JP2021522231A - チオエーテル環状ペプチドアミリン受容体調節因子 - Google Patents
チオエーテル環状ペプチドアミリン受容体調節因子 Download PDFInfo
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/705—Receptors; Cell surface antigens; Cell surface determinants
- C07K14/72—Receptors; Cell surface antigens; Cell surface determinants for hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/26—Glucagons
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Immunology (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Gastroenterology & Hepatology (AREA)
- Animal Behavior & Ethology (AREA)
- Endocrinology (AREA)
- Veterinary Medicine (AREA)
- Zoology (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Cell Biology (AREA)
- Molecular Biology (AREA)
- Toxicology (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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US201862662492P | 2018-04-25 | 2018-04-25 | |
US62/662,492 | 2018-04-25 | ||
PCT/IB2019/053194 WO2019207427A2 (fr) | 2018-04-25 | 2019-04-17 | Modulateurs du récepteur de l'amyline de peptide cyclique thioéther |
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JP2021522231A true JP2021522231A (ja) | 2021-08-30 |
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JP2020558904A Pending JP2021522231A (ja) | 2018-04-25 | 2019-04-17 | チオエーテル環状ペプチドアミリン受容体調節因子 |
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EP (1) | EP3784265A4 (fr) |
JP (1) | JP2021522231A (fr) |
CN (1) | CN112074289A (fr) |
CA (1) | CA3097812A1 (fr) |
WO (1) | WO2019207427A2 (fr) |
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AU2022210988B9 (en) | 2021-01-20 | 2024-02-22 | Viking Therapeutics, Inc. | Compositions and methods for the treatment of metabolic and liver disorders |
CN114057862A (zh) * | 2021-12-14 | 2022-02-18 | 安徽省国平药业有限公司 | 一种glp-1(1-37)多肽的合成方法 |
Citations (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2001526656A (ja) * | 1997-05-06 | 2001-12-18 | アミリン・ファーマシューティカルズ,インコーポレイテッド | アミリンまたはアミリン・アゴニストを用いる胃炎を予防する方法 |
JP2009530250A (ja) * | 2006-03-15 | 2009-08-27 | ノボ・ノルデイスク・エー/エス | アミリン誘導体 |
JP2014516049A (ja) * | 2011-05-25 | 2014-07-07 | アミリン・ファーマシューティカルズ,リミテッド・ライアビリティ・カンパニー | アミリンペプチドおよび誘導体ならびにそれらの使用 |
JP2016531110A (ja) * | 2013-07-25 | 2016-10-06 | ノバルティス アーゲー | 心不全治療のためのジスルフィド環状ポリペプチド |
WO2017075505A2 (fr) * | 2015-10-28 | 2017-05-04 | Tufts University | Nouveaux polypeptides présentant une meilleure stabilité et procédés de préparation et d'utilisation associés |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7399744B2 (en) * | 2004-03-04 | 2008-07-15 | Amylin Pharmaceuticals, Inc. | Methods for affecting body composition |
EP2036923A1 (fr) * | 2007-09-11 | 2009-03-18 | Novo Nordisk A/S | Dérivés d'amyline améliorés |
CA2764108A1 (fr) * | 2009-06-08 | 2010-12-16 | Amunix Operating Inc. | Polypeptides de regulation du glucose et leurs procedes de production et d'utilisation |
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- 2019-04-17 EP EP19791705.7A patent/EP3784265A4/fr not_active Withdrawn
- 2019-04-17 JP JP2020558904A patent/JP2021522231A/ja active Pending
- 2019-04-17 CN CN201980027903.XA patent/CN112074289A/zh active Pending
- 2019-04-17 WO PCT/IB2019/053194 patent/WO2019207427A2/fr unknown
- 2019-04-17 CA CA3097812A patent/CA3097812A1/fr active Pending
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EP3784265A2 (fr) | 2021-03-03 |
EP3784265A4 (fr) | 2022-06-22 |
WO2019207427A3 (fr) | 2020-01-02 |
CN112074289A (zh) | 2020-12-11 |
WO2019207427A2 (fr) | 2019-10-31 |
CA3097812A1 (fr) | 2019-10-31 |
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