JP2014520848A5 - - Google Patents
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- Publication number
- JP2014520848A5 JP2014520848A5 JP2014520224A JP2014520224A JP2014520848A5 JP 2014520848 A5 JP2014520848 A5 JP 2014520848A5 JP 2014520224 A JP2014520224 A JP 2014520224A JP 2014520224 A JP2014520224 A JP 2014520224A JP 2014520848 A5 JP2014520848 A5 JP 2014520848A5
- Authority
- JP
- Japan
- Prior art keywords
- fluticasone propionate
- solvent
- solution
- slurry
- type
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 229960000289 fluticasone propionate Drugs 0.000 claims 21
- WMWTYOKRWGGJOA-CENSZEJFSA-N fluticasone propionate Chemical compound C1([C@@H](F)C2)=CC(=O)C=C[C@]1(C)[C@]1(F)[C@@H]2[C@@H]2C[C@@H](C)[C@@](C(=O)SCF)(OC(=O)CC)[C@@]2(C)C[C@@H]1O WMWTYOKRWGGJOA-CENSZEJFSA-N 0.000 claims 21
- 239000002904 solvent Substances 0.000 claims 17
- 238000000034 method Methods 0.000 claims 16
- 239000002002 slurry Substances 0.000 claims 12
- 239000013078 crystal Substances 0.000 claims 6
- 239000002245 particle Substances 0.000 claims 5
- CSCPPACGZOOCGX-UHFFFAOYSA-N Acetone Chemical compound CC(C)=O CSCPPACGZOOCGX-UHFFFAOYSA-N 0.000 claims 4
- 238000001914 filtration Methods 0.000 claims 4
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 claims 3
- 238000005054 agglomeration Methods 0.000 claims 1
- 230000002776 aggregation Effects 0.000 claims 1
- 238000004519 manufacturing process Methods 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161505612P | 2011-07-08 | 2011-07-08 | |
| US61/505,612 | 2011-07-08 | ||
| PCT/US2012/045660 WO2013009591A1 (en) | 2011-07-08 | 2012-07-06 | Process for the preparation of fluticasone propionate form 1 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016164301A Division JP2017031161A (ja) | 2011-07-08 | 2016-08-25 | １型プロピオン酸フルチカゾンの調製のための方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2014520848A JP2014520848A (ja) | 2014-08-25 |
| JP2014520848A5 true JP2014520848A5 (enExample) | 2014-10-09 |
Family
ID=47506422
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014520224A Pending JP2014520848A (ja) | 2011-07-08 | 2012-07-06 | １型プロピオン酸フルチカゾンの調製のための方法 |
| JP2016164301A Pending JP2017031161A (ja) | 2011-07-08 | 2016-08-25 | １型プロピオン酸フルチカゾンの調製のための方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016164301A Pending JP2017031161A (ja) | 2011-07-08 | 2016-08-25 | １型プロピオン酸フルチカゾンの調製のための方法 |
Country Status (10)
| Country | Link |
|---|---|
| US (2) | US10370402B2 (enExample) |
| EP (1) | EP2729480A4 (enExample) |
| JP (2) | JP2014520848A (enExample) |
| KR (3) | KR20140048237A (enExample) |
| CN (2) | CN103649104A (enExample) |
| AU (1) | AU2012282936B2 (enExample) |
| CA (1) | CA2840401C (enExample) |
| MX (2) | MX376564B (enExample) |
| WO (1) | WO2013009591A1 (enExample) |
| ZA (1) | ZA201309531B (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2013009591A1 (en) * | 2011-07-08 | 2013-01-17 | Pfizer Limited | Process for the preparation of fluticasone propionate form 1 |
| PL3517541T3 (pl) | 2012-05-08 | 2020-12-28 | Nicox Ophthalmics, Inc. | Postać polimorficzna propionianu flutykazonu |
| WO2015118474A1 (en) * | 2014-02-07 | 2015-08-13 | Mylan Laboratories Ltd. | Process for the purification of fluticasone propionate using a ketone solvent and water as anti-solvent |
| CN111662353A (zh) * | 2019-03-05 | 2020-09-15 | 上海谷森医药有限公司 | 一种糠酸氟替卡松晶型1的制备方法 |
| CA3136619A1 (en) * | 2019-04-10 | 2020-10-15 | Eupraxia Pharmaceuticals Inc. | Process for making drug crystals of desired size distribution and morphology |
| CN110759960B (zh) * | 2019-10-30 | 2021-03-23 | 山东赛托生物科技股份有限公司 | 一种丙酸氟替卡松的精制方法 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CY1291A (en) | 1980-02-15 | 1985-10-18 | Glaxo Group Ltd | Androstane 17 beta carbothioates |
| GB9001635D0 (en) * | 1990-01-24 | 1990-03-21 | Ganderton David | Aerosol carriers |
| SE9501384D0 (sv) * | 1995-04-13 | 1995-04-13 | Astra Ab | Process for the preparation of respirable particles |
| GB9622173D0 (en) * | 1996-10-24 | 1996-12-18 | Glaxo Group Ltd | Particulate Products |
| GB9828721D0 (en) * | 1998-12-24 | 1999-02-17 | Glaxo Group Ltd | Novel apparatus and process |
| GB9925934D0 (en) * | 1999-11-03 | 1999-12-29 | Glaxo Group Ltd | Novel apparatus and process |
| GB0015981D0 (en) * | 2000-06-29 | 2000-08-23 | Glaxo Group Ltd | Novel process for preparing crystalline particles |
| GB0125604D0 (en) * | 2001-10-25 | 2001-12-19 | Glaxo Group Ltd | Novel process |
| GB0201400D0 (en) * | 2002-01-22 | 2002-03-13 | Glaxo Group Ltd | Novel apparatus and process |
| GB0202564D0 (en) * | 2002-02-04 | 2002-03-20 | Glaxo Group Ltd | Process |
| AU2003263575A1 (en) * | 2002-06-20 | 2004-01-06 | Sun Pharmaceutical Industries Limited | Convenient synthesis of s-fluoromethyl 6alpha, 9alpha-difluoro-11beta-hydroxy-16alpha- methyl-17alpha-propionyloxy-3-oxoandrosta-1, 4-diene-17beta-carbothioate |
| GB0315509D0 (en) | 2003-07-02 | 2003-08-06 | Meridica Ltd | Dispensing device |
| US7314516B2 (en) * | 2004-12-29 | 2008-01-01 | Five Star Technologies, Inc. | Hydrodynamic cavitation crystallization device and process |
| WO2013009591A1 (en) * | 2011-07-08 | 2013-01-17 | Pfizer Limited | Process for the preparation of fluticasone propionate form 1 |
-
2012
- 2012-07-06 WO PCT/US2012/045660 patent/WO2013009591A1/en not_active Ceased
- 2012-07-06 CN CN201280034030.3A patent/CN103649104A/zh active Pending
- 2012-07-06 EP EP12811395.8A patent/EP2729480A4/en not_active Ceased
- 2012-07-06 KR KR1020147003035A patent/KR20140048237A/ko not_active Ceased
- 2012-07-06 US US14/131,407 patent/US10370402B2/en not_active Expired - Fee Related
- 2012-07-06 AU AU2012282936A patent/AU2012282936B2/en not_active Ceased
- 2012-07-06 MX MX2014000192A patent/MX376564B/es active IP Right Grant
- 2012-07-06 KR KR1020197026105A patent/KR102163368B1/ko not_active Expired - Fee Related
- 2012-07-06 KR KR1020207028182A patent/KR20200117056A/ko not_active Ceased
- 2012-07-06 JP JP2014520224A patent/JP2014520848A/ja active Pending
- 2012-07-06 CN CN201610951505.5A patent/CN106977575A/zh active Pending
- 2012-07-06 CA CA2840401A patent/CA2840401C/en not_active Expired - Fee Related
-
2013
- 2013-12-18 ZA ZA2013/09531A patent/ZA201309531B/en unknown
-
2014
- 2014-01-07 MX MX2020011330A patent/MX2020011330A/es unknown
-
2016
- 2016-08-25 JP JP2016164301A patent/JP2017031161A/ja active Pending
-
2019
- 2019-07-29 US US16/525,111 patent/US20200024298A1/en not_active Abandoned
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