JP2022538576A5 - - Google Patents

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Publication number
JP2022538576A5
JP2022538576A5 JP2021576779A JP2021576779A JP2022538576A5 JP 2022538576 A5 JP2022538576 A5 JP 2022538576A5 JP 2021576779 A JP2021576779 A JP 2021576779A JP 2021576779 A JP2021576779 A JP 2021576779A JP 2022538576 A5 JP2022538576 A5 JP 2022538576A5
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JP
Japan
Prior art keywords
pharmaceutically acceptable
acceptable salt
compound
chloro
fluoro
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021576779A
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English (en)
Japanese (ja)
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JP7498199B2 (ja
JP2022538576A (ja
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Application filed filed Critical
Priority claimed from PCT/IB2020/055974 external-priority patent/WO2020261144A1/en
Publication of JP2022538576A publication Critical patent/JP2022538576A/ja
Publication of JP2022538576A5 publication Critical patent/JP2022538576A5/ja
Application granted granted Critical
Publication of JP7498199B2 publication Critical patent/JP7498199B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2021576779A 2019-06-28 2020-06-24 種々の疾患を処置するために有用なbckdk阻害剤としての5-(チオフェン-2-イル)-1h-テトラゾール誘導体 Active JP7498199B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201962868542P 2019-06-28 2019-06-28
US62/868,542 2019-06-28
US202062960824P 2020-01-14 2020-01-14
US62/960,824 2020-01-14
PCT/IB2020/055974 WO2020261144A1 (en) 2019-06-28 2020-06-24 5-(thiophen-2-yl)-1h-tetrazole derivatives as bckdk inhibitors useful for treating various diseases

Publications (3)

Publication Number Publication Date
JP2022538576A JP2022538576A (ja) 2022-09-05
JP2022538576A5 true JP2022538576A5 (https=) 2023-06-02
JP7498199B2 JP7498199B2 (ja) 2024-06-11

Family

ID=71738227

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021576779A Active JP7498199B2 (ja) 2019-06-28 2020-06-24 種々の疾患を処置するために有用なbckdk阻害剤としての5-(チオフェン-2-イル)-1h-テトラゾール誘導体

Country Status (5)

Country Link
US (1) US20220363673A1 (https=)
EP (1) EP3990452A1 (https=)
JP (1) JP7498199B2 (https=)
CA (1) CA3144848C (https=)
WO (1) WO2020261144A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3240990A1 (en) 2021-12-01 2023-06-08 Pfizer Inc. 3-phenyl-1-benzothiophene-2-carboxylic acid derivatives as branched-chain alpha keto acid dehydrogenase kinase inhibitors for the treatment of diabetes, kidney diseases, nash and heart failure
CN116574084A (zh) * 2023-04-17 2023-08-11 华南理工大学 一种噻吩衍生物及其合成方法与应用

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