JP2012504604A5 - - Google Patents

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Publication number
JP2012504604A5
JP2012504604A5 JP2011530048A JP2011530048A JP2012504604A5 JP 2012504604 A5 JP2012504604 A5 JP 2012504604A5 JP 2011530048 A JP2011530048 A JP 2011530048A JP 2011530048 A JP2011530048 A JP 2011530048A JP 2012504604 A5 JP2012504604 A5 JP 2012504604A5
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JP
Japan
Prior art keywords
alkyl
alkenyl
alkynyl
con
heteroaryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2011530048A
Other languages
English (en)
Japanese (ja)
Other versions
JP2012504604A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2009/005407 external-priority patent/WO2010039237A1/en
Publication of JP2012504604A publication Critical patent/JP2012504604A/ja
Publication of JP2012504604A5 publication Critical patent/JP2012504604A5/ja
Pending legal-status Critical Current

Links

JP2011530048A 2008-10-01 2009-10-01 炎症および免疫関連使用のための化合物 Pending JP2012504604A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US19483108P 2008-10-01 2008-10-01
US61/194,831 2008-10-01
PCT/US2009/005407 WO2010039237A1 (en) 2008-10-01 2009-10-01 Compounds for inflammation and immune-related uses

Publications (2)

Publication Number Publication Date
JP2012504604A JP2012504604A (ja) 2012-02-23
JP2012504604A5 true JP2012504604A5 (OSRAM) 2012-11-22

Family

ID=41263687

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2011530048A Pending JP2012504604A (ja) 2008-10-01 2009-10-01 炎症および免疫関連使用のための化合物

Country Status (7)

Country Link
US (3) US8314130B2 (OSRAM)
EP (1) EP2350064A1 (OSRAM)
JP (1) JP2012504604A (OSRAM)
AU (1) AU2009300317A1 (OSRAM)
CA (1) CA2739322A1 (OSRAM)
TW (1) TW201026693A (OSRAM)
WO (1) WO2010039237A1 (OSRAM)

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Publication number Priority date Publication date Assignee Title
EP2382212B1 (en) 2009-01-23 2014-07-16 Bristol-Myers Squibb Company Substituted oxadiazole derivatives as s1p agonists in the treatment of autoimmune and inflammatory diseases
CN102361869A (zh) 2009-01-23 2012-02-22 百时美施贵宝公司 在治疗自身免疫性疾病和炎性疾病中作为s1p激动剂的取代的噁二唑衍生物
JP2012515789A (ja) 2009-01-23 2012-07-12 ブリストル−マイヤーズ スクイブ カンパニー スフィンゴシン−１−リン酸アゴニストとしてのピラゾール−１，２，４−オキサジアゾール誘導体
US8993612B2 (en) 2009-10-08 2015-03-31 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel and methods for treatment of non-small cell lung cancer
US8377970B2 (en) 2009-10-08 2013-02-19 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel
US10703722B2 (en) 2010-04-27 2020-07-07 Calcimedica, Inc. Compounds that modulate intracellular calcium
WO2011139489A2 (en) 2010-04-27 2011-11-10 Calcimedica Inc. Compounds that modulate intracellular calcium
CA2797533A1 (en) 2010-04-27 2011-11-10 Calcimedica, Inc. Compounds that modulate intracellular calcium
WO2012027710A2 (en) 2010-08-27 2012-03-01 Calcimedica Inc. Compounds that modulate intracellular calcium
US8592456B2 (en) * 2011-01-28 2013-11-26 4Sc Discovery Gmbh IL17 and IFN-gamma inhibition for the treatment of autoimmune inflammation
JP5985611B2 (ja) * 2011-05-03 2016-09-06 シンタ ファーマシューティカルズ コーポレーション 炎症および免疫関連用途のための化合物
WO2012170931A2 (en) 2011-06-10 2012-12-13 Calcimedica, Inc. Compounds that modulate intracellular calcium
WO2013059677A1 (en) 2011-10-19 2013-04-25 Calcimedica, Inc. Compounds that modulate intracellular calcium
US9512116B2 (en) 2012-10-12 2016-12-06 Calcimedica, Inc. Compounds that modulate intracellular calcium
EP3261641B1 (en) 2015-02-27 2023-07-12 Calcimedica, Inc. Pancreatitis treatment
CA2995094A1 (en) 2015-08-07 2017-02-16 Calcimedica, Inc. Use of crac channel inhibitors for the treatment of stroke and traumatic brain injury
WO2019054430A1 (ja) * 2017-09-14 2019-03-21 第一三共株式会社 芳香族複素環を有するアミド化合物
EP3849552A1 (en) 2018-09-14 2021-07-21 Rhizen Pharmaceuticals AG Compositions comprising a crac inhibitor and a corticosteroid and methods of use thereof
MX2022008627A (es) 2020-01-13 2022-11-08 Verge Analytics Inc Pirazolo-pirimidinas sustituidas y usos de las mismas.
CN118084860A (zh) * 2024-02-06 2024-05-28 中国药科大学 芳酰胺类化合物及其药物组合物和应用

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