JP2011510974A - HMG−CoA還元酵素阻害剤の調節放出製剤 - Google Patents

HMG−CoA還元酵素阻害剤の調節放出製剤 Download PDF

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Publication number
JP2011510974A
JP2011510974A JP2010544844A JP2010544844A JP2011510974A JP 2011510974 A JP2011510974 A JP 2011510974A JP 2010544844 A JP2010544844 A JP 2010544844A JP 2010544844 A JP2010544844 A JP 2010544844A JP 2011510974 A JP2011510974 A JP 2011510974A
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JP
Japan
Prior art keywords
rosuvastatin
pharmaceutically acceptable
release
formulation
release pharmaceutical
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Pending
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JP2010544844A
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English (en)
Japanese (ja)
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JP2011510974A5 (https=
Inventor
クルカルニ,シータル
ダス,スリルパ
デシュムク,アシシュ,アショクラオ
ダラル,サティッシュ,クマール
クルカルニ,シリシュクマール
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Lupin Ltd
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Lupin Ltd
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Publication of JP2011510974A publication Critical patent/JP2011510974A/ja
Publication of JP2011510974A5 publication Critical patent/JP2011510974A5/ja
Pending legal-status Critical Current

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Diabetes (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2010544844A 2008-01-30 2009-01-30 HMG−CoA還元酵素阻害剤の調節放出製剤 Pending JP2011510974A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN145KO2008 2008-01-30
PCT/IN2009/000069 WO2009095934A1 (en) 2008-01-30 2009-01-30 Modified release formulations of hmg coa reductase inhibitors

Publications (2)

Publication Number Publication Date
JP2011510974A true JP2011510974A (ja) 2011-04-07
JP2011510974A5 JP2011510974A5 (https=) 2012-03-15

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ID=40638221

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010544844A Pending JP2011510974A (ja) 2008-01-30 2009-01-30 HMG−CoA還元酵素阻害剤の調節放出製剤

Country Status (8)

Country Link
US (1) US20110003837A1 (https=)
EP (1) EP2285353A1 (https=)
JP (1) JP2011510974A (https=)
AU (1) AU2009208610A1 (https=)
BR (1) BRPI0906728A2 (https=)
MX (1) MX2010008466A (https=)
WO (1) WO2009095934A1 (https=)
ZA (1) ZA201006157B (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11590161B2 (en) * 2018-08-13 2023-02-28 Viscera Labs, Inc. Therapeutic composition and methods

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2007510714A (ja) * 2003-11-04 2007-04-26 アスファーマ・リミテッド 担体輸送スタチンの医薬製剤およびそれらの使用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6642268B2 (en) * 1994-09-13 2003-11-04 G.D. Searle & Co. Combination therapy employing ileal bile acid transport inhibiting benzothipines and HMG Co-A reductase inhibitors
IL149422A0 (en) * 1999-11-03 2002-11-10 Smith Howard J & Ass Pty Ltd Oral pharmaceutical compositions for liver therapy
GB0001621D0 (en) * 2000-01-26 2000-03-15 Astrazeneca Ab Pharmaceutical compositions
DE10209979A1 (de) * 2002-03-07 2003-09-25 Ratiopharm Gmbh Arzneimittel mit Cholesterolspiegel-senkenden Wirkstoffen mit zeitverzögerter Wirkstofffreisetzung
GB0217306D0 (en) * 2002-07-25 2002-09-04 Novartis Ag Compositions comprising organic compounds
US20050096391A1 (en) * 2003-10-10 2005-05-05 Per Holm Compositions comprising fenofibrate and rosuvastatin
US20050147620A1 (en) * 2004-01-05 2005-07-07 Karl Bozicevic Cinnamon formulation for reducing cholesterol and/or glucose levels
EP1968593B1 (en) * 2005-12-20 2017-08-23 LEK Pharmaceuticals d.d. Pharmaceutical composition comprising (e)-7-[4-(4-fluorophenyl)-6-isopropyl-2-[methyl(methylsulfonyl)amino]pyrimidin-5-yl-(3r,5s)-3,5-dihydroxyhept-6-enoic acid

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2007510714A (ja) * 2003-11-04 2007-04-26 アスファーマ・リミテッド 担体輸送スタチンの医薬製剤およびそれらの使用

Also Published As

Publication number Publication date
MX2010008466A (es) 2010-10-25
US20110003837A1 (en) 2011-01-06
AU2009208610A1 (en) 2009-08-06
BRPI0906728A2 (pt) 2015-07-07
WO2009095934A1 (en) 2009-08-06
EP2285353A1 (en) 2011-02-23
ZA201006157B (en) 2011-05-25

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