JP2010540424A5 - - Google Patents

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Publication number
JP2010540424A5
JP2010540424A5 JP2010525426A JP2010525426A JP2010540424A5 JP 2010540424 A5 JP2010540424 A5 JP 2010540424A5 JP 2010525426 A JP2010525426 A JP 2010525426A JP 2010525426 A JP2010525426 A JP 2010525426A JP 2010540424 A5 JP2010540424 A5 JP 2010540424A5
Authority
JP
Japan
Prior art keywords
alkyl
aryl
hydrogen
compound according
ethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2010525426A
Other languages
English (en)
Japanese (ja)
Other versions
JP2010540424A (ja
Filing date
Publication date
Priority claimed from GBGB0718432.8A external-priority patent/GB0718432D0/en
Application filed filed Critical
Publication of JP2010540424A publication Critical patent/JP2010540424A/ja
Publication of JP2010540424A5 publication Critical patent/JP2010540424A5/ja
Pending legal-status Critical Current

Links

JP2010525426A 2007-09-21 2008-09-19 チエノピリミジン化合物類および組成物 Pending JP2010540424A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0718432.8A GB0718432D0 (en) 2007-09-21 2007-09-21 New chemical compounds
PCT/GB2008/003180 WO2009037468A1 (en) 2007-09-21 2008-09-19 Thienopyrimidine compounds and compositions

Publications (2)

Publication Number Publication Date
JP2010540424A JP2010540424A (ja) 2010-12-24
JP2010540424A5 true JP2010540424A5 (https=) 2011-11-04

Family

ID=38670287

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010525426A Pending JP2010540424A (ja) 2007-09-21 2008-09-19 チエノピリミジン化合物類および組成物

Country Status (5)

Country Link
US (1) US8354415B2 (https=)
EP (1) EP2207780B1 (https=)
JP (1) JP2010540424A (https=)
GB (1) GB0718432D0 (https=)
WO (1) WO2009037468A1 (https=)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2011157168A (ja) 2010-01-29 2011-08-18 Tokyo Kikai Seisakusho Ltd 新聞製作装置
EP2567959B1 (en) 2011-09-12 2014-04-16 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
RU2637925C2 (ru) 2012-01-10 2017-12-08 Ф. Хоффманн-Ля Рош Аг Соединения тиенопиримидина
CN105793267B (zh) * 2013-10-07 2018-02-06 拜耳制药股份公司 环状噻吩并尿嘧啶甲酰胺类及其用途
UY36586A (es) 2015-03-26 2016-10-31 Bayer Pharma AG Heterociclilmetiltienouracilos y uso de los mismos
WO2018013611A1 (en) 2016-07-11 2018-01-18 Corvus Pharmaceuticals, Inc. Anti-cd73 antibodies
WO2018041771A1 (de) 2016-09-02 2018-03-08 Bayer Pharma Aktiengesellschaft (1-methylcyclopropyl)methyl-substituierte thienouracile und ihre verwendung
WO2018054846A1 (de) 2016-09-23 2018-03-29 Bayer Aktiengesellschaft N3-cyclisch substituierte thienouracile und ihre verwendung
CN111629728A (zh) * 2017-08-31 2020-09-04 科尔沃斯制药股份有限公司 用于调节腺苷a2b受体和腺苷a2a受体的化合物和方法
EP3575287A1 (en) * 2018-05-31 2019-12-04 Universiteit Leiden Inhibitors of n-acylphosphatidylethanolamine phospholipase d (nape-pld)
CN119173276A (zh) 2022-04-13 2024-12-20 吉利德科学公司 用于治疗表达Trop-2的癌症的组合疗法
WO2025137640A1 (en) 2023-12-22 2025-06-26 Gilead Sciences, Inc. Azaspiro wrn inhibitors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9915437D0 (en) 1999-07-01 1999-09-01 Cerebrus Ltd Chemical compounds III
KR100960827B1 (ko) * 2001-12-20 2010-06-08 오에스아이 파마슈티컬스, 인코포레이티드 피롤로피리미딘 A₂b 선택성 길항 화합물, 그의 합성방법 및 용도
CA2544193C (en) * 2003-10-31 2012-03-27 Cv Therapeutics, Inc. A2b adenosine receptor antagonists
CA2644996A1 (en) * 2006-03-02 2007-09-13 Cv Therapeutics, Inc. A2a adenosine receptor antagonists

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