JP2019509253A5 - - Google Patents

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Publication number
JP2019509253A5
JP2019509253A5 JP2018532746A JP2018532746A JP2019509253A5 JP 2019509253 A5 JP2019509253 A5 JP 2019509253A5 JP 2018532746 A JP2018532746 A JP 2018532746A JP 2018532746 A JP2018532746 A JP 2018532746A JP 2019509253 A5 JP2019509253 A5 JP 2019509253A5
Authority
JP
Japan
Prior art keywords
phosphate
alaninyl
benzoxy
gemcitabine
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2018532746A
Other languages
English (en)
Japanese (ja)
Other versions
JP6898329B2 (ja
JP2019509253A (ja
Filing date
Publication date
Priority claimed from PCT/GB2015/054158 external-priority patent/WO2017109444A1/en
Priority claimed from GBGB1609770.1A external-priority patent/GB201609770D0/en
Application filed filed Critical
Priority claimed from PCT/GB2016/054018 external-priority patent/WO2017109486A1/en
Publication of JP2019509253A publication Critical patent/JP2019509253A/ja
Publication of JP2019509253A5 publication Critical patent/JP2019509253A5/ja
Application granted granted Critical
Publication of JP6898329B2 publication Critical patent/JP6898329B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2018532746A 2015-12-23 2016-12-21 併用療法 Expired - Fee Related JP6898329B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GBPCT/GB2015/054158 2015-12-23
PCT/GB2015/054158 WO2017109444A1 (en) 2015-12-23 2015-12-23 Combination therapy
GB1609770.1 2016-06-03
GBGB1609770.1A GB201609770D0 (en) 2016-06-03 2016-06-03 Combination therapy
PCT/GB2016/054018 WO2017109486A1 (en) 2015-12-23 2016-12-21 Combination therapy

Publications (3)

Publication Number Publication Date
JP2019509253A JP2019509253A (ja) 2019-04-04
JP2019509253A5 true JP2019509253A5 (https=) 2020-01-09
JP6898329B2 JP6898329B2 (ja) 2021-07-07

Family

ID=57681677

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2018532746A Expired - Fee Related JP6898329B2 (ja) 2015-12-23 2016-12-21 併用療法

Country Status (29)

Country Link
US (2) US20190022117A1 (https=)
EP (2) EP3738595A1 (https=)
JP (1) JP6898329B2 (https=)
KR (1) KR20180096698A (https=)
CN (1) CN108697725A (https=)
AU (1) AU2016375861B2 (https=)
CA (1) CA3008749C (https=)
CY (1) CY1122835T1 (https=)
DK (1) DK3393478T3 (https=)
EA (1) EA037459B1 (https=)
ES (1) ES2778933T3 (https=)
HR (1) HRP20200423T1 (https=)
HU (1) HUE050290T2 (https=)
IL (1) IL260076A (https=)
LT (1) LT3393478T (https=)
MA (1) MA51576A (https=)
MD (1) MD3393478T2 (https=)
ME (1) ME03677B (https=)
MX (1) MX383988B (https=)
MY (1) MY194629A (https=)
PH (1) PH12018501339A1 (https=)
PL (1) PL3393478T3 (https=)
PT (1) PT3393478T (https=)
RS (1) RS60211B1 (https=)
SG (1) SG11201805184TA (https=)
SI (1) SI3393478T1 (https=)
SM (1) SMT202000154T1 (https=)
WO (1) WO2017109486A1 (https=)
ZA (1) ZA201804155B (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG11201503750YA (en) 2012-11-16 2015-06-29 Univ Cardiff Process for preparing nucleoside prodrugs
HRP20230584T1 (hr) 2014-06-25 2023-09-15 NuCana plc Prolijekovi gemcitabina
JP6855248B2 (ja) 2014-06-25 2021-04-07 ヌカナ ピーエルシー ゲムシタビン−プロドラッグを含む製剤
GB201417644D0 (en) 2014-10-06 2014-11-19 Nucana Biomed Ltd Method of separating phosphate diastereoisomers
PH12018500691B1 (en) 2015-10-05 2022-08-10 NuCana plc Combination therapy
HRP20211812T1 (hr) 2015-12-11 2022-03-04 NuCana plc Dijastereoselektivna sinteza derivata fosfata i prolijeka gemcitabina nuc-1031
GB201522771D0 (en) 2015-12-23 2016-02-03 Nucana Biomed Ltd Crystalline form of a phosphate derivative
GB201709471D0 (en) 2017-06-14 2017-07-26 Nucana Biomed Ltd Diastereoselective synthesis of hosphate derivatives

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0317009D0 (en) * 2003-07-21 2003-08-27 Univ Cardiff Chemical compounds
TW200916094A (en) * 2007-06-27 2009-04-16 Poniard Pharmaceuticals Inc Stabilized picoplatin dosage form
SG11201501147WA (en) * 2012-08-13 2015-04-29 Regulon Inc Methods for treatment of cancer using lipoplatin
CN104968353B (zh) * 2012-11-13 2017-12-22 博研医药开发股份有限公司 吉西他滨前药及其用途
EP3415149A1 (en) * 2015-05-14 2018-12-19 NuCana plc Cancer treatments
PH12018500691B1 (en) * 2015-10-05 2022-08-10 NuCana plc Combination therapy

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