JP2021513965A5 - - Google Patents

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Publication number
JP2021513965A5
JP2021513965A5 JP2020543314A JP2020543314A JP2021513965A5 JP 2021513965 A5 JP2021513965 A5 JP 2021513965A5 JP 2020543314 A JP2020543314 A JP 2020543314A JP 2020543314 A JP2020543314 A JP 2020543314A JP 2021513965 A5 JP2021513965 A5 JP 2021513965A5
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Japan
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cancer
composition according
compound
approximately
disease
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JP2020543314A
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English (en)
Japanese (ja)
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JP7417527B2 (ja
JP2021513965A (ja
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Priority claimed from PCT/US2019/018009 external-priority patent/WO2019161054A1/en
Publication of JP2021513965A publication Critical patent/JP2021513965A/ja
Publication of JP2021513965A5 publication Critical patent/JP2021513965A5/ja
Priority to JP2023177591A priority Critical patent/JP2023171662A/ja
Application granted granted Critical
Publication of JP7417527B2 publication Critical patent/JP7417527B2/ja
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JP2020543314A 2018-02-16 2019-02-14 アゾロピリミジン化合物による投薬 Active JP7417527B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023177591A JP2023171662A (ja) 2018-02-16 2023-10-13 アゾロピリミジン化合物による投薬

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862710394P 2018-02-16 2018-02-16
US62/710,394 2018-02-16
PCT/US2019/018009 WO2019161054A1 (en) 2018-02-16 2019-02-14 Dosing with an azolopyrimidine compound

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023177591A Division JP2023171662A (ja) 2018-02-16 2023-10-13 アゾロピリミジン化合物による投薬

Publications (3)

Publication Number Publication Date
JP2021513965A JP2021513965A (ja) 2021-06-03
JP2021513965A5 true JP2021513965A5 (https=) 2022-02-21
JP7417527B2 JP7417527B2 (ja) 2024-01-18

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ID=67619607

Family Applications (2)

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JP2020543314A Active JP7417527B2 (ja) 2018-02-16 2019-02-14 アゾロピリミジン化合物による投薬
JP2023177591A Pending JP2023171662A (ja) 2018-02-16 2023-10-13 アゾロピリミジン化合物による投薬

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JP2023177591A Pending JP2023171662A (ja) 2018-02-16 2023-10-13 アゾロピリミジン化合物による投薬

Country Status (9)

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US (2) US11478479B2 (https=)
EP (1) EP3755333A4 (https=)
JP (2) JP7417527B2 (https=)
KR (1) KR102823186B1 (https=)
CN (1) CN111818923A (https=)
AU (1) AU2019222747B2 (https=)
CA (1) CA3090922A1 (https=)
TW (1) TWI879727B (https=)
WO (1) WO2019161054A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3090922A1 (en) 2018-02-16 2019-08-22 Arcus Biosciences, Inc. Dosing with an azolopyrimidine compound
EP3823614A4 (en) 2018-07-18 2022-03-30 Arcus Biosciences, Inc. SOLID FORMS OF AN AZOLOPYRIMIDINE COMPOUND
CN113795267A (zh) 2019-03-12 2021-12-14 艾库斯生物科学有限公司 致癌基因驱动的癌症的治疗
WO2020205527A1 (en) 2019-03-29 2020-10-08 Arcus Biosciences, Inc. Treatment of cancer utilizing an identified adenosine fingerprint
CN113121502A (zh) * 2019-12-31 2021-07-16 山东铂源生物医药有限公司 一种杂芳烃类化合物、中间体、组合物及应用
KR102646627B1 (ko) * 2021-03-24 2024-03-13 주식회사 스탠다임 아데노신 a2a 수용체 및 아데노신 a2b 수용체의 이중 길항제, 및 이의 용도
WO2024097736A1 (en) * 2022-11-02 2024-05-10 Arcus Biosciences, Inc. Processes for preparing azolopyrimidine compounds

Family Cites Families (35)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI330183B (https=) 2001-10-22 2010-09-11 Eisai R&D Man Co Ltd
CA2551944A1 (en) 2003-12-15 2005-06-30 Almirall Prodesfarma Ag 2, 6 bisheteroaryl-4-aminopyrimidines as adenosine receptor antagonists
TWI380996B (zh) 2004-09-17 2013-01-01 Hoffmann La Roche 抗ox40l抗體
PT2343320T (pt) 2005-03-25 2018-01-23 Gitr Inc Anticorpos anti-gitr e as suas utilizações
PT1907424E (pt) 2005-07-01 2015-10-09 Squibb & Sons Llc Anticorpos monoclonais humanos para o ligando 1 de morte programada (pd-l1)
EP1987839A1 (en) 2007-04-30 2008-11-05 I.N.S.E.R.M. Institut National de la Sante et de la Recherche Medicale Cytotoxic anti-LAG-3 monoclonal antibody and its use in the treatment or prevention of organ transplant rejection and autoimmune disease
US8591886B2 (en) 2007-07-12 2013-11-26 Gitr, Inc. Combination therapies employing GITR binding molecules
EP2044949A1 (en) 2007-10-05 2009-04-08 Immutep Use of recombinant lag-3 or the derivatives thereof for eliciting monocyte immune response
AR072999A1 (es) 2008-08-11 2010-10-06 Medarex Inc Anticuerpos humanos que se unen al gen 3 de activacion linfocitaria (lag-3) y los usos de estos
EP3255060A1 (en) 2008-12-09 2017-12-13 F. Hoffmann-La Roche AG Anti-pd-l1 antibodies and their use to enhance t-cell function
KR101790802B1 (ko) 2009-09-03 2017-10-27 머크 샤프 앤드 돔 코포레이션 항-gitr 항체
ES2722300T3 (es) 2009-12-10 2019-08-09 Hoffmann La Roche Anticuerpos que se unen preferentemente al dominio extracelular 4 de CSF1R y su uso
US9169323B2 (en) 2010-03-05 2015-10-27 Hoffmann-La Roche Inc. Antibodies against human CSF-1R
JP5989547B2 (ja) 2010-03-05 2016-09-07 エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト ヒトcsf−1rに対する抗体及びその使用
ES2365960B1 (es) * 2010-03-31 2012-06-04 Palobiofarma, S.L Nuevos antagonistas de los receptores de adenosina.
HRP20190047T1 (hr) 2010-05-04 2019-02-22 Five Prime Therapeutics, Inc. Protutijela koja se vežu na csf1r
MX337040B (es) 2010-09-09 2016-02-09 Pfizer Moleculas de union a 4-1bb.
DE102011008352A1 (de) 2011-01-12 2012-07-12 Merck Patent Gmbh 5-([1,2,3]Triazol-4-yl)-7H-pyrrolo-[2,3-d]pyrimidinderivate
JP6072771B2 (ja) 2011-04-20 2017-02-01 メディミューン,エルエルシー B7−h1およびpd−1に結合する抗体およびその他の分子
KR101764096B1 (ko) 2011-11-28 2017-08-02 메르크 파텐트 게엠베하 항-pd-l1 항체 및 그의 용도
RU2658603C2 (ru) 2011-12-15 2018-06-21 Ф.Хоффманн-Ля Рош Аг Антитела против человеческого csf-1r и их применения
KR20140127855A (ko) 2012-02-06 2014-11-04 제넨테크, 인크. Csf1r 억제제를 사용하는 조성물 및 방법
AR090263A1 (es) 2012-03-08 2014-10-29 Hoffmann La Roche Terapia combinada de anticuerpos contra el csf-1r humano y las utilizaciones de la misma
RU2670743C9 (ru) 2012-05-11 2018-12-19 Файв Прайм Терапьютикс, Инк. Способы лечения состояний антителами, которые связывают рецептор колониестимулирующего фактора 1 (csf1r)
UY34887A (es) 2012-07-02 2013-12-31 Bristol Myers Squibb Company Una Corporacion Del Estado De Delaware Optimización de anticuerpos que se fijan al gen de activación de linfocitos 3 (lag-3) y sus usos
CN107759690A (zh) 2012-08-31 2018-03-06 戊瑞治疗有限公司 用结合群落刺激因子1受体(csf1r)的抗体治疗病状的方法
BR112017021386A2 (pt) * 2015-04-08 2018-07-03 Lewis And Clark Pharmaceuticals, Inc. carbamatos de alquinila com xantina substituída/carbamatos reversos como antagonistas de a2b.
MX373318B (es) * 2015-08-11 2020-05-21 Novartis Ag 5-bromo-2,6-di-(1h-pirazol-1-il) pirimidin-4-amina-para su uso en el tratamiento del cáncer.
HUE064141T2 (hu) * 2017-01-20 2024-02-28 Arcus Biosciences Inc Azolopirimidin rákkal összefüggõ rendellenességek kezelésére
US20200055883A1 (en) 2017-02-17 2020-02-20 Eisai R&D Management Co., Ltd. Cyclic di-nucleotides derivative for the treatment of cancer
EP3601259B1 (en) 2017-03-30 2022-02-23 F. Hoffmann-La Roche AG Isoquinolines as inhibitors of hpk1
JP6453507B2 (ja) 2017-03-30 2019-01-16 アムジエン・インコーポレーテツド Mcl−1タンパク質を阻害する化合物
AR111307A1 (es) 2017-03-30 2019-06-26 Takeda Pharmaceuticals Co Derivados de 1’,2’-dihidroespiro[ciclohexan-1,3’-indol] o 1’,2’-dihidroespiro[ciclohexan-1,3’-pirrolo[3,2-b]piridina] como inhibidores de hexakisfosfato quinasa
EP3642240A1 (en) * 2017-06-22 2020-04-29 Novartis AG Antibody molecules to cd73 and uses thereof
CA3090922A1 (en) 2018-02-16 2019-08-22 Arcus Biosciences, Inc. Dosing with an azolopyrimidine compound

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