971 (1971-01-13), US, pages 217 - 224, ISSN: 0005426711 * |
| YURI GOTO, YUMI SHIMA, SATOSHI MORIMOTO, YUKIHIRO SHOYAMA, HIROKI MURAKAMI, AKIHIKO KUSAI AND KAZUTE: "Determination of tetrahydrocannabinolic acid-carrier protein conjugate by matrix-assisted laser deso", ORGANIC MASS SPECTROMETRY, vol. 29(11), JPN6024038763, 1994, pages 668 - 671, ISSN: 0005426715 * |
Also Published As
| Publication number | Publication date |
|---|---|
| EP4038058A4 (en) | 2023-10-25 |
| WO2021062557A1 (en) | 2021-04-08 |
| US20220340582A1 (en) | 2022-10-27 |
| EP4038058A1 (en) | 2022-08-10 |
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