JP2016521277A5 - - Google Patents

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Publication number
JP2016521277A5
JP2016521277A5 JP2016511017A JP2016511017A JP2016521277A5 JP 2016521277 A5 JP2016521277 A5 JP 2016521277A5 JP 2016511017 A JP2016511017 A JP 2016511017A JP 2016511017 A JP2016511017 A JP 2016511017A JP 2016521277 A5 JP2016521277 A5 JP 2016521277A5
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JP
Japan
Prior art keywords
alkyl
group
formula
bond
independently
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JP2016511017A
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English (en)
Japanese (ja)
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JP6353032B2 (ja
JP2016521277A (ja
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Priority claimed from PCT/EP2014/058462 external-priority patent/WO2014177469A1/en
Publication of JP2016521277A publication Critical patent/JP2016521277A/ja
Publication of JP2016521277A5 publication Critical patent/JP2016521277A5/ja
Application granted granted Critical
Publication of JP6353032B2 publication Critical patent/JP6353032B2/ja
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JP2016511017A 2013-04-30 2014-04-25 ジアミノピラジン化合物、前記化合物を含有する医薬、その使用、およびその調製方法 Active JP6353032B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP13165963 2013-04-30
EP13165963.3 2013-04-30
PCT/EP2014/058462 WO2014177469A1 (en) 2013-04-30 2014-04-25 Diaminopyrazine compounds, medicaments containing said compounds, use thereof and processes for the preparation thereof

Publications (3)

Publication Number Publication Date
JP2016521277A JP2016521277A (ja) 2016-07-21
JP2016521277A5 true JP2016521277A5 (https=) 2017-08-24
JP6353032B2 JP6353032B2 (ja) 2018-07-04

Family

ID=48227015

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2016511017A Active JP6353032B2 (ja) 2013-04-30 2014-04-25 ジアミノピラジン化合物、前記化合物を含有する医薬、その使用、およびその調製方法

Country Status (4)

Country Link
US (1) US9018215B2 (https=)
EP (1) EP2991981B1 (https=)
JP (1) JP6353032B2 (https=)
WO (1) WO2014177469A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016126726A1 (en) 2015-02-02 2016-08-11 Forma Therapeutics, Inc. Bicyclic [4,6,0] hydroxamic acids as hdac6 inhibitors
SG11201708622UA (en) 2015-02-02 2017-11-29 Forma Therapeutics Inc 3-aryl-4-amido-bicyclic [4,5,0] hydroxamic acids as hdac inhibitors
EP3472131B1 (en) 2016-06-17 2020-02-19 Forma Therapeutics, Inc. 2-spiro-5- and 6-hydroxamic acid indanes as hdac inhibitors
GB201610854D0 (en) 2016-06-21 2016-08-03 Entpr Therapeutics Ltd Compounds
GB201619694D0 (en) 2016-11-22 2017-01-04 Entpr Therapeutics Ltd Compounds
GB201717051D0 (en) 2017-10-17 2017-11-29 Enterprise Therapeutics Ltd Compounds
GB201808093D0 (en) 2018-05-18 2018-07-04 Enterprise Therapeutics Ltd Compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2432529T3 (es) * 2003-08-18 2013-12-04 Parion Sciences, Inc. Bloqueadores del canal de sodio de pirazinoilguanidina rematada
DE602008005140D1 (de) * 2007-05-07 2011-04-07 Novartis Ag Organische verbindungen
MX2010006421A (es) * 2007-12-10 2010-06-25 Novartis Ag Compuestos organicos.
US8859559B2 (en) * 2011-12-20 2014-10-14 Boehringer Ingelheim International Gmbh Substituted pyrazines and their use in the treatment of disease
EP2861577B1 (en) * 2012-05-25 2017-01-04 Boehringer Ingelheim International GmbH Tertiary amines, medicaments containing said amines, use thereof and processes for the preparation thereof

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